Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
301 |
EN300-214172_1_1 |
|
Cn1cnc(n1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.2
± 0.2
|
302 |
VLA-UCB-34f3ed0c-21_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)C(=O)CC[C@H]5CC(=O)NC5 |
−12.2
± 0.4
|
303 |
EN300-208236_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@H]5CCCc6c5nn[nH]6 |
−12.2
± 0.4
|
304 |
EN300-204133_1_1 |
|
COC1(CCOCC1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.2
± 0.3
|
305 |
EN300-19926_4_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCCNC(=O)CC#N |
−12.2
± 0.3
|
306 |
EN300-23942_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cccn5 |
−12.2
± 0.2
|
307 |
EN300-1601684_1_1 |
|
CC1([C@@H](OCCO1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)C |
−12.2
± 0.3
|
308 |
EN300-245098_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC[C@@H]5C(=O)N |
−12.2
± 0.3
|
309 |
EN300-174668_1_2 |
|
CO[C@]1(CCOC1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.2
± 0.4
|
310 |
EN300-261210_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@@]5(CCOC5)C#N |
−12.2
± 0.3
|
311 |
EN300-268087_1_1 |
|
CC(C)(C)n1nc(nn1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.2
± 0.3
|
312 |
EN300-198515_1_2 |
|
C[C@H](C(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)n5cnc(n5)C#N |
−12.2
± 0.3
|
313 |
EN300-254883_1_1 |
|
Cc1c(non1)CC(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.2
± 0.2
|
314 |
EN300-114082_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)C5(CC5)C#N |
−12.2
± 0.2
|
315 |
EN300-27341_1_1 |
|
CS(=O)(=O)N1CCC[C@@H](C1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.2
± 0.5
|
316 |
EN300-7540889_1_1 |
|
COc1ccc(nn1)CC(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.2
± 0.2
|
317 |
EN300-1589101_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cc5c[nH]nc5 |
−12.2
± 0.3
|
318 |
VLA-UCB-551c2366-1_1
|
|
CN(C)c1ccc(cc1)[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.2
± 0.2
|
319 |
EN300-315238_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@H]5CC[C@H](O5)C(=O)N |
−12.2
± 0.4
|
320 |
DAR-DIA-5ff57136-13_1
|
|
C#CCN(c1cncc2c1cccc2)C(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−12.2
± 0.1
|
321 |
EN300-1662365_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCc6ncnn6C5 |
−12.2
± 0.3
|
322 |
EN300-1696962_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCCCn5cnnn5 |
−12.2
± 0.3
|
323 |
EN300-2910941_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cc(nn5)C(F)(F)F |
−12.2
± 0.3
|
324 |
EN300-94945_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCNC5=O |
−12.2
± 0.2
|
325 |
EN300-178876_1_1 |
|
C[C@@]1(CCCNC1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.2
± 0.4
|
326 |
EN300-4293814_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)CS(=O)(=O)CCO |
−12.2
± 0.5
|
327 |
EN300-111006_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ccncn5 |
−12.1
± 0.2
|
328 |
EN300-313062_1_4 |
|
CC(=O)N1C[C@H]2C[C@]2(C1)C(=O)N[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−12.1
± 0.2
|
329 |
EN300-6481287_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCO[C@H]5[C@@H](C[C@H]6[C@@H]5CC6=O)O |
−12.1
± 0.3
|
330 |
EN300-211203_1_1 |
|
CC(C)[C@@]1(CC(=O)NC1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
331 |
EN300-1932780_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@H](C(F)F)O |
−12.1
± 0.3
|
332 |
EN300-12067_3_1 |
|
Cc1csc(=O)n1CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
333 |
EN300-1644723_1_8 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5[C@H]6[C@H]5COCC6 |
−12.1
± 0.2
|
334 |
EN300-7473378_1_1 |
|
CN1CCC(CC1)(C#N)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.4
|
335 |
EN300-1244816_1_1 |
|
Cc1nnnn1CC(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
336 |
EN300-657320_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@@H]5CSCC(=O)N5 |
−12.1
± 0.3
|
337 |
EN300-11714_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5ccccc5=O |
−12.1
± 0.3
|
338 |
EN300-111863_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cnc(n5)C#N |
−12.1
± 0.2
|
339 |
EN300-6745453_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@H]5Cc6nncn6C5 |
−12.1
± 0.3
|
340 |
EN300-373552_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cncc(n5)F |
−12.1
± 0.2
|
341 |
EN300-216978_1_1 |
|
Cn1nc(nn1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.2
|
342 |
EN300-322400_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@H]5[C@H](OCCO5)C(F)(F)F |
−12.1
± 0.4
|
343 |
EN300-1387104_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCS5(=O)=O |
−12.1
± 0.3
|
344 |
EN300-20496_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCO[C@H]5CCOC5=O |
−12.1
± 0.3
|
345 |
EN300-6739879_1_1 |
|
C[C@@H]1CCN([C@@H]2[C@@H]1CNC2=O)C(=O)C[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−12.1
± 0.4
|
346 |
EN300-261210_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@]5(CCOC5)C#N |
−12.1
± 0.3
|
347 |
EN300-217107_1_4 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CC[C@H]5C(=O)N |
−12.1
± 0.2
|
348 |
EN300-7436306_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCC5=NO[C@H]6[C@@H]5COC6 |
−12.1
± 0.3
|
349 |
EN300-6763072_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CS(=O)(=O)C56CC(C5)C6 |
−12.1
± 0.3
|
350 |
EN300-72211_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H](C5CC5)O |
−12.1
± 0.2
|
351 |
EN300-28871_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)CCn5ccnn5 |
−12.1
± 0.3
|
352 |
EN300-28871_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)CCn5ccnn5 |
−12.1
± 0.3
|
353 |
EN300-7456948_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cc5cccnn5 |
−12.1
± 0.2
|
354 |
EN300-174668_1_1 |
|
CO[C@@]1(CCOC1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.4
|
355 |
EN300-207959_1_1 |
|
C[C@@]1(CCNC1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
356 |
EN300-1301381_1_2 |
|
COC[C@]1(CCCO1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
357 |
EN300-310173_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5[C@H](CCO5)Cn6ccnc6 |
−12.1
± 0.4
|
358 |
EN300-301925_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@]5(CCCOC5)C#N |
−12.1
± 0.4
|
359 |
EN300-295905_1_1 |
|
C[C@@H]1CN(C[C@@H](O1)C(=O)N)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
360 |
EN300-04433_4_1 |
|
CSCC[C@@H](C(=O)NCCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)NC(=O)N |
−12.1
± 0.4
|
361 |
EN300-75482_1_1 |
|
Cc1c(c(n(n1)C)OC)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
362 |
EN300-92664_1_1 |
|
COCCn1c(ccn1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
363 |
EN300-255795_1_1 |
|
CN1C[C@@H](NC1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.2
|
364 |
EDJ-MED-28ec730d-5_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCCc5c[nH]nc5 |
−12.1
± 0.2
|
365 |
EN300-754584_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CS(=O)(=O)CC(=O)N5 |
−12.1
± 0.2
|
366 |
EN300-94945_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CCNC5=O |
−12.1
± 0.2
|
367 |
EN300-25446_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cnco5 |
−12.1
± 0.2
|
368 |
VLA-UCB-34f3ed0c-8_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)C(=O)CCc5cc[nH]n5 |
−12.1
± 0.2
|
369 |
EN300-1448674_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCn6c(ncn6)C5 |
−12.1
± 0.2
|
370 |
EN300-185729_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CCc6c(nn[nH]6)C5 |
−12.1
± 0.3
|
371 |
EN300-6745453_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5Cc6nncn6C5 |
−12.1
± 0.2
|
372 |
EN300-6505003_1_2 |
|
C[C@H]1CC[C@@H](C(=O)N1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
373 |
EN300-6494474_3_1 |
|
Cn1cnnc1CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
374 |
EN300-1726073_1_1 |
|
Cn1c(cnn1)C(C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)(F)F |
−12.1
± 0.3
|
375 |
EN300-173006_2_1 |
|
C[C@@H](c1nnnn1C)OC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.1
± 0.3
|
376 |
EN300-226314_3_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCC(=O)[C@H]5CCS(=O)(=O)C5 |
−12.1
± 0.4
|
377 |
EN300-1072199_1_1 |
|
CO[C@@]1(CCCOC1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.3
|
378 |
EN300-69107_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC(=O)NCC5 |
−12.0
± 0.4
|
379 |
EN300-69107_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC(=O)NCC5 |
−12.0
± 0.4
|
380 |
EN300-246440_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)C5(CC5)n6cncn6 |
−12.0
± 0.3
|
381 |
EN300-97847_1_1 |
|
Cn1cc(nc1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.2
|
382 |
EN300-306316_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCc5[nH]cnn5 |
−12.0
± 0.2
|
383 |
EN300-18249_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCC(=O)N |
−12.0
± 0.2
|
384 |
EN300-171522_1_1 |
|
Cn1ccc(=O)c(c1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.3
|
385 |
EN300-246440_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C5(CC5)n6cncn6 |
−12.0
± 0.3
|
386 |
EN300-125874_1_1 |
|
Cn1cnnc1N(C)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.3
|
387 |
EN300-1718836_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cc5nnc6n5CCOC6 |
−12.0
± 0.3
|
388 |
EN300-18928_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@@H]5CSCN5C(=O)C6CC6 |
−12.0
± 0.4
|
389 |
EN300-270710_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCCS(=O)(=O)N |
−12.0
± 0.3
|
390 |
VLA-UCB-34f3ed0c-9_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)C(=O)CCc5c[nH]c(=O)o5 |
−12.0
± 0.3
|
391 |
EN300-27341_3_2 |
|
CS(=O)(=O)N1CCC[C@H](C1)C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−12.0
± 0.5
|
392 |
EN300-783124_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]([C@@H]5CCOC5)F |
−12.0
± 0.2
|
393 |
EN300-21258_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCCO |
−12.0
± 0.2
|
394 |
EN300-93573_1_1 |
|
CN(C)C(=O)CC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−12.0
± 0.2
|
395 |
EN300-122849_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCOC[C@@H]5c6ncon6 |
−12.0
± 0.3
|
396 |
EN300-6759972_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC[C@H](CC5)NC(=O)N |
−12.0
± 0.4
|
397 |
EN300-149013_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)c5c([nH]nn5)Cl |
−12.0
± 0.2
|
398 |
EN300-6477724_3_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@@H]5C[C@@H]5c6[nH]cnn6 |
−12.0
± 0.4
|
399 |
EN300-651307_3_1 |
|
CC[C@@H](C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)n5cncn5 |
−12.0
± 0.4
|
400 |
EN300-188356_2_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CNC(=O)[C@]5(CCOC5)F |
−12.0
± 0.2
|