Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
5001 |
EN300-108022_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)NCCn5cnnn5 |
−9.6
± 0.3
|
5002 |
EN300-187998_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)N5CCC6(C5)CC(=O)NC6 |
−9.6
± 0.3
|
5003 |
EN300-68203_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C[C@@H]5CCC(=O)N5 |
−9.6
± 0.2
|
5004 |
EN300-383824_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)c5cc6c([nH]c5=O)CCOC6 |
−9.6
± 0.4
|
5005 |
EN300-1268020_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCN(CC5)Cc6[nH]nnn6 |
−9.6
± 0.4
|
5006 |
EN300-92662_2_1 |
|
Cn1c(ccn1)CCC(=O)NC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.3
|
5007 |
BEN-DND-c852c98b-5_1
|
|
CS(=O)(=O)c1ccc2cncc(c2c1)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−9.57
± 0.08
|
5008 |
EN300-74856_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N[C@H]5CCCS(=O)(=O)C5 |
−9.6
± 0.3
|
5009 |
EN300-252113_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCS(=O)(=O)[C@H]6[C@@H]5CCOC6 |
−9.6
± 0.6
|
5010 |
EN300-217499_1_1 |
|
C[C@@](C1CCOCC1)(C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−9.6
± 0.3
|
5011 |
EN300-305984_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)c5cccn6c5nnn6 |
−9.6
± 0.3
|
5012 |
EN300-313267_1_1 |
|
CN1CCC[C@@H](C1=O)NC(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.2
|
5013 |
EN300-313267_1_1 |
|
CN1CCC[C@@H](C1=O)NC(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.2
|
5014 |
EN300-183231_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCCc5[nH]nnn5 |
−9.6
± 0.3
|
5015 |
EN300-7355979_1_1 |
|
Cn1cnc2c(c1=O)[nH]nc2C(=O)N[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−9.6
± 0.3
|
5016 |
DAR-DIA-23e5a6a0-8_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCOc4c3cc(cc4C[C@@H]5CC6(N5)COC6)Cl |
−9.6
± 0.3
|
5017 |
EN300-1692359_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)NC[C@]5(CC[C@@H]5CO)CO |
−9.6
± 0.3
|
5018 |
EN300-747207_2_1 |
|
CC(C)(CNC(=O)N)NC(=O)CC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.6
± 0.3
|
5019 |
EN300-1708899_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)NC[C@@H]5C[C@@H](CCO5)O |
−9.6
± 0.3
|
5020 |
EN300-6736394_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)C56CC(CCO5)OC6 |
−9.6
± 0.2
|
5021 |
EN300-70656_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)NCC5(CCC5)O |
−9.6
± 0.3
|
5022 |
EN300-365650_1_1 |
|
C[C@@H](C1CN(C1)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−9.6
± 0.2
|
5023 |
EN300-1722713_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CC6(C5)CC(=O)NC6 |
−9.6
± 0.3
|
5024 |
EN300-96159_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)Cc5[nH]cnn5 |
−9.6
± 0.3
|
5025 |
EN300-255990_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cnn6c5ncc(c6)C#N |
−9.6
± 0.3
|
5026 |
EN300-316193_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)N5C[C@H]6COC(=O)[C@H]6C5 |
−9.6
± 0.3
|
5027 |
EN300-190026_1_4 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N[C@H](CO)[C@H]5CCCO5 |
−9.6
± 0.4
|
5028 |
EN300-749499_2_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@H](C5(CCOCC5)O)O |
−9.6
± 0.3
|
5029 |
EN300-6498726_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)N[C@H](CO)CF |
−9.6
± 0.5
|
5030 |
EN300-11300_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCc5cc(=O)[nH]c(=O)[nH]5 |
−9.6
± 0.3
|
5031 |
EN300-259063_2_2 |
|
CC(=O)N1CCC[C@](C1)(CC(=O)NC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−9.6
± 0.4
|
5032 |
EN300-78135_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)C(=O)NC5CC5 |
−9.6
± 0.3
|
5033 |
EN300-304051_2_1 |
|
Cn1cc(nn1)CN(C)C(=O)CC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.2
|
5034 |
EN300-51028_4_1 |
|
CC(C)S(=O)(=O)CC(=O)NCCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.6
± 0.4
|
5035 |
EN300-1605566_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CN6CCN5CC6 |
−9.6
± 0.3
|
5036 |
EN300-706065_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)C(C5(CCOCC5)O)(F)F |
−9.6
± 0.4
|
5037 |
EN300-746187_2_1 |
|
Cc1nc2n(n1)C[C@@H](CC2)C(=O)NC[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−9.6
± 0.3
|
5038 |
EN300-138170_1_1 |
|
C[C@@H]1CCN(C1)C(=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.2
|
5039 |
EN300-1387104_2_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@H]5CCS5(=O)=O |
−9.6
± 0.4
|
5040 |
EN300-1709315_3_2 |
|
C[C@]1(CCCNS1(=O)=O)C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.4
|
5041 |
EN300-36851_4_1 |
|
C[C@@H]1C[C@@H]1C(=O)NCCC(=O)NCCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.4
|
5042 |
EN300-260262_1_1 |
|
Cn1cc(nn1)CCNC(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.2
|
5043 |
EN300-1605433_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC6(C5)CCNC6=O |
−9.6
± 0.4
|
5044 |
EN300-43047_3_1 |
|
CC(=O)N[C@@H](CC=C)C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.6
± 0.3
|
5045 |
EN300-204935_2_1 |
|
Cn1ncc(n1)C(=O)COC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.3
|
5046 |
EN300-210553_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC[C@@](C5)(C(=O)N)O |
−9.6
± 0.3
|
5047 |
EN300-210553_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC[C@@](C5)(C(=O)N)O |
−9.6
± 0.3
|
5048 |
EN300-366852_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CC[C@@H](C5)c6[nH]nnn6 |
−9.6
± 0.4
|
5049 |
EN300-42591_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)CNC(=O)NC5CC5 |
−9.6
± 0.3
|
5050 |
EN300-109535_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)C[C@@H]5CC(=O)OC5 |
−9.6
± 0.3
|
5051 |
EN300-39005_1_1 |
|
CN(CC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)C(=O)OC |
−9.6
± 0.3
|
5052 |
EN300-1273172_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)c5cnc(cn5)C(=O)N |
−9.6
± 0.3
|
5053 |
EN300-305282_3_1 |
|
COC[C@@H](C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)OC |
−9.6
± 0.4
|
5054 |
EN300-256798_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)N[C@@H]5CCc6nnnn6CC5 |
−9.6
± 0.3
|
5055 |
EN300-55744_1_1 |
|
CCCC[C@@H](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)NC(=O)N |
−9.6
± 0.3
|
5056 |
EN300-100180_3_2 |
|
CC(=O)N1CC[C@H](C1)C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.6
± 0.5
|
5057 |
EN300-118045_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cnc([nH]c5=O)C6CC6 |
−9.5
± 0.4
|
5058 |
EN300-6494158_4_4 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCCOC[C@H]5C[C@H](CO5)CO |
−9.5
± 0.3
|
5059 |
EN300-43972_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)NCc5[nH]cnn5 |
−9.5
± 0.3
|
5060 |
EN300-43972_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)NCc5[nH]cnn5 |
−9.5
± 0.3
|
5061 |
EN300-259060_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC[C@@](C5)(CC(=O)N)O |
−9.5
± 0.4
|
5062 |
EN300-1911992_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OC[C@H]([C@@H]5CCOC5)O |
−9.5
± 0.3
|
5063 |
EN300-02623_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)Nc5[nH]c(nn5)CCCO |
−9.5
± 0.3
|
5064 |
EN300-116885_2_1 |
|
Cc1c(nc(c(=O)[nH]1)C(=O)NC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)C |
−9.5
± 0.3
|
5065 |
EN300-717276_2_1 |
|
CCn1cc(nn1)CC(=O)NC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.5
± 0.3
|
5066 |
EN300-211403_1_1 |
|
CN(C(=O)C[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)C5(CC5)CO |
−9.5
± 0.4
|
5067 |
EN300-7438451_2_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)N[C@H]5CCn6c(nnn6)C5 |
−9.5
± 0.3
|
5068 |
EN300-37195_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCC(=O)N[C@@H]5CCCCNC5=O |
−9.5
± 0.2
|
5069 |
EN300-36931_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)NCC5(CCOCC5)C(=O)N |
−9.5
± 0.3
|
5070 |
EN300-310254_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N[C@H]5C(=O)NCC56CCOCC6 |
−9.5
± 0.4
|
5071 |
EN300-6482296_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CO[C@@H]6[C@@H]5COC6 |
−9.5
± 0.2
|
5072 |
EN300-1723663_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@H]5CCN(C(=O)C5)CCO |
−9.5
± 0.3
|
5073 |
EN300-81629_2_1 |
|
Cc1nncn1CCNC(=O)CC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.5
± 0.3
|
5074 |
EN300-331828_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)O[C@@H]5COC[C@H]5O |
−9.5
± 0.2
|
5075 |
EN300-63781_1_1 |
|
Cc1c2c(c(=O)n(nc2C(=O)N[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6)C)no1 |
−9.5
± 0.3
|
5076 |
EN300-199359_3_1 |
|
CC(C)[C@@H](C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O |
−9.5
± 0.3
|
5077 |
EN300-7430501_2_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@H]5CCn6c(cnn6)C5 |
−9.5
± 0.3
|
5078 |
EN300-7430501_2_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@H]5CCn6c(cnn6)C5 |
−9.5
± 0.3
|
5079 |
EN300-02067_2_2 |
|
C[C@H](COC)NC(=O)COC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.5
± 0.3
|
5080 |
EN300-04492_3_1 |
|
COCCCNC(=O)COCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.5
± 0.3
|
5081 |
EN300-6504697_4_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCCOC[C@H]5CC6(CC6)S(=O)(=O)N5 |
−9.5
± 0.4
|
5082 |
EN300-70064_4_1 |
|
CNC(=O)C1(CCC1)C(=O)NCCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.5
± 0.4
|
5083 |
EN300-46832_2_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)COCC(=O)NC[C@H]5CCOC5 |
−9.5
± 0.3
|
5084 |
EN300-318305_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C5CC6(C5)CS(=O)(=O)C6 |
−9.5
± 0.3
|
5085 |
EN300-181492_2_1 |
|
C=C[C@@H](C(=O)NC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O |
−9.5
± 0.3
|
5086 |
EN300-48886_2_2 |
|
CC(=O)N[C@H]1CCCN(C1)C(=O)COC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.5
± 0.3
|
5087 |
EN300-182084_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CNC(=O)c5cscn5 |
−9.5
± 0.3
|
5088 |
EN300-185729_2_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@H]5CCc6c(nn[nH]6)C5 |
−9.5
± 0.5
|
5089 |
EN300-6733147_1_1 |
|
C[C@@H]1CCNC(=O)[C@@H]1CNC(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.5
± 0.3
|
5090 |
EN300-1081277_3_1 |
|
CNC(=O)CCC(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.5
± 0.3
|
5091 |
EN300-366050_2_2 |
|
CC[C@H](Cn1cc(nn1)C(=O)NC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−9.5
± 0.4
|
5092 |
EN300-1699100_2_1 |
|
CN(c1[nH]cnn1)C(=O)CC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.5
± 0.3
|
5093 |
EN300-322100_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)c5ccnc6n5ncc6 |
−9.5
± 0.3
|
5094 |
EN300-18074_1_1 |
|
CC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−9.5
± 0.2
|
5095 |
EN300-116234_4_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCCNC(=O)[C@H]5CCCO5 |
−9.5
± 0.4
|
5096 |
EN300-151423_4_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCCNC(=O)CC5(CCOCC5)O |
−9.5
± 0.3
|
5097 |
EN300-6478526_2_1 |
|
CNC(=O)N1CCC(CC1)C(=O)NC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−9.5
± 0.3
|
5098 |
EN300-67191_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CCN5CCCC5=O |
−9.5
± 0.3
|
5099 |
EN300-6735421_4_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCCOCC5(CN(C5)C6CC6)CO |
−9.5
± 0.5
|
5100 |
EN300-155498_4_1 |
|
CC(=C)[C@H](CC(=O)NCCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O |
−9.5
± 0.2
|