Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
401 |
EN300-114133_1_1 |
|
CCC(=O)N1CC[C@@H](C1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.4
|
402 |
EN300-220676_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C[C@@H]5CCCS(=O)(=O)C5 |
−12.0
± 0.3
|
403 |
EN300-62574_2_1 |
|
Cn1c(nnn1)COC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.2
|
404 |
EN300-1074262_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cccn6c5cnn6 |
−12.0
± 0.3
|
405 |
EN300-658559_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C5(CC5)n6ccnn6 |
−12.0
± 0.3
|
406 |
EN300-301925_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@]5(CCCOC5)C#N |
−12.0
± 0.3
|
407 |
EN300-21221_1_1 |
|
Cc1ccn2c(n1)nc(n2)C(=O)N[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−12.0
± 0.2
|
408 |
EN300-370792_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N(CCO)c5cnccn5 |
−12.0
± 0.3
|
409 |
EN300-212266_1_1 |
|
CC(C)C(=O)N[C@@H](CO)C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−12.0
± 0.4
|
410 |
EN300-6277108_3_4 |
|
CO[C@H]([C@H]1CCCO1)C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.3
|
411 |
EN300-20980_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cnnn5 |
−12.0
± 0.2
|
412 |
EN300-225560_1_1 |
|
CCn1c(cnn1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.2
|
413 |
EN300-201551_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5COCCN5CC(F)(F)F |
−12.0
± 0.4
|
414 |
EN300-7435929_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ncc6c(n5)CCOC6 |
−12.0
± 0.3
|
415 |
EN300-108413_1_2 |
|
C[C@H](CC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)C(=O)OC |
−12.0
± 0.2
|
416 |
EN300-45182_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CCCN5CCOC5=O |
−12.0
± 0.3
|
417 |
EN300-237561_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5c(=O)cccn5 |
−12.0
± 0.3
|
418 |
EN300-60514_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)Cn5cc(cn5)S(=O)(=O)N |
−12.0
± 0.4
|
419 |
EN300-7501017_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5[C@@H]6[C@H]5C(=O)NC6 |
−12.0
± 0.2
|
420 |
EN300-180069_1_1 |
|
Cn1c(c(cn1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)S(=O)(=O)C |
−12.0
± 0.3
|
421 |
EN300-69811_1_1 |
|
Cn1cccc(c1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.3
|
422 |
EN300-28894_1_1 |
|
Cc1c(nn(c(=O)c1C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)C)C |
−12.0
± 0.2
|
423 |
EN300-1248064_1_1 |
|
CC(C)(C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)n5cnnn5 |
−12.0
± 0.3
|
424 |
EN300-260816_3_2 |
|
CN1CC[C@H](C1=O)COCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.3
|
425 |
EN300-1178005_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc(on5)C#N |
−12.0
± 0.2
|
426 |
VLA-UCB-50c39ae8-8_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCOc4c3cc(cc4O[C@@H]5CC(=O)N5)Cl |
−12.0
± 0.2
|
427 |
EN300-1301381_3_1 |
|
COC[C@@]1(CCCO1)C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.3
|
428 |
EN300-64193_3_1 |
|
Cc1nnc(o1)CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.3
|
429 |
EN300-202922_3_2 |
|
C[C@H]([C@@](C)(C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O)O |
−12.0
± 0.4
|
430 |
EN300-169955_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5[C@@H](CC(=O)N5)C(F)(F)F |
−12.0
± 0.3
|
431 |
EN300-143449_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)CCCN(=O)=O |
−12.0
± 0.3
|
432 |
EN300-78753_3_1 |
|
CC1(COC1)C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.3
|
433 |
EN300-107267_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCO[C@@H]5CCCNC5=O |
−12.0
± 0.3
|
434 |
EN300-120820_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cn[nH]c5=O |
−12.0
± 0.2
|
435 |
EN300-113112_2_1 |
|
Cn1cnnc1COC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.2
|
436 |
EN300-1600517_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOC[C@@H](CO)F |
−12.0
± 0.3
|
437 |
EN300-94900_3_1 |
|
CS(=O)(=O)Cc1nc(on1)COCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.4
|
438 |
EN300-148421_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@]5(CCOC5)O |
−12.0
± 0.3
|
439 |
EN300-109540_3_1 |
|
C[C@@H](c1cn(nn1)CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−12.0
± 0.4
|
440 |
EN300-80230_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ncccn5 |
−11.9
± 0.2
|
441 |
EN300-80230_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ncccn5 |
−11.9
± 0.2
|
442 |
EN300-6745081_1_1 |
|
C[C@@]1(CCCCNC1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.4
|
443 |
EN300-36158_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5COCCO5 |
−11.9
± 0.2
|
444 |
EN300-133128_1_1 |
|
CN(C)S(=O)(=O)CC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.9
± 0.3
|
445 |
EN300-220194_1_4 |
|
C[C@H]([C@H](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O)OC |
−11.9
± 0.2
|
446 |
EN300-248883_1_1 |
|
COC[C@@]1(CCOC1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.3
|
447 |
EN300-1726277_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H](n5cccn5)F |
−11.9
± 0.3
|
448 |
EN300-123589_1_1 |
|
CC(C)(C)S(=O)(=O)CC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.9
± 0.2
|
449 |
EN300-6729747_1_1 |
|
Cc1nnc2n1C[C@@H](C2)C(=O)N[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−11.9
± 0.3
|
450 |
EN300-175425_1_2 |
|
CC[C@H](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)C(=O)OC |
−11.9
± 0.3
|
451 |
EN300-7431629_3_2 |
|
Cc1nnc2n1CC[C@]2(C)C(=O)NCC[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−11.9
± 0.3
|
452 |
EN300-7430501_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CCn6c(cnn6)C5 |
−11.9
± 0.3
|
453 |
EN300-7430501_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CCn6c(cnn6)C5 |
−11.9
± 0.3
|
454 |
EN300-341337_3_3 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@@]56CCO[C@H]5CCOC6 |
−11.9
± 0.3
|
455 |
EN300-1387145_1_1 |
|
CS(=O)(=O)[C@@H]1CCC[C@@H]1C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.3
|
456 |
EN300-210552_3_2 |
|
CC(=O)N1CCC[C@](C1)(C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−11.9
± 0.5
|
457 |
EN300-21009_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCCO5 |
−11.9
± 0.2
|
458 |
EN300-6764836_1_3 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CC6[C@H]([C@@H](C5O6)O)O |
−11.9
± 0.3
|
459 |
EN300-6482296_1_8 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CO[C@H]6[C@H]5COC6 |
−11.9
± 0.3
|
460 |
EN300-10747_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CN5CSCC5=O |
−11.9
± 0.2
|
461 |
EN300-6494158_1_4 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OC[C@H]5C[C@H](CO5)CO |
−11.9
± 0.3
|
462 |
EN300-1700760_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C5CC6(C5)CC(=O)N6 |
−11.9
± 0.3
|
463 |
EN300-14458_3_2 |
|
C[C@H](C(=O)N(C)C)OCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.9
± 0.3
|
464 |
EN300-6744028_1_3 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CC6CC5[C@H]([C@@H]6O)O |
−11.9
± 0.3
|
465 |
EN300-702756_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CS(=O)(=O)CC(=O)N5 |
−11.9
± 0.2
|
466 |
EN300-245265_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CCCn5cnc(n5)C#N |
−11.9
± 0.4
|
467 |
EN300-20375_1_1 |
|
COCCOCC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.9
± 0.2
|
468 |
EN300-1719432_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5nc(nn5)C6CC6 |
−11.9
± 0.3
|
469 |
EN300-181492_1_2 |
|
C=C[C@H](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O |
−11.9
± 0.2
|
470 |
EN300-79180_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H](C5CCOCC5)O |
−11.9
± 0.3
|
471 |
EN300-6733459_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@]56CCCN5S(=O)(=O)CC6 |
−11.9
± 0.5
|
472 |
EN300-184266_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CC(=O)N5 |
−11.9
± 0.3
|
473 |
EN300-72730_2_2 |
|
C[C@H](C#N)C(=O)NC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.9
± 0.2
|
474 |
EN300-150212_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc(n[nH]5)F |
−11.9
± 0.2
|
475 |
EN300-209048_1_2 |
|
CN1CC[C@H](C1=O)N(C)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.3
|
476 |
EN300-209048_1_2 |
|
CN1CC[C@H](C1=O)N(C)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.3
|
477 |
EN300-83864_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C5CCC(CC5)S(=O)(=O)N |
−11.9
± 0.4
|
478 |
EN300-300217_1_4 |
|
C/C=C/[C@H](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O |
−11.9
± 0.2
|
479 |
EN300-127197_3_1 |
|
COc1cc(on1)CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.4
|
480 |
EN300-258477_3_1 |
|
C[C@@H](C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)OC |
−11.9
± 0.3
|
481 |
EN300-1719432_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)Cn5nc(nn5)C6CC6 |
−11.9
± 0.3
|
482 |
EN300-393121_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc6c(=O)[nH]ccn6n5 |
−11.9
± 0.3
|
483 |
EN300-70431_1_1 |
|
COc1c(c(ncn1)OC)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.2
|
484 |
EN300-6494474_1_1 |
|
Cn1cnnc1CC(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.2
|
485 |
EN300-171766_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCc5n[nH]c(=O)s5 |
−11.9
± 0.3
|
486 |
EN300-132157_2_1 |
|
C[C@@]1(CC(=O)NC1)C(=O)NC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.3
|
487 |
EN300-270422_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5C[C@H](C[C@@H](C5)F)O |
−11.9
± 0.3
|
488 |
EN300-113218_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)CS[C@@H]5CCOC5=O |
−11.9
± 0.3
|
489 |
EN300-97758_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)CCF |
−11.9
± 0.2
|
490 |
EN300-123416_1_1 |
|
CCCn1cc(nn1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.3
|
491 |
EN300-7461217_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5C[C@H]([C@@H](C5)F)O |
−11.9
± 0.3
|
492 |
EN300-1789253_1_1 |
|
Cn1cc(nn1)c2cc(no2)C(=O)N[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−11.9
± 0.2
|
493 |
EN300-6729572_1_6 |
|
C[C@H]([C@@H]1C[C@H]1C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−11.9
± 0.2
|
494 |
EN300-25960_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C5(CCCC5)O |
−11.9
± 0.3
|
495 |
EN300-245264_1_2 |
|
CC[C@H](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)n5cnc(n5)C#N |
−11.9
± 0.3
|
496 |
EN300-7444950_3_1 |
|
COc1cc(ncn1)CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.3
|
497 |
EN300-1932780_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@@H](C(F)F)O |
−11.9
± 0.3
|
498 |
EN300-172179_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CN5CCOC5=O |
−11.9
± 0.3
|
499 |
EN300-1138792_1_1 |
|
Cn1cnnc1CCC(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.2
|
500 |
EN300-66845_3_2 |
|
COC(=O)N1CCC[C@H]1C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.9
± 0.3
|