Rank |
Compound |
SMILES |
ΔG / kcal M-1 |
pIC50 |
201 |
EDJ-MED-40e596c8-3
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CCNC(=O)C6CC6 |
−8.4
± 0.5
|
6.1
± 0.4
|
202 |
EDJ-MED-6b23330e-3
|
|
CC(C)(CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl)C#N |
−8.4
± 0.4
|
6.1
± 0.3
|
203 |
EDJ-MED-33064c06-10
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC(=O)NCC6(CC6)CO |
−8.4
± 0.3
|
6.1
± 0.2
|
204 |
MAT-POS-853c0ffa-11
|
|
CC(C)(c1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)O |
−8.4
± 0.8
|
6.1
± 0.6
|
205 |
MIK-ENA-794411b8-1
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.4
± 0.3
|
6.1
± 0.2
|
206 |
LUO-POS-9931618f-2
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.4
± 0.3
|
6.1
± 0.2
|
207 |
MAT-POS-e75f6e44-6
|
|
CNC1(CC1)CNC(=O)CN2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−8.4
± 0.6
|
6.1
± 0.5
|
208 |
MAT-POS-e75f6e44-18
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NCC6CC(C6)F |
−8.4
± 0.3
|
6.1
± 0.3
|
209 |
ALP-POS-ecbed2ba-16
|
|
CN(CCC#N)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−8.4
± 1.0
|
6.1
± 0.7
|
210 |
ALP-POS-c3a90b22-1
|
|
CNC(=O)C1(CCC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.3
± 0.7
|
6.1
± 0.5
|
211 |
MIK-ENA-37e0b697-1
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.3
± 0.3
|
6.1
± 0.2
|
212 |
PET-UNK-94036022-7
|
|
CNC(=O)CN1Cc2ccc(cc2[C@]3(C1)C(=O)C(=C)N(C3=O)c4cncc5c4cccc5)Cl |
−8.3
± 0.3
|
6.1
± 0.2
|
213 |
ALP-POS-c3a90b22-5
|
|
CNC(=O)CCN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.3
± 0.4
|
6.1
± 0.3
|
214 |
JOH-MSK-51c67e7d-1
|
|
CN1Cc2ccc(cc2[C@@]3(C1)CC(=O)N(C3=O)c4cncc5c4cccc5)Cl |
−8.3
± 0.3
|
6.1
± 0.2
|
215 |
VLA-UNK-61877630-10
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C(F)(F)F |
−8.3
± 0.9
|
6.0
± 0.7
|
216 |
EDJ-MED-cc48ee33-3
|
|
Cn1c(ccn1)C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−8.3
± 0.2
|
6.0
± 0.2
|
217 |
VLA-UNK-e334495f-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)c5cc(ccc5CN(C4C(F)F)S(=O)(=O)CC6(CC6)C#N)Cl |
−8.3
± 0.5
|
6.0
± 0.4
|
218 |
EDJ-MED-ee81482e-5
|
|
c1cc2cncc(c2cc1CN3CC4(C3)COC4)N5CCC6(C5=O)CN(Cc7c6cc(cc7)Cl)S(=O)(=O)CC8(CC8)C#N |
−8.3
± 0.8
|
6.0
± 0.6
|
219 |
PET-UNK-626a1084-2
|
|
C#CCN1C[C@]2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.3
± 0.4
|
6.0
± 0.3
|
220 |
MIK-ENA-e143773d-1
|
|
CC[C@H]1CN(C(=O)[C@@]12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−8.3
± 0.8
|
6.0
± 0.6
|
221 |
LUO-POS-e1dab717-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.2
± 0.3
|
6.0
± 0.2
|
222 |
MAT-POS-853c0ffa-1
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3c(ccc4)Cl)c5cc(ccc5C1=O)Cl |
−8.2
± 0.1
|
5.99
± 0.09
|
223 |
PET-UNK-37c7074c-2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6ccon6 |
−8.2
± 0.2
|
6.0
± 0.1
|
224 |
EDJ-MED-9f4ac58c-2
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.2
± 0.6
|
6.0
± 0.4
|
225 |
EDJ-MED-94fddcec-5
|
|
CS(=O)(=O)c1ccc2c(c1)cncc2N3CCC4(C3=O)CCS(=O)(=O)c5c4cc(cc5)Cl |
−8.2
± 0.5
|
6.0
± 0.3
|
226 |
PET-UNK-c6bcc80b-11
|
|
CS(=O)(=O)Nc1cc2cncc(c2cc1F)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.2
± 0.9
|
6.0
± 0.6
|
227 |
EDJ-MED-33064c06-13
|
|
CNC(=O)C1(COC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.2
± 0.3
|
6.0
± 0.2
|
228 |
VLA-UNK-61877630-3
|
|
CNC(=O)CN1C([C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl)C(F)(F)F |
−8.2
± 0.3
|
5.9
± 0.2
|
229 |
PET-UNK-94036022-14
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)C(=O)C(=C)N(C3=O)c4cncc5c4cccc5)Cl |
−8.2
± 0.3
|
5.9
± 0.2
|
230 |
PET-UNK-37c7074c-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6ccno6 |
−8.1
± 0.2
|
5.9
± 0.1
|
231 |
MAT-POS-e75f6e44-20
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NCC6CS(=O)(=O)C6 |
−8.1
± 0.5
|
5.9
± 0.3
|
232 |
MAT-POS-50a80394-5
|
|
CCC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5 |
−8.1
± 0.2
|
5.9
± 0.1
|
233 |
MAT-POS-1d5ab790-3
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3c(ccc4)Cl)c5cc(ccc5C1=O)Cl |
−8.1
± 0.1
|
5.91
± 0.09
|
234 |
BEN-BAS-c2bc0d80-6
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CCOc5c4cc(cc5)Cl |
−8.1
± 0.1
|
5.90
± 0.08
|
235 |
MAT-POS-50a80394-7
|
|
CC1(CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5)C |
−8.1
± 0.3
|
5.9
± 0.3
|
236 |
MAT-POS-c7726e07-5
|
|
CNC(=O)CN1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−8.1
± 0.2
|
5.9
± 0.1
|
237 |
PET-UNK-626a1084-4
|
|
C#CCN1CC2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.1
± 0.3
|
5.9
± 0.3
|
238 |
EDJ-MED-40e596c8-2
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CS(=O)(=O)NCC6CC6 |
−8.1
± 0.7
|
5.9
± 0.5
|
239 |
MAT-POS-e75f6e44-17
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NCC6(CCC6)O |
−8.0
± 0.3
|
5.9
± 0.2
|
240 |
MAT-POS-566864e2-3
|
|
CNC(=O)C1(CC1)N2Cc3ccc(cc3[C@]4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−8.0
± 0.2
|
5.8
± 0.2
|
241 |
ALP-POS-4483ae88-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CNS(=O)(=O)c5c4cc(cc5)Cl |
−8.0
± 0.4
|
5.8
± 0.3
|
242 |
ALP-POS-c3a90b22-8
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CS(=O)(=O)CC6(CC6)C#N |
−8.0
± 0.4
|
5.8
± 0.3
|
243 |
MAT-POS-576f7758-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.0
± 0.3
|
5.8
± 0.3
|
244 |
MAT-POS-be048f2c-7
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)C(=O)c6ccnn6C7CC7 |
−8.0
± 0.3
|
5.8
± 0.2
|
245 |
EDJ-MED-94fddcec-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CCS(=O)(=O)c5c4cc(cc5)Cl |
−7.9
± 0.4
|
5.8
± 0.3
|
246 |
MAT-POS-ddfe83c6-1
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)OC)c5cc(ccc5C1=O)Cl |
−7.9
± 0.3
|
5.8
± 0.2
|
247 |
PET-UNK-aa57768f-3
|
|
C#CCN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.9
± 0.3
|
5.8
± 0.2
|
248 |
EDJ-MED-98c0a822-1
|
|
CNC(=O)C1(CCC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6S2(=O)=O)Cl |
−7.9
± 0.7
|
5.7
± 0.5
|
249 |
PET-UNK-626a1084-3
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC#N |
−7.9
± 0.2
|
5.7
± 0.2
|
250 |
VLA-UNK-61877630-6
|
|
CNC(=O)CN1C([C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl)C(F)F |
−7.8
± 0.3
|
5.7
± 0.2
|
251 |
MAT-POS-576f7758-1
|
|
CNC(=O)C1(CC1)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.8
± 0.3
|
5.7
± 0.2
|
252 |
JOH-MSK-1f2dff76-2
|
|
CNC(=O)CN1Cc2ccc(cc2[C@]3(C1)CC(=O)N(C3=O)c4cncc5c4cccc5)Cl |
−7.8
± 0.2
|
5.7
± 0.2
|
253 |
PET-UNK-14142a25-10
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.8
± 0.3
|
5.7
± 0.2
|
254 |
EDJ-MED-ede5c6cb-1
|
|
CS(=O)(=O)Nc1ccc2c(c1)cncc2N3CCC4(C3=O)CCS(=O)(=O)c5c4cc(cc5)Cl |
−7.8
± 0.4
|
5.7
± 0.3
|
255 |
EDJ-MED-33064c06-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC(=O)NCC6CS(=O)(=O)C6 |
−7.8
± 0.4
|
5.7
± 0.3
|
256 |
ALP-POS-ecbed2ba-15
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCCC6)C#N |
−7.8
± 1.0
|
5.7
± 0.7
|
257 |
MIK-ENA-5d9157e9-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.7
± 0.6
|
5.6
± 0.5
|
258 |
PET-UNK-626a1084-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC#N |
−7.7
± 0.3
|
5.6
± 0.2
|
259 |
VLA-UNK-5d8210f0-4
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1C(F)(F)F)CCN(C3=O)c4cncc5c4cccc5)Cl |
−7.7
± 0.4
|
5.6
± 0.3
|
260 |
JOH-MSK-4bb3d434-2
|
|
COC(=O)CN1CC2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.7
± 0.3
|
5.6
± 0.2
|
261 |
LUO-POS-e1dab717-5
|
|
CNC(=O)C1(CC1)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)OC)Cl |
−7.7
± 0.3
|
5.6
± 0.2
|
262 |
EDJ-MED-59d5ca70-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)C6(CC6)C(=O)NCC7CC7 |
−7.7
± 0.3
|
5.6
± 0.2
|
263 |
JOH-MSK-4bb3d434-1
|
|
COC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.6
± 0.3
|
5.5
± 0.2
|
264 |
EDJ-MED-40e596c8-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CCNC(=O)C6CC6 |
−7.6
± 0.3
|
5.5
± 0.2
|
265 |
LUO-POS-e1dab717-11
|
|
CCNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5S1(=O)=O)Cl |
−7.6
± 0.5
|
5.5
± 0.3
|
266 |
EDJ-MED-33064c06-5
|
|
CN(C)C1(CC1)CNC(=O)CN2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−7.6
± 0.4
|
5.5
± 0.3
|
267 |
MAT-POS-853c0ffa-12
|
|
CC(C)(c1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)OC)O |
−7.5
± 0.8
|
5.5
± 0.6
|
268 |
EDJ-MED-33064c06-11
|
|
CNC(=O)C1(CCOCC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−7.5
± 0.5
|
5.5
± 0.4
|
269 |
VLA-UNK-61877630-4
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(cc(c5C1=O)F)Cl |
−7.5
± 0.3
|
5.5
± 0.2
|
270 |
MAT-POS-38eb6498-4
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)OCCN(C)C)c5cc(ccc5C1=O)Cl |
−7.5
± 0.5
|
5.4
± 0.4
|
271 |
ALP-POS-c3a90b22-4
|
|
CNC(=O)C1(COC1)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.4
± 0.3
|
5.4
± 0.2
|
272 |
MAT-POS-be048f2c-6
|
|
CC(C)n1c(ccn1)C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.4
± 0.4
|
5.4
± 0.3
|
273 |
VLA-UNK-61877630-8
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(c(c5)F)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.4
± 0.8
|
5.4
± 0.6
|
274 |
VLA-UNK-e334495f-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5F)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.4
± 0.8
|
5.4
± 0.6
|
275 |
EDJ-MED-b6c6ee2b-3
|
|
COc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.4
± 0.9
|
5.4
± 0.6
|
276 |
VLA-UNK-3bd6fc51-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(F)(F)Cl |
−7.4
± 0.2
|
5.4
± 0.1
|
277 |
EDJ-MED-8bb691af-8
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.4
± 0.3
|
5.4
± 0.2
|
278 |
ALP-POS-ecbed2ba-8
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCC6)C#N |
−7.4
± 0.9
|
5.4
± 0.6
|
279 |
ALP-POS-ecbed2ba-1
|
|
CC1(CS(=O)(=O)C1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.3
± 0.8
|
5.4
± 0.6
|
280 |
MIC-UNK-c85ea37c-1
|
|
c1ccc2c(c1)cncc2N3CC(C4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)CC7CCCCC7 |
−7.3
± 0.9
|
5.3
± 0.6
|
281 |
MAT-POS-853c0ffa-7
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5c(ccc6)Cl)Cl |
−7.3
± 0.6
|
5.3
± 0.5
|
282 |
EDJ-MED-94fddcec-6
|
|
CN(c1ccc2c(c1)cncc2N3CCC4(C3=O)CCS(=O)(=O)c5c4cc(cc5)Cl)S(=O)(=O)C |
−7.3
± 0.5
|
5.3
± 0.4
|
283 |
VLA-UNK-61877630-7
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(cc5F)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.3
± 0.9
|
5.3
± 0.6
|
284 |
EDJ-MED-4138fde9-6
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCNCC(F)(F)F)c6cc(ccc6C2=O)Cl |
−7.3
± 0.6
|
5.3
± 0.5
|
285 |
MAT-POS-853c0ffa-13
|
|
c1cc2cncc(c2cc1F)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.3
± 0.9
|
5.3
± 0.6
|
286 |
EDJ-MED-4138fde9-4
|
|
CNC(=O)C1(CC1)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)OCCNCC(F)(F)F)Cl |
−7.3
± 0.4
|
5.3
± 0.3
|
287 |
VLA-UNK-8e615992-2
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(c(cc5C1=O)F)Cl |
−7.2
± 0.4
|
5.3
± 0.3
|
288 |
EDJ-MED-33064c06-6
|
|
CN1CC(C1)CNC(=O)CN2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−7.2
± 0.4
|
5.3
± 0.3
|
289 |
12_-111-3e02a1cd-2
|
|
COC(=O)CN1C[C@]2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.2
± 0.3
|
5.3
± 0.2
|
290 |
PET-UNK-94036022-11
|
|
C#CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CC(=O)N(C4=O)c5cncc6c5cccc6)Cl |
−7.2
± 0.8
|
5.2
± 0.6
|
291 |
MAT-POS-853c0ffa-17
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5c(ccc6)Cl)Cl |
−7.1
± 0.9
|
5.2
± 0.6
|
292 |
MAT-POS-853c0ffa-5
|
|
c1cc2cncc(c2c(c1)Cl)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.1
± 0.1
|
5.15
± 0.10
|
293 |
EDJ-MED-33064c06-3
|
|
CNC1(CC1)CNC(=O)CN2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−7.0
± 0.5
|
5.1
± 0.4
|
294 |
MAT-POS-1d5ab790-1
|
|
c1cc2cncc(c2c(c1)Cl)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.0
± 0.1
|
5.09
± 0.10
|
295 |
MIK-ENA-be04d1d4-1
|
|
CC[C@H]1CN(C(=O)[C@]12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−7.0
± 0.8
|
5.1
± 0.6
|
296 |
EDJ-MED-b6c6ee2b-4
|
|
c1cc2cncc(c2cc1Cl)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−6.9
± 0.7
|
5.0
± 0.5
|
297 |
PET-UNK-94036022-4
|
|
C#CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3[C@]4(C2)CC(=O)N(C4=O)c5cncc6c5cccc6)Cl |
−6.9
± 0.6
|
5.0
± 0.4
|
298 |
EDJ-MED-40e596c8-5
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CS(=O)(=O)NCC6CC6 |
−6.8
± 0.4
|
5.0
± 0.3
|
299 |
EDJ-MED-dfa1d800-1
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN6CCCC6)c7cc(ccc7C2=O)Cl |
−6.8
± 0.4
|
5.0
± 0.3
|
300 |
VLA-UNK-f2612802-3
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(cc(c5S1(=O)=O)F)Cl |
−6.8
± 0.5
|
4.9
± 0.3
|