Rank |
Compound |
SMILES |
ΔG / kcal M-1 |
pIC50 |
1 |
EDJ-MED-33064c06-2
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC(=O)NCC6(CC6)N |
−14.8
± 0.3
|
10.7
± 0.2
|
2 |
ALP-POS-c3a90b22-7
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CS(=O)(=O)CC6(CC6)C#N |
−14.7
± 0.3
|
10.7
± 0.2
|
3 |
ALP-POS-c3a90b22-12
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC(=O)NCC6COC6 |
−14.5
± 0.2
|
10.6
± 0.2
|
4 |
EDJ-MED-33064c06-8
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC(=O)NCC6(CC6)O |
−14.4
± 0.3
|
10.5
± 0.2
|
5 |
EDJ-MED-33064c06-14
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC(=O)NCC6(CCC6)O |
−14.1
± 0.4
|
10.3
± 0.3
|
6 |
ALP-POS-c3a90b22-6
|
|
CNC(=O)CCN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−14.0
± 0.4
|
10.2
± 0.3
|
7 |
ALP-POS-4483ae88-2
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5S1(=O)=O)Cl |
−14.0
± 0.5
|
10.2
± 0.4
|
8 |
EDJ-MED-4cb9dd84-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC(=O)NCC6CC6 |
−13.8
± 0.3
|
10.1
± 0.2
|
9 |
MAT-POS-c7726e07-6
|
|
CNC(=O)CN1Cc2ccc(cc2[C@@]3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−13.8
± 0.2
|
10.1
± 0.1
|
10 |
MAT-POS-69786b79-3
|
|
CC1(CC1)NC(=O)CN2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−13.7
± 0.2
|
10.0
± 0.1
|
11 |
LUO-POS-8484f2d3-2
|
|
CN(C)CCOc1ccc2cncc(c2c1)N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−13.5
± 0.9
|
9.8
± 0.7
|
12 |
PET-UNK-37c7074c-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6ccon6 |
−13.3
± 0.2
|
9.7
± 0.2
|
13 |
ALP-POS-c3a90b22-2
|
|
CNC(=O)C1(CCC1)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−13.2
± 0.3
|
9.6
± 0.2
|
14 |
EDJ-MED-33064c06-15
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC(=O)NC6(CC6)C#N |
−13.0
± 0.2
|
9.5
± 0.2
|
15 |
ALP-POS-afe0272e-1
|
|
CNC(=O)CN1Cc2cc(c(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl)Cl |
−13.0
± 0.2
|
9.5
± 0.1
|
16 |
EDJ-MED-33064c06-17
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC(=O)NCC6(CC6)C#N |
−12.8
± 0.3
|
9.3
± 0.2
|
17 |
EDJ-MED-b6c6ee2b-1
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cc(cc5)OCCN(C)C)Cl |
−12.6
± 0.4
|
9.2
± 0.3
|
18 |
EDJ-MED-0d144977-2
|
|
Cn1cncc1CN2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−12.6
± 0.5
|
9.2
± 0.3
|
19 |
MAT-POS-38eb6498-3
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cc(cc5)OCCN(C)C)Cl |
−12.6
± 0.4
|
9.1
± 0.3
|
20 |
MAT-POS-e48723dc-2
|
|
CNC(=O)C1(CC1)N2C[C@@]3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−12.5
± 0.3
|
9.1
± 0.2
|
21 |
LUO-POS-e1dab717-18
|
|
CC1(CC2(CN(Cc3c2cc(cc3)Cl)CC(=O)NC)C(=O)N1c4cncc5c4cccc5)C |
−12.5
± 0.4
|
9.1
± 0.3
|
22 |
MAT-POS-b4d6b7fc-6
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4c(ccc5)Cl)Cl |
−12.4
± 0.4
|
9.0
± 0.3
|
23 |
MIK-ENA-7066949b-1
|
|
CN(C)CCOc1ccc2cncc(c2c1)N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−12.2
± 0.9
|
8.9
± 0.7
|
24 |
PET-UNK-14142a25-1
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−12.2
± 0.3
|
8.9
± 0.2
|
25 |
MAT-POS-38eb6498-6
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)C(=O)NC)c5cc(ccc5C1=O)Cl |
−12.1
± 0.5
|
8.8
± 0.3
|
26 |
DAR-DIA-0f7b7cd9-9
|
|
c1ccc2c(c1)cncc2N3CC(=O)C4(C3=O)CCOc5c4cc(cc5)Cl |
−12.1
± 0.4
|
8.8
± 0.3
|
27 |
VLA-UNK-8e615992-5
|
|
CNC(=O)CN1C(C2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl)C(F)F |
−11.9
± 0.3
|
8.7
± 0.2
|
28 |
PET-UNK-aa57768f-2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC#N |
−11.9
± 0.3
|
8.7
± 0.2
|
29 |
EDJ-MED-cc48ee33-5
|
|
Cc1cc(n(n1)C)C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−11.9
± 0.5
|
8.6
± 0.3
|
30 |
PET-UNK-c6bcc80b-4
|
|
CS(=O)(=O)Nc1cc2cncc(c2cc1F)N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−11.6
± 0.9
|
8.4
± 0.7
|
31 |
EDJ-MED-0d144977-5
|
|
Cn1ccnc1CN2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−11.3
± 0.3
|
8.2
± 0.2
|
32 |
PET-UNK-c6bcc80b-6
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cc(c(c4)NS(=O)(=O)C)F)c5cc(ccc5C1=O)Cl |
−11.3
± 0.4
|
8.2
± 0.3
|
33 |
PET-UNK-c6bcc80b-12
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cc(c(c5)NS(=O)(=O)C)F)Cl |
−11.2
± 0.3
|
8.2
± 0.2
|
34 |
VLA-UNK-61877630-5
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(c(cc5C1=O)F)Cl |
−11.2
± 0.3
|
8.2
± 0.2
|
35 |
EDJ-MED-5cd3920d-6
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C(F)(F)F |
−11.2
± 0.8
|
8.1
± 0.6
|
36 |
MAT-POS-38eb6498-2
|
|
CNC(=O)c1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−11.1
± 0.9
|
8.1
± 0.6
|
37 |
MAT-POS-ddfe83c6-6
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cc(cc5)Cl)Cl |
−11.0
± 0.3
|
8.0
± 0.3
|
38 |
JOH-MSK-1f2dff76-1
|
|
CNC(=O)CN1Cc2ccc(cc2[C@@]3(C1)CC(=O)N(C3=O)c4cncc5c4cccc5)Cl |
−10.9
± 0.5
|
8.0
± 0.4
|
39 |
LUO-POS-e1dab717-8
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN(C)C)c6cc(ccc6C2=O)Cl |
−10.9
± 0.7
|
7.9
± 0.5
|
40 |
MAT-POS-50a80394-2
|
|
CCC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−10.9
± 0.9
|
7.9
± 0.7
|
41 |
PET-UNK-6af7266d-3
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nncs6 |
−10.9
± 0.2
|
7.9
± 0.1
|
42 |
ALP-POS-c3a90b22-3
|
|
CNC(=O)C1(COC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−10.8
± 0.4
|
7.9
± 0.3
|
43 |
PET-UNK-aa57768f-9
|
|
C#CCN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−10.8
± 0.3
|
7.9
± 0.2
|
44 |
PET-UNK-94036022-3
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−10.7
± 0.7
|
7.8
± 0.5
|
45 |
MIK-ENA-99706bb8-1
|
|
C[C@H]1CN(C(=O)[C@]12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−10.7
± 0.8
|
7.8
± 0.6
|
46 |
PET-UNK-c6bcc80b-13
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(c(c4)NS(=O)(=O)C)F)c5cc(ccc5C1=O)Cl |
−10.6
± 0.4
|
7.8
± 0.3
|
47 |
MAT-POS-be048f2c-8
|
|
CCCn1c(ccn1)C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−10.6
± 0.5
|
7.7
± 0.4
|
48 |
PET-UNK-aa57768f-8
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC#N |
−10.6
± 0.3
|
7.7
± 0.2
|
49 |
LUO-POS-b4dec3be-1
|
|
CNC(=O)CN1Cc2ccc(cc2[C@@]3(C1)CCN(C3=O)c4cncc5c4cc(cc5)F)Cl |
−10.6
± 0.2
|
7.7
± 0.2
|
50 |
PET-UNK-c6bcc80b-5
|
|
CNC(=O)CN1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cc(c(c5)NS(=O)(=O)C)F)Cl |
−10.6
± 0.3
|
7.7
± 0.2
|
51 |
EDJ-MED-4138fde9-8
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6COC6 |
−10.6
± 0.8
|
7.7
± 0.6
|
52 |
VLA-UNK-8e615992-1
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(cc(c5C1=O)F)Cl |
−10.6
± 0.5
|
7.7
± 0.4
|
53 |
MAT-POS-e48723dc-1
|
|
CNC(=O)C1(CC1)N2C[C@]3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−10.5
± 0.3
|
7.7
± 0.2
|
54 |
EDJ-MED-98c0a822-4
|
|
CNC(=O)C1(COC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−10.5
± 0.4
|
7.7
± 0.3
|
55 |
EDJ-MED-b6c6ee2b-7
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)F)c6cc(ccc6C2=O)Cl |
−10.5
± 0.4
|
7.6
± 0.3
|
56 |
LUO-POS-e1dab717-6
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OC)c6cc(ccc6C2=O)Cl |
−10.5
± 0.4
|
7.6
± 0.3
|
57 |
EDJ-MED-cc48ee33-7
|
|
Cn1c(ccn1)CN2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−10.5
± 0.3
|
7.6
± 0.2
|
58 |
ALP-POS-c3a90b22-9
|
|
CNC(=O)C1(CCOCC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−10.4
± 0.4
|
7.6
± 0.3
|
59 |
PET-UNK-6af7266d-2
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nncs6 |
−10.4
± 0.4
|
7.6
± 0.3
|
60 |
PET-UNK-7e9559de-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)Cc6nncs6 |
−10.3
± 0.4
|
7.5
± 0.3
|
61 |
PET-UNK-6af7266d-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nncs6 |
−10.3
± 0.2
|
7.5
± 0.1
|
62 |
MAT-POS-e75f6e44-19
|
|
CC1(CCC1)CNC(=O)CN2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−10.3
± 0.2
|
7.5
± 0.2
|
63 |
ALP-POS-41e2080f-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CCS(=O)(=O)c5c4cc(cc5)Cl |
−10.3
± 0.5
|
7.5
± 0.3
|
64 |
EDJ-MED-7d88f880-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4ccc(c5)S(=N)(=O)C)c6cc(ccc6C2=O)Cl |
−10.3
± 0.3
|
7.5
± 0.2
|
65 |
EDJ-MED-0d144977-3
|
|
Cn1c(ccn1)CN2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−10.2
± 0.4
|
7.5
± 0.3
|
66 |
EDJ-MED-0d144977-4
|
|
Cn1c(ncn1)CN2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−10.2
± 0.4
|
7.5
± 0.3
|
67 |
EDJ-MED-6b23330e-4
|
|
CC(C)(CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl)O |
−10.2
± 0.3
|
7.5
± 0.2
|
68 |
PET-UNK-7e9559de-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)Cc6nncs6 |
−10.2
± 0.5
|
7.5
± 0.4
|
69 |
MAT-POS-1bed62cf-3
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CC(=O)N(C3=O)c4cncc5c4cccc5)Cl |
−10.2
± 0.5
|
7.5
± 0.4
|
70 |
MAT-POS-e75f6e44-2
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NCC6(CC6)F |
−10.2
± 0.3
|
7.4
± 0.2
|
71 |
EDJ-MED-8bb691af-4
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−10.2
± 0.3
|
7.4
± 0.2
|
72 |
PET-UNK-6af7266d-4
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nncs6 |
−10.1
± 0.3
|
7.4
± 0.2
|
73 |
EDJ-MED-4cb9dd84-3
|
|
c1cc2cncc(c2cc1Cl)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NCC6CC6 |
−10.1
± 0.3
|
7.4
± 0.2
|
74 |
LUO-POS-f7b1afe6-4
|
|
CC1(CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5)C |
−10.1
± 0.3
|
7.4
± 0.2
|
75 |
EDJ-MED-dfa1d800-5
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN6CC(C6)(F)F)c7cc(ccc7C2=O)Cl |
−10.1
± 0.5
|
7.4
± 0.3
|
76 |
PET-UNK-aa57768f-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−10.1
± 0.2
|
7.3
± 0.1
|
77 |
PET-UNK-aa57768f-7
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−10.1
± 0.2
|
7.3
± 0.1
|
78 |
MAT-POS-1d5ab790-2
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4c(ccc5)Cl)Cl |
−10.0
± 0.2
|
7.3
± 0.2
|
79 |
EDJ-MED-6b23330e-1
|
|
CC(C)CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−10.0
± 0.4
|
7.3
± 0.3
|
80 |
MAT-POS-983b399a-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CCOc5c4cc(cc5)Cl |
−10.0
± 0.3
|
7.3
± 0.3
|
81 |
ALP-POS-ecbed2ba-12
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NCC6CC6 |
−10.0
± 0.3
|
7.3
± 0.2
|
82 |
ALP-POS-c3a90b22-10
|
|
CNC(=O)C1(CCOCC1)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−10.0
± 0.3
|
7.3
± 0.2
|
83 |
EDJ-MED-5cd3920d-5
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C(F)F |
−10.0
± 0.8
|
7.3
± 0.6
|
84 |
PET-UNK-77d5678a-5
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−10.0
± 0.3
|
7.3
± 0.2
|
85 |
EDJ-MED-9f4ac58c-1
|
|
c1cc2c(cc1Cl)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−10.0
± 0.4
|
7.3
± 0.3
|
86 |
EDJ-MED-7e491f08-1
|
|
c1ccc2c(c1)cncc2N3CC([C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)(F)F |
−10.0
± 0.9
|
7.3
± 0.6
|
87 |
EDJ-MED-4138fde9-9
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6CC(C6)O |
−9.9
± 0.8
|
7.2
± 0.6
|
88 |
MAT-POS-69786b79-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NC6(CC6)C#N |
−9.9
± 0.4
|
7.2
± 0.3
|
89 |
LUO-POS-e1dab717-12
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(S(=O)(=O)c5c4cc(cc5)Cl)CC(=O)NCC6CC6 |
−9.9
± 0.6
|
7.2
± 0.5
|
90 |
LUO-POS-868e8996-12
|
|
CNC(=O)CN1Cc2ccc(cc2[C@@]3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−9.9
± 0.4
|
7.2
± 0.3
|
91 |
MAT-POS-e75f6e44-14
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NCC6COC6 |
−9.9
± 0.4
|
7.2
± 0.3
|
92 |
MAT-POS-e75f6e44-16
|
|
CN1CC(C1)CNC(=O)CN2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−9.9
± 0.3
|
7.2
± 0.2
|
93 |
PET-UNK-77d5678a-6
|
|
COC(=O)CN1CC2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.9
± 0.2
|
7.2
± 0.2
|
94 |
MAT-POS-96396902-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)Cc6nncs6 |
−9.9
± 0.3
|
7.2
± 0.2
|
95 |
MAT-POS-e75f6e44-11
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NCC6(CC6)C#N |
−9.8
± 0.2
|
7.2
± 0.2
|
96 |
EDJ-MED-6b23330e-7
|
|
CC(C)(CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl)N |
−9.8
± 0.4
|
7.2
± 0.3
|
97 |
PET-UNK-77d5678a-2
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−9.8
± 0.3
|
7.2
± 0.2
|
98 |
MAT-POS-853c0ffa-18
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5c(cc(c6)F)Cl)Cl |
−9.8
± 0.7
|
7.1
± 0.5
|
99 |
MAT-POS-e75f6e44-13
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NCC6CCC6 |
−9.8
± 0.3
|
7.1
± 0.2
|
100 |
12_-111-3e02a1cd-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−9.7
± 0.3
|
7.1
± 0.2
|