Rank |
Compound |
SMILES |
ΔG / kcal M-1 |
pIC50 |
1 |
MAT-POS-c2d406ed-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)NC3=O |
−12.7
± 0.3
|
9.3
± 0.2
|
2 |
LUO-POS-b5068a05-1
|
|
CN(C)NC1=NC2(CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
−12.1
± 0.5
|
8.8
± 0.4
|
3 |
VLA-UNK-f702bf1c-6
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CC6CCCCC6 |
−11.3
± 0.1
|
8.25
± 0.09
|
4 |
MAT-POS-c2d406ed-2
|
|
CN1C(=O)N(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−11.3
± 0.2
|
8.2
± 0.2
|
5 |
VLA-UNK-f702bf1c-5
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CC6CCC(=O)NC6 |
−11.0
± 0.2
|
8.0
± 0.1
|
6 |
VLA-UCB-34f3ed0c-14
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CC6CCCCC6 |
−11.0
± 0.1
|
7.99
± 0.09
|
7 |
VLA-UNK-56836b69-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(c(c5)Cl)Cl)NC3=O |
−10.92
± 0.08
|
7.96
± 0.06
|
8 |
MAT-POS-c2d406ed-4
|
|
CN1C(=S)N(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−10.8
± 0.4
|
7.9
± 0.3
|
9 |
VLA-UNK-3a43cd95-1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(c(c5)F)Cl)NC3=O |
−10.72
± 0.07
|
7.81
± 0.05
|
10 |
VLA-UNK-f702bf1c-1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CCc6cc[nH]n6 |
−10.7
± 0.1
|
7.79
± 0.09
|
11 |
LUO-POS-b5068a05-2
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)N=C3NC#N |
−10.7
± 0.3
|
7.8
± 0.2
|
12 |
VLA-UNK-f702bf1c-4
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CC6CC(=O)NC6 |
−10.6
± 0.1
|
7.75
± 0.08
|
13 |
VLA-UNK-56836b69-5
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CC(=O)Nc5c4cc(c(c5)Cl)Cl)NC3=O |
−10.62
± 0.09
|
7.74
± 0.07
|
14 |
EDJ-MED-9f4ac58c-3
|
|
CS(=O)(=O)Nc1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−10.4
± 0.6
|
7.6
± 0.4
|
15 |
VLA-UCB-34f3ed0c-11
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)NC3=O |
−10.38
± 0.06
|
7.56
± 0.04
|
16 |
VLA-UCB-29506327-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCOc5c4cc(cc5)Cl)NC3=O |
−10.38
± 0.06
|
7.56
± 0.04
|
17 |
MAT-POS-2e8b2191-8
|
|
CN1C(=O)N(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)C)c4cncc5c4cccc5 |
−10.37
± 0.08
|
7.56
± 0.06
|
18 |
VLA-MRT-8c78ee15-4
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@]4(CN(Cc5c4cc(cc5)Cl)CC(=O)N)NC3=O |
−10.4
± 0.1
|
7.56
± 0.10
|
19 |
VLA-UNK-cf7facf1-1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@]4(CCOc5c4cc(cc5)Cl)NC3=O |
−10.36
± 0.06
|
7.55
± 0.04
|
20 |
MAT-POS-be048f2c-8
|
|
CCCn1c(ccn1)C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−10.2
± 0.1
|
7.4
± 0.1
|
21 |
EDJ-MED-fed7ac0b-3
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN3)CN(C(=O)c5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−10.2
± 0.4
|
7.4
± 0.3
|
22 |
VLA-MRT-8c78ee15-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CNCc5c4cc(cc5)Cl)NC3=O |
−10.2
± 0.2
|
7.4
± 0.1
|
23 |
VLA-UNK-f702bf1c-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)Cc6cc[nH]n6 |
−10.2
± 0.1
|
7.42
± 0.08
|
24 |
EDJ-MED-8bb691af-9
|
|
CNC(=O)CN1CC2(CC(=O)N(C2)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−10.2
± 0.1
|
7.40
± 0.08
|
25 |
VLA-UNK-f702bf1c-3
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)Cc6nc[nH]n6 |
−10.1
± 0.1
|
7.39
± 0.10
|
26 |
VLA-UNK-56836b69-3
|
|
CN1C(=O)N(C(=O)[C@@]12CCOc3c2cc(c(c3)Cl)Cl)c4cncc5c4cccc5 |
−10.13
± 0.09
|
7.38
± 0.06
|
27 |
VLA-MRT-a639d434-1
|
|
CNC(=O)CN1Cc2ccc(cc2[C@@]3(C1)C(=O)N(C(=O)N3)c4cncc5c4cccc5)Cl |
−10.1
± 0.2
|
7.4
± 0.1
|
28 |
EDJ-MED-7587a9ee-1
|
|
CN1C(=O)N(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)C)c4cncc5c4cccc5 |
−10.13
± 0.08
|
7.38
± 0.06
|
29 |
EDJ-MED-8bb691af-3
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CC(=O)N(C3)c4cncc5c4cccc5)Cl |
−10.1
± 0.2
|
7.4
± 0.1
|
30 |
VLA-MRT-a639d434-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CN(Cc5c4cc(cc5)Cl)CC(=O)N)NC3=O |
−10.1
± 0.1
|
7.4
± 0.1
|
31 |
JOH-MSK-1f2dff76-1
|
|
CNC(=O)CN1Cc2ccc(cc2[C@@]3(C1)CC(=O)N(C3=O)c4cncc5c4cccc5)Cl |
−10.1
± 0.2
|
7.3
± 0.2
|
32 |
LUO-POS-868e8996-9
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−10.0
± 0.3
|
7.3
± 0.2
|
33 |
MAT-POS-1bed62cf-2
|
|
CNC(=O)CN1CC2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.9
± 0.1
|
7.24
± 0.07
|
34 |
PET-UNK-94036022-4
|
|
C#CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3[C@]4(C2)CC(=O)N(C4=O)c5cncc6c5cccc6)Cl |
−9.9
± 0.2
|
7.2
± 0.1
|
35 |
VLA-MRT-8c78ee15-3
|
|
CNC(=O)CN1Cc2ccc(cc2[C@]3(C1)C(=O)N(C(=O)N3)c4cncc5c4cccc5)Cl |
−9.9
± 0.2
|
7.2
± 0.1
|
36 |
PET-UNK-94036022-11
|
|
C#CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CC(=O)N(C4=O)c5cncc6c5cccc6)Cl |
−9.8
± 0.2
|
7.2
± 0.2
|
37 |
MAT-POS-be048f2c-5
|
|
CCn1c(ccn1)C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−9.8
± 0.1
|
7.17
± 0.09
|
38 |
LUO-POS-868e8996-8
|
|
CNC(=O)CN1C[C@]2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.8
± 0.1
|
7.17
± 0.08
|
39 |
PET-UNK-94036022-5
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−9.7
± 0.2
|
7.1
± 0.1
|
40 |
LUO-POS-868e8996-7
|
|
CNC(=O)CN1C[C@@]2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.7
± 0.1
|
7.06
± 0.08
|
41 |
JOH-MSK-1f2dff76-2
|
|
CNC(=O)CN1Cc2ccc(cc2[C@]3(C1)CC(=O)N(C3=O)c4cncc5c4cccc5)Cl |
−9.6
± 0.2
|
7.0
± 0.2
|
42 |
VLA-UNK-f702bf1c-8
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CCc6nc[nH]n6 |
−9.6
± 0.2
|
7.0
± 0.1
|
43 |
EDJ-MED-8bb691af-5
|
|
c1ccc2c(c1)cncc2N3CC4(CC3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.6
± 0.3
|
7.0
± 0.2
|
44 |
MAT-POS-50a80394-3
|
|
CC(C)C1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−9.6
± 0.3
|
7.0
± 0.3
|
45 |
MAT-POS-1bed62cf-1
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.5
± 0.2
|
6.9
± 0.2
|
46 |
MAT-POS-be048f2c-7
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)C(=O)c6ccnn6C7CC7 |
−9.4
± 0.1
|
6.9
± 0.1
|
47 |
PET-UNK-94036022-12
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−9.4
± 0.2
|
6.9
± 0.1
|
48 |
MAT-POS-50a80394-2
|
|
CCC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−9.4
± 0.3
|
6.8
± 0.2
|
49 |
MAT-POS-c2d406ed-3
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)NC3=S |
−9.3
± 0.2
|
6.8
± 0.2
|
50 |
EDJ-MED-dfa1d800-5
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN6CC(C6)(F)F)c7cc(ccc7C2=O)Cl |
−9.3
± 0.2
|
6.8
± 0.1
|
51 |
BEN-BAS-c2bc0d80-7
|
|
CN1C(=O)N(C(=O)C12CCOc3c2cc(cc3)Cl)c4cncc5c4cccc5 |
−9.29
± 0.07
|
6.77
± 0.05
|
52 |
VLA-UNK-3a43cd95-3
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CCOc5c4cc(c(c5)F)Cl |
−9.18
± 0.06
|
6.69
± 0.04
|
53 |
VLA-MRT-8c78ee15-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@]4(CNCc5c4cc(cc5)Cl)NC3=O |
−9.2
± 0.2
|
6.7
± 0.1
|
54 |
MAT-POS-983b399a-3
|
|
c1ccc2c(c1)cncc2N3CC4(CCOc5c4cc(cc5)Cl)CC3=O |
−9.13
± 0.07
|
6.65
± 0.05
|
55 |
EDJ-MED-9f4ac58c-6
|
|
COC1(CC1)CS(=O)(=O)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−9.1
± 0.4
|
6.6
± 0.3
|
56 |
LUO-POS-868e8996-10
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.1
± 0.2
|
6.6
± 0.2
|
57 |
VLA-UCB-50c39ae8-2
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
58 |
VLA-UCB-05e51b3f-5
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@]4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
59 |
BEN-BAS-c2bc0d80-6
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
60 |
MAT-POS-94643566-1
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
61 |
VLA-UNK-f702bf1c-7
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CCN6CCNCC6 |
−9.0
± 0.2
|
6.5
± 0.1
|
62 |
EDJ-MED-9f4ac58c-2
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.9
± 0.4
|
6.5
± 0.3
|
63 |
MAT-POS-576f7758-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.9
± 0.1
|
6.51
± 0.08
|
64 |
EDJ-MED-159244ea-3
|
|
c1ccc2c(c1)cncc2N3C[C@@]4(CCOc5c4cc(cc5)Cl)CC3=O |
−8.89
± 0.08
|
6.48
± 0.06
|
65 |
EDJ-MED-98c0a822-3
|
|
CNC(=O)C1(CCC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.9
± 0.2
|
6.5
± 0.2
|
66 |
EDJ-MED-9f4ac58c-8
|
|
COC1(CC1)CS(=O)(=O)N2CC3(CCN(C3=O)c4cncc5c4ccc(c5)S(=O)(=O)C)c6cc(ccc6C2=O)Cl |
−8.8
± 0.5
|
6.4
± 0.3
|
67 |
MAT-POS-90505e2b-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCOc5c4cc(cc5)Cl)OC3=O |
−8.81
± 0.05
|
6.42
± 0.03
|
68 |
EDJ-MED-dfa1d800-1
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN6CCCC6)c7cc(ccc7C2=O)Cl |
−8.7
± 0.3
|
6.3
± 0.2
|
69 |
MAT-POS-ec6d90b7-1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)OC3=O |
−8.67
± 0.05
|
6.32
± 0.03
|
70 |
MAT-POS-1bed62cf-3
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CC(=O)N(C3=O)c4cncc5c4cccc5)Cl |
−8.7
± 0.2
|
6.3
± 0.1
|
71 |
EDJ-MED-cc48ee33-5
|
|
Cc1cc(n(n1)C)C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−8.7
± 0.1
|
6.3
± 0.1
|
72 |
MAT-POS-ec6d90b7-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@]4(CCOc5c4cc(cc5)Cl)OC3=O |
−8.66
± 0.05
|
6.31
± 0.03
|
73 |
EDJ-MED-9f4ac58c-5
|
|
COC1(CC1)CS(=O)(=O)N2CC3(CCN(C3=O)c4cncc5c4ccc(c5)Cl)c6cc(ccc6C2=O)Cl |
−8.5
± 0.4
|
6.2
± 0.3
|
74 |
EDJ-MED-468565e0-5
|
|
c1cc2cncc(c2cc1OCCN3CC(C3)(F)F)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−8.4
± 0.4
|
6.1
± 0.3
|
75 |
VLA-MRT-a639d434-3
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CNCc5c4cc(cc5)Cl)NC3=O |
−8.4
± 0.2
|
6.1
± 0.1
|
76 |
MAT-POS-853c0ffa-9
|
|
CN(C)CCOc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.4
± 0.4
|
6.1
± 0.3
|
77 |
EDJ-MED-5cd3920d-3
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OC(F)F)c6cc(ccc6C2=O)Cl |
−8.4
± 0.1
|
6.1
± 0.1
|
78 |
EDJ-MED-ee81482e-3
|
|
CN(C)CC(COc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)O |
−8.3
± 0.9
|
6.1
± 0.6
|
79 |
EDJ-MED-7e491f08-2
|
|
CNC(=O)C1(CC1)N2C[C@]3(c4cc(ccc4C2=O)Cl)C(=O)N(CC3(F)F)c5cncc6c5cccc6 |
−8.3
± 0.2
|
6.1
± 0.1
|
80 |
ALP-POS-ecbed2ba-16
|
|
CN(CCC#N)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−8.3
± 0.5
|
6.0
± 0.4
|
81 |
MAT-POS-50a80394-1
|
|
CC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−8.3
± 0.4
|
6.0
± 0.3
|
82 |
EDJ-MED-cc48ee33-2
|
|
Cn1c(ccn1)C(=O)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.3
± 0.1
|
6.0
± 0.1
|
83 |
PET-UNK-aa57768f-7
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−8.2
± 0.1
|
5.99
± 0.08
|
84 |
EDJ-MED-dfa1d800-3
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN6CCS(=O)(=O)CC6)c7cc(ccc7C2=O)Cl |
−8.1
± 0.3
|
5.9
± 0.2
|
85 |
EDJ-MED-dfa1d800-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN6CCOCC6)c7cc(ccc7C2=O)Cl |
−8.1
± 0.3
|
5.9
± 0.2
|
86 |
JOH-MSK-1f2dff76-4
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CNCc5c4cc(cc5)Cl |
−8.1
± 0.2
|
5.9
± 0.1
|
87 |
EDJ-MED-b6c6ee2b-5
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)OCCN(C)C)c5cc(ccc5C1=O)Cl |
−8.0
± 0.2
|
5.9
± 0.2
|
88 |
JOH-MSK-51c67e7d-2
|
|
CN1Cc2ccc(cc2[C@]3(C1)CC(=O)N(C3=O)c4cncc5c4cccc5)Cl |
−8.04
± 0.08
|
5.86
± 0.06
|
89 |
VLA-UCB-34f3ed0c-15
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CN6CCNCC6 |
−8.0
± 0.3
|
5.8
± 0.2
|
90 |
ALP-POS-ecbed2ba-20
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)N6CCC6 |
−7.9
± 0.7
|
5.8
± 0.5
|
91 |
EDG-MED-b1ef7fe3-1
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)Cl)c5cc(ccc5C1=O)Cl |
−7.9
± 0.1
|
5.75
± 0.10
|
92 |
EDJ-MED-fed7ac0b-2
|
|
CNC(=O)C1(CC1)N2CC3(CNN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−7.9
± 0.1
|
5.8
± 0.1
|
93 |
ALP-POS-ecbed2ba-10
|
|
COC1CN(C1)S(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.9
± 0.7
|
5.8
± 0.5
|
94 |
EDJ-MED-cc48ee33-4
|
|
Cc1cnn(c1C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl)C |
−7.9
± 0.2
|
5.7
± 0.1
|
95 |
EDJ-MED-976a33d5-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4ccc(c5)S(=O)(=O)C)c6cc(ccc6C2=O)Cl |
−7.8
± 0.2
|
5.7
± 0.1
|
96 |
ALP-POS-ecbed2ba-18
|
|
CCN(C)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−7.8
± 0.4
|
5.7
± 0.3
|
97 |
MAT-POS-40ad851a-2
|
|
CCN(C)CCOc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.8
± 0.4
|
5.7
± 0.3
|
98 |
PET-UNK-aa57768f-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−7.8
± 0.1
|
5.7
± 0.1
|
99 |
LUO-POS-ed2cfb03-1
|
|
CN1CCN(CC1)S(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.8
± 0.5
|
5.7
± 0.4
|
100 |
MAT-POS-40ad851a-4
|
|
CN(C)CCCOc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.8
± 0.5
|
5.6
± 0.4
|