Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
101 |
EDG-MED-90036822-77_1
|
|
c1cc2c(c(cnc2)NC(=O)[C@]3(c4c(ccc(c4)Cl)OCC3)NC(=O)[C@H]5C[C@](C5)(F)CO)cc1 |
−9.9
± 0.2
|
102 |
MAT-POS-89e65850-1_1
|
|
CO[C@@]1(CC(=O)Nc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.9
± 0.3
|
103 |
MAT-POS-b5746674-108_2
|
|
Cc1ccc(cc1)C[N@H+]2CC[C@@H](C2)CNC(=O)Nc3cn(c(=O)c4c3cccc4)CC(C)C |
−9.9
± 0.2
|
104 |
MAK-UNK-ffc90da7-4_7
|
|
C[C@@H](C[NH2+]C[C@H]1CCCO1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.9
± 0.2
|
105 |
MAK-UNK-83e0a0b4-4_2
|
|
CCCCc1ccc2c(c1)[C@H](CCO2)C(=O)N(CCNC3C[NH2+]C3)c4cncc5c4cccc5 |
−9.9
± 0.4
|
106 |
MIC-UNK-9582b2c5-2_3
|
|
CC(=O)N1CC[C@@H]2[C@H](C1)C[C@@H](C(=O)N2c3cccc(c3)Cl)c4cncc5c4cccc5 |
−9.9
± 0.2
|
107 |
MIC-UNK-cdc2493e-13_1
|
|
c1ccc2c(c1)cncc2NC(=O)N(c3cccc(c3)Cl)C4CCC(CC4)[NH+]5CCCCC5 |
−9.9
± 0.2
|
108 |
EDJ-MED-50011917-2_1
|
|
Cc1c(cc(cc1O[C@@H]2CC(=O)N2)Cl)CC(=O)Nc3cncc4c3cccc4 |
−9.9
± 0.5
|
109 |
ALP-POS-2da19ca7-7_3
|
|
C[C@@H]1C[N@](CC[C@@H]1NC(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)S(=O)(=O)C |
−9.9
± 0.4
|
110 |
MAK-UNK-c749d764-8_8
|
|
c1ccc2c(c1)cncc2NC(=O)C[C@H]3CCC[C@H]([C@H]3O)C(F)F |
−9.9
± 0.2
|
111 |
VLA-UCB-34f3ed0c-17_1
|
|
c1ccc2c(c1)cncc2N3C(=O)CN([C@@]4(C3=O)CCOc5c4cc(cc5)Cl)C(=O)C6CCCCC6 |
−9.9
± 0.2
|
112 |
ADA-UCB-dc2b944c-11_1
|
|
c1ccc2c(c1)c(cnc2Br)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.9
± 0.3
|
113 |
KAD-UNI-877d7bed-11_3
|
|
CC(C)([C@@H]1CCN(C1)C(=O)COc2cc(cc3c2OCC[C@H]3C(=O)Nc4cncc5c4cccc5)Cl)O |
−9.9
± 0.2
|
114 |
MAK-UNK-c749d764-26_4
|
|
c1ccc2c(c1)cncc2NC(=O)C[C@H]3CCCC[C@H]([C@@H]3O)Cl |
−9.9
± 0.3
|
115 |
MIC-UNK-bcd487e9-4_1
|
|
c1ccc2c(c1)cncc2NC(=O)N(C[C@@H]3CCCO3)c4cccc(c4)Cl |
−9.9
± 0.2
|
116 |
DAR-DIA-ecdbc7dd-11_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)C[NH+]5CCCCC5 |
−9.9
± 0.1
|
117 |
LON-WEI-4d77710c-28_1
|
|
CC(C)Cn1cc(c2ccccc2c1=O)NC(=O)NCc3cc(ccc3OC)OC |
−9.9
± 0.3
|
118 |
MAK-UNK-919546f0-5_1
|
|
CN(CC(=O)Nc1cncc2c1cccc2)C=O |
−9.9
± 0.2
|
119 |
RAL-THA-8416115c-2_1
|
|
CN1CC[C@@H](c2c1ccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.9
± 0.2
|
120 |
MAK-UNK-c749d764-15_12
|
|
C[C@H](N(c1cncc2c1cccc2)C(=O)C[C@H]3CCC[C@@H]([C@H]3O)C(F)F)OCC4CCCCC4 |
−9.9
± 0.2
|
121 |
VLA-UCB-1dbca3b4-16_1
|
|
c1ccc2c(c1)cncc2NC(=O)C3=C(COc4c3cc(cc4)Cl)O |
−9.8
± 0.3
|
122 |
ALP-POS-fab80cf2-1_1
|
|
c1ccc2c(c1)cncc2NC(=O)Cc3cc(cc(c3)Cl)C([C@@H]4CC(=O)N4)(F)F |
−9.8
± 0.2
|
123 |
NAU-LAT-b7d8c353-8_1
|
|
c1cc(c2cncc(c2c1)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl)C[NH3+] |
−9.8
± 0.3
|
124 |
MAT-POS-b5746674-105_1
|
|
CC(C)Cn1cc(c2ccccc2c1=O)NC(=O)NC3CC[NH+](CC3)Cc4ccccc4 |
−9.8
± 0.2
|
125 |
ALP-POS-2da19ca7-1_1
|
|
CCNC(=O)C[NH+]1CCN(CC1)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.8
± 0.2
|
126 |
MAT-POS-a13804f0-3_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCOc4c3cc(c(c4)F)Cl |
−9.82
± 0.09
|
127 |
DAR-DIA-0d514e7d-31_2
|
|
C[C@H]1CCO[C@@H]2C=CC(=C[C@@H]2[C@@H]1C(=O)Nc3cncc4c3cccc4)Cl |
−9.8
± 0.3
|
128 |
MAT-POS-bbbbc21a-1_1
|
|
COc1ccc(cc1CC(=O)Nc2cncc3c2cccc3)Cl |
−9.8
± 0.5
|
129 |
LON-WEI-4d77710c-54_1
|
|
CC(C)Cn1cc(c2ccccc2c1=O)NC(=O)N3CCC(CC3)Cc4ccccc4 |
−9.8
± 0.2
|
130 |
JOH-SUS-a69c159d-6_2
|
|
c1ccc2c(c1)c(c(nc2F)F)NC(=O)[C@H]3CCOc4c3cc(cc4)Cl |
−9.8
± 0.2
|
131 |
FRA-DIA-0fa076fe-2_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H]3COc4c3cc(cc4Cl)O |
−9.8
± 0.3
|
132 |
MAK-UNK-c749d764-33_4
|
|
CS(=O)(=O)N(c1cncc2c1cccc2)C(=O)C[C@H]3CCC[C@H]([C@@H]3O)C(F)F |
−9.8
± 0.3
|
133 |
LON-WEI-adc59df6-52_2
|
|
CC(C)(C)c1ccc(cc1)N([C@H](c2cncc3c2cccc3)C(=O)NC(C)(C)C)C(=O)C=C |
−9.8
± 0.3
|
134 |
VLA-UCB-34f3ed0c-19_1
|
|
c1ccc2c(c1)cncc2N(C(=O)c3ccco3)C(=O)[C@@H]4CCOc5c4cc(cc5)Cl |
−9.8
± 0.3
|
135 |
ALP-UNI-44c99a80-4_1
|
|
c1ccc2c(c1)cncc2N(Cc3cnco3)C(=O)Cc4cccc(c4)Cl |
−9.8
± 0.3
|
136 |
EDJ-MED-28ec730d-2_1
|
|
COCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.8
± 0.2
|
137 |
ED_-GRI-5b13fbe2-63_1
|
|
Cc1c(nnn1CCCCO[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)C[NH3+] |
−9.7
± 0.2
|
138 |
MIC-UNK-d36ab305-5_1
|
|
CN(C)c1ccc(cc1)N(c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.7
± 0.2
|
139 |
MIC-UNK-50cce87d-11_2
|
|
Cc1cccc2c1c(cnc2)N3CCC[C@H](C3=O)c4cccc(c4)Cl |
−9.7
± 0.2
|
140 |
DAR-DIA-0d514e7d-32_7
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3[C@H]4C[C@H]4CO[C@@H]5[C@@H]3C=C(C=C5)Cl |
−9.7
± 0.2
|
141 |
MAT-POS-f9802937-8_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCNc4c3cc(c(c4)Cl)Cl |
−9.70
± 0.10
|
142 |
MAK-UNK-c749d764-29_5
|
|
c1ccc2c(c1)cncc2N(C(=O)C[C@@H]3CCC[C@@H]([C@H]3O)C(F)F)C(=O)ON |
−9.7
± 0.3
|
143 |
EDG-MED-ba1ac7b9-5_1
|
|
CC[C@@H](CO)[NH+]1CCN(CC1)C(=O)C[C@@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.7
± 0.5
|
144 |
MAK-UNK-8be7dca9-3_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H]3c4cc(ccc4OC[C@@H]3C[NH3+])Cl |
−9.7
± 0.2
|
145 |
MIC-UNK-cdc2493e-8_6
|
|
c1ccc2c(c1)cncc2NC(=O)N(c3cccc(c3)Cl)[C@H]4CC[C@@H]5CCCC[C@H]5C4 |
−9.7
± 0.2
|
146 |
ALP-UNI-8e43a71e-1_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCS(=O)(=O)[N@@]6[C@@H]5CCCC6 |
−9.7
± 0.1
|
147 |
MIC-UNK-cdc2493e-20_1
|
|
CC(=O)N(C)C1CCC(CC1)N(c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.7
± 0.2
|
148 |
JOH-SUS-a69c159d-6_1
|
|
c1ccc2c(c1)c(c(nc2F)F)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.7
± 0.2
|
149 |
ALF-EVA-650655fc-4_5
|
|
C[N@@H+]1CC[C@@H](C1)CCN(c2cc(cc(c2)Cl)O[C@H]3CC(=O)N3)C(=O)Nc4cncc5c4cccc5 |
−9.7
± 0.1
|
150 |
MIC-UNK-5a93dd5f-3_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](c3cccc(c3)Cl)[N@@H+]4CC[C@@H]5CCCC[C@@H]5C4 |
−9.7
± 0.2
|
151 |
MAK-UNK-c749d764-24_3
|
|
CCN(c1cncc2c1cccc2)C(=O)C[C@@H]3CCC[C@H]([C@@H]3O)C(F)F |
−9.6
± 0.3
|
152 |
MAT-POS-3b92565d-3_2
|
|
c1ccc2c(c1)cncc2NC(=O)Cc3cc(cc(c3)Cl)O[C@H]4CC(=O)N4 |
−9.6
± 0.3
|
153 |
RAL-THA-1d44ff04-5_1
|
|
CNC(=O)c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2cccc3 |
−9.6
± 0.4
|
154 |
LON-WEI-5e7d1b3e-56_1
|
|
CC(C)Cn1cc(c2ccccc2c1=O)NC(=O)Nc3ccsc3C(=O)OC |
−9.6
± 0.2
|
155 |
MIC-UNK-0a05c952-2_4
|
|
c1ccc2c(c1)cncc2N3[C@H](CC[C@H](C3=O)c4cccc(c4)Cl)[C@@H]5CO5 |
−9.6
± 0.2
|
156 |
ADA-UCB-dc2b944c-14_1
|
|
C[C@H]1COc2ccc(cc2[C@H]1C(=O)Nc3cncc4c3cccc4)Cl |
−9.6
± 0.2
|
157 |
KAD-UNI-80f122c8-5_2
|
|
C[N@@](C1CCN(CC1)C(=O)C[C@@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)S(=O)(=O)C |
−9.6
± 0.4
|
158 |
MIC-UNK-644c43c7-3_1
|
|
c1ccc2c(c1)cncc2NC(=O)Cc3cc(cc(c3)Cl)CNCC(F)(F)F |
−9.6
± 0.2
|
159 |
VLA-UCB-34f3ed0c-12_1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)CNC3=O |
−9.6
± 0.4
|
160 |
MAK-UNK-f481d203-3_1
|
|
c1ccc(cc1)[C@H](C(=O)Nc2cncc3c2cccc3)[NH3+] |
−9.6
± 0.3
|
161 |
MAT-POS-4223bc15-18_1
|
|
CN(C)C(=O)N1Cc2ccc(cc2[C@@H](C1)C(=O)Nc3cncc4c3cccc4)Cl |
−9.56
± 0.09
|
162 |
RAL-THA-4aa06b95-4_1
|
|
CN(C)C(=O)N1CC[C@@H](c2c1ccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.6
± 0.3
|
163 |
MAK-UNK-c749d764-2_7
|
|
CC[C@@H]1CCC[C@H]([C@H]1O)CC(=O)Nc2cncc3c2cccc3 |
−9.6
± 0.3
|
164 |
MAK-UNK-c749d764-31_6
|
|
CC/C=C(/c1cncc2c1cccc2)\C(=O)C[C@H]3CCC[C@@H]([C@H]3O)C(F)F |
−9.5
± 0.2
|
165 |
ALP-UNI-0676e700-24_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@H]5[C@H](CC(=O)N5)C(F)(F)F |
−9.5
± 0.4
|
166 |
MAT-POS-2492181e-9_1
|
|
CC1CC[NH+](CC1)Cc2ccc(cc2)NC(=O)Nc3cn(c(=O)c4c3cccc4)CC(C)C |
−9.5
± 0.2
|
167 |
ALP-UNI-0676e700-11_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)c5ccc(cc5)CC(=O)N |
−9.5
± 0.3
|
168 |
ALP-POS-e0fe77e5-7_1
|
|
c1ccc2c(c1)cncc2N3CCC[C@]4(C3=O)CCOc5c4cc(cc5)Cl |
−9.5
± 0.3
|
169 |
MIC-UNK-d36ab305-4_2
|
|
CN(C)c1ccc(cc1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.5
± 0.3
|
170 |
PET-UNK-1b92fa34-4_1
|
|
c1cc2cncc(c2cc1F)NC(=O)[C@@H]3CS(=O)(=O)Cc4c3cc(c(c4)F)Cl |
−9.5
± 0.3
|
171 |
MIC-UNK-cdc2493e-22_1
|
|
c1ccc2c(c1)cncc2NC(=O)N(CCn3ccnn3)c4cccc(c4)Cl |
−9.5
± 0.3
|
172 |
MIC-UNK-cdc2493e-5_2
|
|
c1ccc2c(c1)cncc2NC(=O)N(c3cccc(c3)Cl)C4C[C@H]5CCCC[C@@H]5C4 |
−9.5
± 0.3
|
173 |
VLA-UCB-34f3ed0c-6_1
|
|
c1ccc2c(c1)cncc2NC(=O)N(c3cccc(c3)Cl)C(=O)CC4CCCCC4 |
−9.5
± 0.3
|
174 |
MIC-UNK-cdc2493e-21_4
|
|
CC(=O)N(C)[C@H]1CC[C@H](C1)N(c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.5
± 0.2
|
175 |
ALP-UNI-8e43a71e-5_14
|
|
C[C@H]1C[N@@](CC[C@H]1NC(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)S(=O)(=O)C |
−9.5
± 0.2
|
176 |
MIC-UNK-cdc2493e-3_1
|
|
c1ccc(cc1)CCN(c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.5
± 0.3
|
177 |
ALP-POS-e0fe77e5-4_1
|
|
c1ccc2c(c1)cncc2N3CCC[C@@]4(C3=O)CCOc5c4cc(c(c5)Cl)Cl |
−9.5
± 0.2
|
178 |
DAR-DIA-9e4459de-15_1
|
|
c1cc2c(c(c1)NC(=O)CCC(=O)Nc3ccc4c(c3)cncc4NC(=O)[C@@H]5CCOc6c5cc(cc6)Cl)c(n(c2O)[C@@H]7CCC(=O)NC7=O)O |
−9.5
± 0.3
|
179 |
LON-WEI-4d77710c-29_1
|
|
CCOC(=O)Cc1csc(n1)NC(=O)Nc2cn(c(=O)c3c2cccc3)CC(C)C |
−9.5
± 0.2
|
180 |
MIC-UNK-5a93dd5f-7_2
|
|
CC(=O)N(C)[C@H]1CC[N@@H+](C1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.5
± 0.3
|
181 |
DAR-DIA-0d514e7d-31_6
|
|
C[C@H]1CCO[C@@H]2C=CC(=C[C@H]2[C@@H]1C(=O)Nc3cncc4c3cccc4)Cl |
−9.5
± 0.2
|
182 |
LON-WEI-af038623-3_1
|
|
C=CC(=O)Nc1cncc2c1cccc2 |
−9.5
± 0.3
|
183 |
MAK-UNK-ffc90da7-9_1
|
|
C[C@@H]1[C@@H](CCO1)SC[C@@H](C)c2ccc3c(c2)cncc3NC(=O)Cc4cccc(c4)Cl |
−9.5
± 0.3
|
184 |
ERI-UCB-ce40166b-10_1
|
|
c1ccc2c(c1)cncc2CC(=O)Nc3cc(cc(c3)O[C@@H]4CCC(=O)N4)C#N |
−9.5
± 0.2
|
185 |
LAU-MED-88a3970a-14_1
|
|
COCCCc1cc(cc2c1OCC[C@@H]2C(=O)Nc3cncc4c3cccc4)Cl |
−9.5
± 0.2
|
186 |
MAT-POS-4223bc15-26_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H]3C[N@@](Cc4c3cc(cc4)Cl)CC(F)(F)F |
−9.4
± 0.2
|
187 |
KAD-UNI-8a629cb0-2_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)NCC56CC(C5)(CO6)C(=O)N |
−9.4
± 0.4
|
188 |
ALP-POS-966f8da6-1_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H]3CCN(c4c3cc(cc4)Cl)Cc5cnc[nH]5 |
−9.4
± 0.3
|
189 |
DAR-DIA-0cde14eb-50_1
|
|
CC1(CC1)c2cccc(c2)NC(=O)Nc3cncc4c3cccc4 |
−9.4
± 0.2
|
190 |
MAK-UNK-919546f0-4_1
|
|
c1ccc2c(c1)cncc2NC(=O)Cc3ccccc3O |
−9.4
± 0.3
|
191 |
JAG-UCB-706446eb-1_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)NCC(F)(F)F |
−9.4
± 0.4
|
192 |
LON-WEI-4d77710c-7_1
|
|
Cn1cc(c2ccccc2c1=O)NC(=O)NCCC[N@@H+]3CCc4ccccc4C3 |
−9.4
± 0.2
|
193 |
MAT-POS-e69ad64a-1_2
|
|
C=CC(=O)N(c1cncc2c1cccc2)C(=O)[C@H]3CCNc4c3cc(cc4)Cl |
−9.4
± 0.4
|
194 |
MIC-UNK-9582b2c5-2_1
|
|
CC(=O)N1CC[C@@H]2[C@@H](C1)C[C@@H](C(=O)N2c3cccc(c3)Cl)c4cncc5c4cccc5 |
−9.4
± 0.5
|
195 |
MAK-UNK-c749d764-15_3
|
|
C[C@@H](N(c1cncc2c1cccc2)C(=O)C[C@H]3CCC[C@@H]([C@@H]3O)C(F)F)OCC4CCCCC4 |
−9.4
± 0.2
|
196 |
EDJ-MED-28ec730d-3_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OC5CCOCC5 |
−9.4
± 0.3
|
197 |
MAT-POS-53907a1c-3_2
|
|
c1ccc2c(c1)cncc2NC(=O)N(CCC3CCCCC3)c4cc(cc(c4)Cl)O[C@H]5CC(=O)N5 |
−9.41
± 0.10
|
198 |
VLA-UCB-05e51b3f-1_1
|
|
CC(=O)N1CC[NH+](CC1)CC(=O)Nc2cncc3c2cccc3 |
−9.4
± 0.3
|
199 |
RAL-THA-e002e396-1_1
|
|
CS(=O)(=O)C[C@@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.4
± 0.2
|
200 |
ALP-POS-2da19ca7-3_1
|
|
Cn1cnc2c(c1=O)CCN(C2)C(=O)C[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−9.4
± 0.3
|