Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
801 |
EN300-217494_1_1 |
|
C[C@@]([C@@H]1CCOC1)(C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−11.5
± 0.3
|
802 |
EN300-52382_1_1 |
|
CN(C)C(=O)Cn1cc(nn1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
803 |
EN300-212814_1_3 |
|
C[C@@H]1CN(C[C@H](O1)CCO)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
804 |
EN300-50561_1_2 |
|
Cc1nnc2n1C[C@H](CC2)C(=O)N[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−11.5
± 0.3
|
805 |
EN300-399606_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc6n(n5)CCC[C@@H]6O |
−11.5
± 0.2
|
806 |
EN300-6736413_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCO[C@@H]5CCNC5=O |
−11.5
± 0.2
|
807 |
EN300-6736413_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCO[C@@H]5CCNC5=O |
−11.5
± 0.2
|
808 |
EN300-298184_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N[C@@H]5CCNC5=O |
−11.5
± 0.3
|
809 |
VLA-UCB-50c39ae8-10_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC5CCCCC5 |
−11.5
± 0.2
|
810 |
EN300-6736413_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCO[C@H]5CCNC5=O |
−11.5
± 0.3
|
811 |
EN300-6736413_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCO[C@H]5CCNC5=O |
−11.5
± 0.3
|
812 |
EN300-7432415_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@@H]5C6(CCC6)OC(=O)N5 |
−11.5
± 0.3
|
813 |
EN300-1273249_1_1 |
|
CO[C@@H]1COC[C@H]1n2cc(nn2)C(=O)N[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−11.5
± 0.4
|
814 |
EN300-219496_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCCN(C5)S(=O)(=O)N |
−11.5
± 0.5
|
815 |
EN300-152418_1_1 |
|
Cn1cncc1CC(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
816 |
EN300-189563_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCCC5CS(=O)(=O)C5 |
−11.5
± 0.3
|
817 |
EN300-61694_1_1 |
|
Cn1ncc(n1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.2
|
818 |
EN300-6277108_1_1 |
|
CO[C@@H]([C@@H]1CCCO1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
819 |
EN300-157776_1_3 |
|
C[C@@H]1CN(C[C@H](O1)CO)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
820 |
EN300-378044_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CC=CCO5 |
−11.5
± 0.3
|
821 |
EN300-6494158_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OC[C@H]5C[C@@H](CO5)CO |
−11.5
± 0.3
|
822 |
EN300-205616_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCOC[C@@H]5c6[nH]cnn6 |
−11.5
± 0.3
|
823 |
EN300-301925_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@@]5(CCCOC5)C#N |
−11.5
± 0.3
|
824 |
EN300-68618_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cocn5 |
−11.5
± 0.2
|
825 |
EN300-1726277_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@H](n5cccn5)F |
−11.5
± 0.3
|
826 |
DAR-DIA-5ff57136-18_1
|
|
c1ccc2c(c1)cncc2N(C(=O)[C@@H]3CCOc4c3cc(cc4)Cl)N=C=S |
−11.5
± 0.1
|
827 |
JOH-SUS-a69c159d-7_1
|
|
c1cc2c(cc1F)c(c(nc2F)F)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−11.51
± 0.06
|
828 |
EN300-203402_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ccc6c(n5)[nH]c(=O)[nH]6 |
−11.5
± 0.3
|
829 |
EN300-297927_3_1 |
|
CC(C)(C)n1nc(nn1)CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.4
|
830 |
EN300-120586_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCC(=O)NCC(F)F |
−11.5
± 0.3
|
831 |
EN300-54417_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CNC(=O)c5cccc(c5)O |
−11.5
± 0.3
|
832 |
EN300-651665_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5C[C@@H]6[C@H]5CCO6 |
−11.5
± 0.3
|
833 |
EN300-95698_3_2 |
|
C[C@H]1CC(=O)NC[C@@H]1C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.2
|
834 |
EN300-180532_1_1 |
|
C[C@@H]1CN(CCS(=O)(=O)C1)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.4
|
835 |
EN300-863933_1_2 |
|
C[C@H](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)N(C)C(=O)C |
−11.5
± 0.3
|
836 |
EN300-7464289_1_2 |
|
C[C@](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)(C(=O)OC)F |
−11.5
± 0.3
|
837 |
EN300-74029_1_1 |
|
C[C@@H]1CC(=O)NCCN1C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
838 |
EN300-80083_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCCCC(=O)N5 |
−11.5
± 0.3
|
839 |
EN300-6497444_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cnn6c5OC[C@H](C6)O |
−11.5
± 0.2
|
840 |
EN300-171766_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCc5n[nH]c(=O)s5 |
−11.5
± 0.2
|
841 |
EN300-149013_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5c([nH]nn5)Cl |
−11.5
± 0.3
|
842 |
EN300-56202_3_2 |
|
CC(=O)N1CSC[C@H]1C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.4
|
843 |
EN300-306316_4_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCCOCc5[nH]cnn5 |
−11.5
± 0.3
|
844 |
EN300-70489_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCO[C@@H](C5)C#N |
−11.5
± 0.3
|
845 |
EN300-658865_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc([nH]n5)CO |
−11.5
± 0.3
|
846 |
EN300-153257_1_1 |
|
CC(C)[C@@H](CO)C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.5
± 0.3
|
847 |
EN300-6760290_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5[C@@H]6CC[C@H]([C@H]5CC[C@H]6O)O |
−11.5
± 0.3
|
848 |
EN300-1718364_3_1 |
|
CC1(CS(=O)(=O)C1)C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
849 |
EN300-731622_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C[C@@H]5COCCO5 |
−11.5
± 0.3
|
850 |
EN300-53423_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCOC5 |
−11.5
± 0.3
|
851 |
EN300-259062_1_2 |
|
CNC(=O)C[C@]1(CCCN(C1)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−11.5
± 0.4
|
852 |
EN300-219531_3_1 |
|
CCC[C@@H](C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O |
−11.5
± 0.3
|
853 |
EN300-51257_1_2 |
|
C[C@H](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)OC |
−11.5
± 0.2
|
854 |
EN300-6744028_1_4 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CC6CC5[C@H]([C@@H]6O)O |
−11.5
± 0.3
|
855 |
EN300-249421_3_2 |
|
C[C@H]([C@@H]1CCC(=O)N1)C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
856 |
EN300-6487407_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOC[C@@H]5[C@H](CC(=O)O5)O |
−11.5
± 0.3
|
857 |
EN300-269453_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@@H]5CCc6nnnn6C5 |
−11.5
± 0.3
|
858 |
EN300-7537194_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ccn6cnnc6c5 |
−11.5
± 0.2
|
859 |
EN300-191904_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CCn5cnnn5 |
−11.5
± 0.3
|
860 |
EN300-182665_1_1 |
|
Cc1nc(on1)[C@H]2C[C@@H](CN2C(=O)C[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6)O |
−11.5
± 0.3
|
861 |
EN300-6473108_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc6cccnn6n5 |
−11.5
± 0.2
|
862 |
EN300-149975_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C5(CCC5)CO |
−11.5
± 0.2
|
863 |
EN300-249764_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@H](C5CCC5)O |
−11.5
± 0.4
|
864 |
EN300-343562_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC[C@H]([C@H]5CO)CO |
−11.5
± 0.4
|
865 |
EN300-7385329_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5Cc6nccn6C5 |
−11.5
± 0.3
|
866 |
EN300-113234_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CC(=O)OC5 |
−11.5
± 0.3
|
867 |
EN300-114082_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C5(CC5)C#N |
−11.5
± 0.2
|
868 |
EN300-120436_3_1 |
|
Cn1cnn(c1=O)CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
869 |
EN300-6487680_1_1 |
|
Cc1nnn(n1)CC(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.3
|
870 |
EN300-91609_1_3 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCO[C@@H]6[C@H]5C6 |
−11.5
± 0.3
|
871 |
EN300-1726277_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H](n5cccn5)F |
−11.5
± 0.2
|
872 |
EN300-80083_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@@H]5CCCCC(=O)N5 |
−11.5
± 0.3
|
873 |
EN300-40225_1_1 |
|
Cc1c(cnn1CCO)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.5
± 0.4
|
874 |
EN300-06654_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cncn5 |
−11.5
± 0.2
|
875 |
EN300-06654_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cncn5 |
−11.5
± 0.2
|
876 |
EN300-6491117_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)Cc5cnco5 |
−11.5
± 0.3
|
877 |
EN300-6738887_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5C6CCC5[C@H](CC[C@H]6O)O |
−11.5
± 0.3
|
878 |
EN300-246248_2_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)COC[C@H]5CCNC5=O |
−11.5
± 0.3
|
879 |
EN300-783124_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@@H]([C@@H]5CCOC5)F |
−11.5
± 0.2
|
880 |
EN300-95507_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc(on5)CO |
−11.5
± 0.2
|
881 |
EN300-341337_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@@]56CCO[C@@H]5CCOC6 |
−11.4
± 0.3
|
882 |
EN300-7089802_3_1 |
|
C[C@@H]([C@@H](C)O)C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.4
± 0.3
|
883 |
EN300-2908024_3_1 |
|
CC[C@@](C)(C(=O)N)C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.4
± 0.3
|
884 |
EN300-7473354_3_1 |
|
Cc1ncn(n1)CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.4
± 0.4
|
885 |
EN300-129441_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cccc6n5ncn6 |
−11.4
± 0.2
|
886 |
EN300-98143_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5c(cn[nH]5)F |
−11.4
± 0.2
|
887 |
EN300-262604_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cnc(n5)C(=O)N |
−11.4
± 0.3
|
888 |
EN300-39405_3_2 |
|
C[C@H](C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)S(=O)(=O)C |
−11.4
± 0.4
|
889 |
EN300-222969_1_1 |
|
CN1C[C@@H](OC1=O)CO[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.4
± 0.4
|
890 |
EN300-100916_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5nccn5 |
−11.4
± 0.3
|
891 |
EN300-37123_1_1 |
|
Cn1cc(c(=O)[nH]c1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.4
± 0.3
|
892 |
EN300-141695_1_2 |
|
CN1CC[C@H](C1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.4
± 0.2
|
893 |
EN300-6491316_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ccc6cnnn6c5 |
−11.4
± 0.2
|
894 |
EN300-7459545_3_2 |
|
CN(C)C[C@](C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)(C(F)(F)F)O |
−11.4
± 0.6
|
895 |
EN300-143449_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CCCN(=O)=O |
−11.4
± 0.2
|
896 |
EN300-50009_3_1 |
|
COC(=O)NCC(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.4
± 0.3
|
897 |
EN300-90225_4_1 |
|
Cn1nc(nn1)COCCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.4
± 0.3
|
898 |
EN300-10895_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCC(=O)NCCC#N |
−11.4
± 0.2
|
899 |
EN300-123614_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C5(CC5)NC(=O)N |
−11.4
± 0.4
|
900 |
EN300-69162_3_1 |
|
C[C@@H](COC)C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.4
± 0.3
|