Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
201 |
KAD-UNI-cb0f2bbc-22_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)C[NH2+]CCN5C(=O)c6ccccc6C5=O |
−9.4
± 0.1
|
202 |
LAU-MED-88a3970a-8_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H]3CCOc4c3cc(cc4CCCCO)Cl |
−9.4
± 0.2
|
203 |
MAT-POS-4223bc15-11_16
|
|
C[C@H]1CC[N@](C1)S(=O)(=O)[N@]2Cc3ccc(cc3[C@H](C2)C(=O)Nc4cncc5c4cccc5)Cl |
−9.39
± 0.08
|
204 |
MAT-POS-ec6d90b7-6_1
|
|
COc1ccc2cncc(c2c1)NC(=O)[C@H]3CCNc4c3cc(c(c4)Cl)Cl |
−9.38
± 0.09
|
205 |
EDJ-MED-50011917-3_1
|
|
COc1c(cc(cc1CC(=O)Nc2cncc3c2cccc3)Cl)C[C@@H]4CC(=O)N4 |
−9.4
± 0.3
|
206 |
LON-WEI-4d77710c-47_1
|
|
CCc1ccccc1N(CC)C(=O)Nc2cn(c(=O)c3c2cccc3)C |
−9.4
± 0.3
|
207 |
LON-WEI-4d77710c-13_1
|
|
CC(C)Cn1cc(c2ccccc2c1=O)NC(=O)NC[C@@H]3CCCO3 |
−9.4
± 0.4
|
208 |
DAR-DIA-5ff57136-11_1
|
|
C=C=CC(=O)N(c1cncc2c1cccc2)C(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.4
± 0.2
|
209 |
MIC-UNK-cdc2493e-21_3
|
|
CC(=O)N(C)[C@@H]1CC[C@H](C1)N(c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.4
± 0.3
|
210 |
EDG-MED-ba1ac7b9-26_2
|
|
C[C@@H]1C[N@H+]([C@H](CN1C(=O)C[C@@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)C)CCO |
−9.4
± 0.2
|
211 |
ALP-POS-5bb456a5-2_6
|
|
C[C@H]1C[N@@](CC[C@H]1NC(=O)C[C@@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)S(=O)(=O)C |
−9.4
± 0.4
|
212 |
ALF-EVA-ced740bd-4_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3COc4c3cc(cc4)F |
−9.3
± 0.1
|
213 |
KAD-UNI-cb0f2bbc-13_1
|
|
Cn1c(nc2c1c(=O)[nH]c(=O)n2C)C[NH2+]C[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−9.3
± 0.1
|
214 |
EDJ-MED-841e0cf0-6_1
|
|
CN(C)S(=O)(=O)[N@@]1Cc2ccc(cc2[C@@H](C1)C(=O)Nc3cncc4c3cc(cc4)F)Cl |
−9.3
± 0.1
|
215 |
MAK-UNK-919546f0-2_2
|
|
c1ccc(cc1)[C@H](C(=O)Nc2cncc3c2cccc3)[NH3+] |
−9.3
± 0.2
|
216 |
ED_-GRI-5b13fbe2-35_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCCn5c(c(cn5)C6=CC[NH2+]CC6)N |
−9.3
± 0.4
|
217 |
PET-UNK-5d7c542f-5_1
|
|
C=CS(=O)(=O)CCO[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.3
± 0.1
|
218 |
DAR-DIA-0d514e7d-32_13
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3[C@@H]4C[C@H]4CO[C@H]5[C@@H]3C=C(C=C5)Cl |
−9.3
± 0.2
|
219 |
ALF-EVA-5b152d2f-2_1
|
|
Cc1ccc2cncc(c2c1)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.3
± 0.3
|
220 |
LON-WEI-4d77710c-60_1
|
|
CC1CC[NH+](CC1)CCCNC(=O)Nc2cn(c(=O)c3c2cccc3)CC(C)C |
−9.3
± 0.5
|
221 |
MAK-UNK-c749d764-31_8
|
|
CC/C=C(/c1cncc2c1cccc2)\C(=O)C[C@H]3CCC[C@H]([C@H]3O)C(F)F |
−9.3
± 0.3
|
222 |
EDJ-MED-841e0cf0-4_2
|
|
C[C@@]1(C[N@](Cc2c1cc(cc2)Cl)S(=O)(=O)C)C(=O)Nc3cncc4c3cc(cc4)S(=O)(=O)C |
−9.3
± 0.2
|
223 |
RAL-THA-1d44ff04-2_1
|
|
c1ccc2c(c1)cncc2NC(=O)Cc3cc(cc(c3)Cl)OCc4[nH]ncn4 |
−9.3
± 0.2
|
224 |
EDJ-MED-e4b030d8-11_1
|
|
C[C@H]1COc2ccc(cc2[C@@H]1C(=O)Nc3cncc4c3cccc4)Cl |
−9.28
± 0.09
|
225 |
DAR-DIA-f6ee7aeb-4_1
|
|
c1ccc2c(c1)cncc2N3C[C@@H]([C@@H](CC3=O)c4cc(cc(c4)Cl)OCCC(F)(F)F)c5c[nH]c(=O)[nH]c5=O |
−9.3
± 0.2
|
226 |
MIC-UNK-5a93dd5f-3_11
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](c3cccc(c3)Cl)[N@H+]4CC[C@@H]5CCCC[C@H]5C4 |
−9.3
± 0.2
|
227 |
MAK-UNK-c749d764-26_5
|
|
c1ccc2c(c1)cncc2NC(=O)C[C@@H]3CCCC[C@@H]([C@H]3O)Cl |
−9.3
± 0.3
|
228 |
MIC-UNK-cdc2493e-10_2
|
|
CC(=O)N[C@H]1CC[C@@H](C1)N(c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.3
± 0.3
|
229 |
PET-UNK-c5865d42-2_2
|
|
c1ccc2c(c1)cncc2NC(=O)Cc3cc(cc(c3)Cl)C([C@H]4CCN4)(F)F |
−9.3
± 0.3
|
230 |
ALP-UNI-8e43a71e-5_10
|
|
C[C@H]1C[N@@](CC[C@@H]1NC(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)S(=O)(=O)C |
−9.3
± 0.3
|
231 |
MAT-POS-96f51285-6_1
|
|
COc1ccc2cncc(c2c1)NC(=O)[C@@H]3CCNc4c3cc(c(c4)Cl)Cl |
−9.25
± 0.09
|
232 |
VLA-UNK-f702bf1c-4_2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)C[C@H]6CC(=O)NC6 |
−9.2
± 0.4
|
233 |
MIC-UNK-9582b2c5-2_5
|
|
CC(=O)N1CC[C@@H]2[C@@H](C1)C[C@H](C(=O)N2c3cccc(c3)Cl)c4cncc5c4cccc5 |
−9.2
± 0.3
|
234 |
MIC-UNK-bcd487e9-9_1
|
|
Cn1cc(nn1)CN(c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.2
± 0.2
|
235 |
ERI-UCB-d6de1f3c-5_1
|
|
c1ccc2c(c1)cncc2C(=O)N3C[C@@H](N(C(=O)C3)c4cccc(c4)Cl)CC5CCCCC5 |
−9.2
± 0.3
|
236 |
JAG-UCB-7b680c2b-1_1
|
|
CC(C)(C)OC(=O)NCc1cccc(c1)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.2
± 0.3
|
237 |
RAL-THA-8416115c-4_3
|
|
CCCN1CC[C@H](c2c1ccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.2
± 0.2
|
238 |
EDJ-MED-611d11e7-7_1
|
|
COc1ccc2cncc(c2c1)NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OC |
−9.21
± 0.09
|
239 |
ALP-POS-ce760d3f-6_1
|
|
COc1ccc2cncc(c2c1)NC(=O)C3=CCOc4c3cc(cc4)Cl |
−9.2
± 0.3
|
240 |
EDJ-MED-e4b030d8-6_1
|
|
CCC[C@H]1COc2ccc(cc2[C@@H]1C(=O)Nc3cncc4c3cccc4)Cl |
−9.2
± 0.2
|
241 |
PET-UNK-bcc8fd08-1_1
|
|
[2H]C([2H])([2H])O[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.20
± 0.09
|
242 |
ALP-UNI-3735e77e-4_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H]3CCNc4c3cc(c(c4)Cl)Cl |
−9.20
± 0.10
|
243 |
EDG-MED-0e5afe9d-3_1
|
|
CO[C@@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.20
± 0.10
|
244 |
ALP-POS-2da19ca7-6_1
|
|
Cn1c(nnn1)C2=CCN(CC2)C(=O)C[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−9.2
± 0.3
|
245 |
MAT-POS-b3e365b9-1_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.20
± 0.10
|
246 |
RAL-THA-4aa06b95-3_1
|
|
CNC(=O)N1CC[C@@H](c2c1ccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.2
± 0.3
|
247 |
ALP-UNI-3496895b-6_1
|
|
CCN1CC[NH+](CC1)C2CN(C2)C(=O)C[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−9.2
± 0.4
|
248 |
MAK-UNK-c749d764-2_8
|
|
CC[C@H]1CCC[C@H]([C@H]1O)CC(=O)Nc2cncc3c2cccc3 |
−9.2
± 0.4
|
249 |
NIR-THE-af15c15d-1_1
|
|
CC#CC(=O)N(c1cncc2c1cccc2)C(=O)[C@@H]3COc4c3cc(cc4)Cl |
−9.2
± 0.2
|
250 |
MAK-UNK-8be7dca9-8_1
|
|
c1cc2cncc(c2cc1CC(=O)[O-])NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.2
± 0.3
|
251 |
MIC-UNK-c66144cb-2_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](CCc3ccc(cc3)F)c4cccc(c4)Cl |
−9.2
± 0.3
|
252 |
MAT-POS-3b92565d-8_1
|
|
Cn1cc(c2ccccc2c1=O)NC(=O)Cc3cc(cc(c3)Cl)OC |
−9.2
± 0.4
|
253 |
ALP-UNI-0676e700-10_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)c5ccc6nnnn6c5 |
−9.2
± 0.4
|
254 |
MAT-POS-f7918075-1_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H]3CCOc4c3cc(cc4)Cl |
−9.2
± 0.2
|
255 |
ED_-GRI-5b13fbe2-16_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OC[C@H](c5cn(nn5)CC6CC6)[NH3+] |
−9.2
± 0.2
|
256 |
DAR-DIA-0cde14eb-47_1
|
|
c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)C4(CC4)Cl |
−9.2
± 0.2
|
257 |
RAL-THA-b00e3cbf-1_1
|
|
c1ccc2c(c1)c(cnc2C#N)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.2
± 0.2
|
258 |
DAR-DIA-076fb6ea-3_1
|
|
COC(=O)/C=C/C(=O)N(c1cncc2c1cccc2)C(=O)Cc3cccc(c3)Cl |
−9.2
± 0.2
|
259 |
DAR-DIA-6a508060-3_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCOc4c3cc(cc4)C#N |
−9.2
± 0.3
|
260 |
ALP-POS-2da19ca7-7_8
|
|
C[C@H]1C[N@](CC[C@H]1NC(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)S(=O)(=O)C |
−9.2
± 0.3
|
261 |
MAT-POS-afd4d4fd-3_1
|
|
c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3Cl)Cl |
−9.2
± 0.3
|
262 |
MIC-UNK-cdc2493e-8_2
|
|
c1ccc2c(c1)cncc2NC(=O)N(c3cccc(c3)Cl)[C@H]4CC[C@@H]5CCCC[C@@H]5C4 |
−9.1
± 0.3
|
263 |
MAK-UNK-8be7dca9-7_1
|
|
c1cc2cncc(c2cc1C(=O)[O-])NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.1
± 0.2
|
264 |
ALP-UNI-3496895b-1_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCS(=O)(=O)[N@@]6[C@@H]5CCCC6 |
−9.1
± 0.5
|
265 |
LON-WEI-4d77710c-15_1
|
|
CC(C)Cn1cc(c2ccccc2c1=O)NC(=O)NCCCN3CCCC3=O |
−9.1
± 0.2
|
266 |
MIC-UNK-cdc2493e-8_4
|
|
c1ccc2c(c1)cncc2NC(=O)N(c3cccc(c3)Cl)[C@H]4CC[C@H]5CCCC[C@@H]5C4 |
−9.1
± 0.3
|
267 |
MAT-POS-4223bc15-24_1
|
|
CN(C)C(=O)C[N@@H+]1Cc2ccc(cc2[C@@H](C1)C(=O)Nc3cncc4c3cccc4)Cl |
−9.13
± 0.09
|
268 |
BEN-DND-c852c98b-4_1
|
|
c1cc2cncc(c2cc1O)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.13
± 0.10
|
269 |
PET-UNK-bcc8fd08-2_1
|
|
[2H]C([2H])([2H])O[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cc(cc4)F |
−9.12
± 0.09
|
270 |
MAK-UNK-8be7dca9-2_1
|
|
c1cc2c(cc1CC(=O)N)cncc2NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.1
± 0.3
|
271 |
EDJ-MED-d203f206-16_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC[C@H]5c6n[n-]nn6 |
−9.1
± 0.3
|
272 |
ALP-UNI-8e43a71e-15_24
|
|
c1ccc2c(c1)cncc2NC(=O)[C@]3(CCOc4c3cc(cc4)Cl)CC(=O)N[C@H]5C[C@H]6[C@@H]5C[C@H](C6)C(=O)N |
−9.1
± 0.2
|
273 |
KAD-UNI-8a629cb0-20_1
|
|
C[C@@H](C(=O)N1CCC(CC1)C(=O)N)O[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.1
± 0.4
|
274 |
MAT-POS-f9802937-7_1
|
|
COc1ccc2cncc(c2c1)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.10
± 0.10
|
275 |
MIC-UNK-91acba05-1_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CNC(=O)c4c3cc(cc4)Cl |
−9.10
± 0.10
|
276 |
MAK-UNK-ffc90da7-2_2
|
|
c1ccc2c(c1)cncc2NC(=O)C[C@H]3CCC[C@@H]([C@@H]3O)Cl |
−9.1
± 0.3
|
277 |
DAR-DIA-53551c05-6_1
|
|
c1ccc2c(c1)cncc2CN3c4ccccc4C(=O)C3=O |
−9.1
± 0.2
|
278 |
DAR-DIA-ecdbc7dd-12_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCNc4c3cc(cc4)Cl)C[NH+]5CCCCC5 |
−9.1
± 0.1
|
279 |
DAR-DIA-6be260fc-1_1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CNc5c4cc(cc5)Cl |
−9.1
± 0.3
|
280 |
VLA-UCB-34f3ed0c-1_1
|
|
C=C(C#N)C(=O)N(c1cncc2c1cccc2)C(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.1
± 0.3
|
281 |
LON-WEI-4d77710c-59_1
|
|
Cn1cc(c2ccccc2c1=O)NC(=O)N(Cc3ccco3)C[C@@H]4CCCO4 |
−9.1
± 0.1
|
282 |
ERI-UCB-fbdd3ea1-27_2
|
|
CC(C)(C)c1cc(no1)N([C@H](c2cncc3c2cccc3)C(=O)NC(C)(C)C)C(=O)C=C |
−9.1
± 0.3
|
283 |
VLA-UNK-83c3754c-1_1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(COc5c4cc(cc5)Cl)NC3=O |
−9.1
± 0.4
|
284 |
PET-UNK-8df914d1-1_1
|
|
COc1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl |
−9.1
± 0.1
|
285 |
MIC-UNK-0a05c952-3_1
|
|
c1ccc2c(c1)cncc2N3[C@@H](C[C@@H](C3=O)c4ccc(c(c4)Cl)Cl)[C@@H]5CO5 |
−9.1
± 0.2
|
286 |
EDJ-MED-c314995a-1_1
|
|
c1ccc2c(c1)cncc2NC(=O)N(CCC3CCCCC3)c4cccc(c4)Cl |
−9.07
± 0.09
|
287 |
MIC-UNK-cdc2493e-14_1
|
|
c1ccc2c(c1)cncc2NC(=O)N(c3cccc(c3)Cl)[C@@H]4CC[C@@H](C4)[NH+]5CCCCC5 |
−9.1
± 0.3
|
288 |
ALP-POS-a0a4abd7-3_2
|
|
Cn1c(=O)c(c[nH]c1=O)NC[C@]2(CCOc3c2ccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.1
± 0.3
|
289 |
MIC-UNK-cdc2493e-2_1
|
|
c1ccc2c(c1)cncc2NC(=O)N(CC[C@@H]3CCCO3)c4cccc(c4)Cl |
−9.1
± 0.3
|
290 |
DAR-DIA-0d514e7d-4_1
|
|
C[C@H]1COc2c(cc(cc2OC3CCCC3)Cl)[C@@H]1C(=O)Nc4cncc5c4cccc5 |
−9.0
± 0.2
|
291 |
MAT-POS-0c8fa4a7-1_1
|
|
c1ccc2c(c1)cncc2NC(=O)C3=CCCc4c3cc(cc4)Cl |
−9.05
± 0.10
|
292 |
MAK-UNK-8be7dca9-4_1
|
|
c1cc2cncc(c2cc1N3CC[NH2+]CC3)NC(=O)[C@@H]4CCOc5c4cc(cc5)Cl |
−9.0
± 0.2
|
293 |
MIC-UNK-d36ab305-1_2
|
|
CC(=O)Nc1ccc(cc1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.0
± 0.2
|
294 |
VLA-UCB-1dbca3b4-18_1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@H](CNC3=O)c4cccc(c4)Cl |
−9.0
± 0.2
|
295 |
RAL-THA-05e671eb-10_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCOc4c3cc(c(c4)F)Cl |
−9.03
± 0.10
|
296 |
ERI-UCB-ce40166b-9_1
|
|
c1ccc2c(c1)cncc2CC(=O)Nc3cc(cc(c3)O[C@@H]4CC(=O)N4)C#N |
−9.0
± 0.2
|
297 |
EDG-MED-90036822-79_1
|
|
Cc1c(c(n[nH]1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)F |
−9.0
± 0.4
|
298 |
ALF-EVA-5b152d2f-6_1
|
|
C[C@H]1CCOc2ccc(cc2[C@@H]1C(=O)Nc3cncc4c3cccc4)Cl |
−9.0
± 0.4
|
299 |
MIC-UNK-cdc2493e-10_4
|
|
CC(=O)N[C@H]1CC[C@H](C1)N(c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.0
± 0.3
|
300 |
MIC-UNK-91acba05-5_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H]3CCNc4c3cc(cc4)Cl |
−9.0
± 0.4
|