Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
501 |
EDJ-MED-d203f206-31_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N(CC(=O)N)C5CCOCC5 |
−11.4
± 0.3
|
502 |
MAK-UNK-3875bbc8-2_1
|
|
CN(c1cncc2c1cccc2)C(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−11.39
± 0.09
|
503 |
DAR-DIA-076fb6ea-9_2
|
|
c1ccc2c(c1)cncc2N(C#C[C@H]3CCC[NH2+]3)C(=O)Cc4cccc(c4)Cl |
−11.4
± 0.5
|
504 |
EN300-7432302_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@]56CC[C@H](C5)[C@@H]([C@@H]6O)O |
−11.4
± 0.3
|
505 |
MIC-UNK-50cce87d-12_1
|
|
COc1cccc2c1c(cnc2)N3CCC[C@@H](C3=O)c4cccc(c4)Cl |
−11.4
± 0.2
|
506 |
EN300-1915260_4_2_1 |
|
COC[C@H](COCCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O |
−11.4
± 0.5
|
507 |
EN300-54891_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC[C@@H]5CO |
−11.4
± 0.3
|
508 |
EN300-1072972_3_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)C[C@@H]5CCOC5=O |
−11.4
± 0.4
|
509 |
EN300-1600363_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5C[C@H]5C#N |
−11.4
± 0.2
|
510 |
EN300-157527_1_1_1 |
|
Cn1c(c(cn1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)n6cnnc6 |
−11.4
± 0.3
|
511 |
EN300-105267_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCC(=O)Nc5cnccn5 |
−11.4
± 0.2
|
512 |
EN300-1273172_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cnc(cn5)C(=O)N |
−11.4
± 0.3
|
513 |
EDG-MED-90036822-79_1
|
|
Cc1c(c(n[nH]1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)F |
−11.4
± 0.3
|
514 |
EN300-5253939_1_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5COC(=O)O5 |
−11.4
± 0.2
|
515 |
EN300-310173_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5[C@H](CCO5)Cn6ccnc6 |
−11.4
± 0.4
|
516 |
EN300-6745081_1_1_1 |
|
C[C@@]1(CCCCNC1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.4
± 0.3
|
517 |
EN300-143564_1_1_1 |
|
CN\1C(=O)CS/C1=C\C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.4
± 0.2
|
518 |
EN300-101291_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cn(c(=O)[nH]c5=O)CCO |
−11.4
± 0.4
|
519 |
EN300-20668_3_1_1 |
|
COC(=O)CC(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.4
± 0.3
|
520 |
EN300-06030_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ccc(cc5)n6cnnn6 |
−11.4
± 0.3
|
521 |
EN300-6526669_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cnn6c5C(=O)NCC6 |
−11.4
± 0.3
|
522 |
EN300-260152_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cc5cnns5 |
−11.4
± 0.2
|
523 |
EN300-102487_1_1_1 |
|
Cn1c(=O)c(c[nH]c1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.4
± 0.3
|
524 |
EN300-174603_3_1_1 |
|
CN(C(=O)CCOCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)OC |
−11.4
± 0.3
|
525 |
EN300-44821_1_1_1 |
|
C=CCOCC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.4
± 0.2
|
526 |
MIC-UNK-9582b2c5-3_4
|
|
CC(=O)N1CC[C@H]2[C@H](C1)CN(C(=O)N2c3cccc(c3)Cl)c4cncc5c4cccc5 |
−11.4
± 0.3
|
527 |
EN300-6744028_1_4_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5C[C@H]6C[C@@H]5[C@H]([C@@H]6O)O |
−11.4
± 0.3
|
528 |
EN300-80230_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ncccn5 |
−11.3
± 0.2
|
529 |
EN300-80230_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5ncccn5 |
−11.3
± 0.2
|
530 |
EN300-365398_2_1_1 |
|
Cn1c(nnn1)CCOC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.3
|
531 |
EDG-MED-90036822-99_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]([C@@H](C5CCC5)O)F |
−11.3
± 0.3
|
532 |
EDJ-MED-6864a934-7_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc6c(nc5)n[nH]n6 |
−11.3
± 0.2
|
533 |
EN300-244278_1_1_2 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5C=C6COCC[N@@]6N5 |
−11.3
± 0.3
|
534 |
EN300-1600517_3_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOC[C@@H](CO)F |
−11.3
± 0.3
|
535 |
EN300-94945_1_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCNC5=O |
−11.3
± 0.2
|
536 |
EN300-4293814_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CS(=O)(=O)CCO |
−11.3
± 0.5
|
537 |
EN300-213358_1_1_1 |
|
Cn1c(ncn1)COCC(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.2
|
538 |
EN300-97697_1_1_1 |
|
CN(C1CC(C1)O)C(=O)C[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.3
|
539 |
EN300-7463171_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCCS(=O)(=O)CCO |
−11.3
± 0.4
|
540 |
EN300-205622_1_1_1 |
|
CS(=O)(=O)c1nccc(n1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.3
|
541 |
EN300-42131_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc6c([nH]c(=O)[nH]c6=O)nc5 |
−11.3
± 0.3
|
542 |
EN300-107892_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cc(nn5)C6CC6 |
−11.3
± 0.3
|
543 |
EDJ-MED-d203f206-3_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCOC[C@@H]5c6ncon6 |
−11.3
± 0.4
|
544 |
EN300-6238494_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCC(=O)[C@@H]5COCCO5 |
−11.3
± 0.3
|
545 |
EN300-41423_1_1_1 |
|
Cc1ccc(c(=O)n1C)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.3
|
546 |
EN300-6733459_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@]56CCC[N@@]5S(=O)(=O)CC6 |
−11.3
± 0.5
|
547 |
VLA-UCB-50c39ae8-1_1
|
|
CC(=O)N(c1cncc2c1cccc2)C(=O)[C@@H]3CCOc4c3cc(cc4)Cl |
−11.3
± 0.1
|
548 |
EDJ-MED-d203f206-41_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCC[C@@H]5CO |
−11.3
± 0.3
|
549 |
EN300-102347_3_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCC5(COC5)CO |
−11.3
± 0.3
|
550 |
EN300-6744028_1_6_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5C[C@H]6C[C@@H]5[C@@H]([C@H]6O)O |
−11.3
± 0.2
|
551 |
EN300-1268016_1_11_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N[C@@H]5C[C@H]6[C@@H]5C[C@H](C6)C(=O)N |
−11.3
± 0.4
|
552 |
EN300-59285_3_1_1 |
|
CC(C)(C(=O)NCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4)O |
−11.3
± 0.3
|
553 |
EN300-2011083_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5CCC(=O)OCC5 |
−11.3
± 0.3
|
554 |
EN300-52983_1_1_1 |
|
CN1C[C@@H](CCC1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.3
|
555 |
EN300-298552_1_2_1 |
|
CO[C@H]([C@@H]1CCOC1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.2
|
556 |
EN300-111863_3_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)Cn5cnc(n5)C#N |
−11.3
± 0.3
|
557 |
EN300-226964_1_1_1 |
|
Cc1ccn(n1)CC(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.2
|
558 |
EN300-169955_1_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5[C@@H](CC(=O)N5)C(F)(F)F |
−11.3
± 0.2
|
559 |
EN300-227218_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CC[N@@H+]6CC[C@H]5C6 |
−11.3
± 0.3
|
560 |
EN300-195924_3_2_1 |
|
C[C@]1(CCC(=O)NC1)C(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.4
|
561 |
EDJ-MED-28ec730d-5_1_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)OCCc5c[nH]nc5 |
−11.3
± 0.3
|
562 |
EN300-6759512_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cn(nn5)[C@@H]6COC[C@@H]6F |
−11.3
± 0.3
|
563 |
EN300-731622_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C[C@@H]5COCCO5 |
−11.3
± 0.2
|
564 |
EN300-140582_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5COCC[N@]5CC(F)F |
−11.3
± 0.3
|
565 |
EN300-1696962_3_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCCCn5cnnn5 |
−11.3
± 0.3
|
566 |
EN300-7434209_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cncc6c5[nH]c(=O)[nH]6 |
−11.3
± 0.3
|
567 |
ALP-UNI-44c99a80-3_1
|
|
c1ccc2c(c1)cncc2N(Cc3cnco3)C(=O)[C@@H]4CCOc5c4cc(cc5)Cl |
−11.3
± 0.2
|
568 |
EN300-29220_1_1_1 |
|
Cc1c(n[nH]c(=O)c1C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)C |
−11.3
± 0.3
|
569 |
EN300-23942_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)Cn5cccn5 |
−11.3
± 0.2
|
570 |
EN300-54304_1_1_1 |
|
CCOCCOCC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.3
± 0.2
|
571 |
EN300-138676_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N(CC(=O)N)CC(F)(F)F |
−11.3
± 0.3
|
572 |
ED_-GRI-5b13fbe2-74_1
|
|
C[N@@H+]1CCO[C@@H](C1)c2nccc(n2)CO[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−11.3
± 0.3
|
573 |
EN300-254883_3_1_1 |
|
Cc1c(non1)CC(=O)NCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.3
|
574 |
EN300-1273362_3_1_1 |
|
C[C@@]1(CN(C1=O)C)COCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.3
|
575 |
EDJ-MED-d203f206-13_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)Nc5cnncn5 |
−11.3
± 0.2
|
576 |
VLA-UCB-50c39ae8-8_2_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCOc4c3cc(cc4O[C@H]5C[C@@H]([NH2+]5)O)Cl |
−11.3
± 0.3
|
577 |
EN300-175186_3_2_1 |
|
C[C@H](CO)OCC[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.3
± 0.3
|
578 |
EN300-18928_1_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CSCN5C(=O)C6CC6 |
−11.3
± 0.3
|
579 |
EN300-131465_1_1_1 |
|
COc1cc(on1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.2
|
580 |
EDG-MED-90036822-94_8
|
|
C[C@H]1C[C@H]1[C@H]([C@@H](C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)F)O |
−11.3
± 0.3
|
581 |
EN300-21258_3_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCCO |
−11.3
± 0.2
|
582 |
EN300-322400_3_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)[C@H]5[C@H](OCCO5)C(F)(F)F |
−11.3
± 0.3
|
583 |
EN300-178876_1_1_1 |
|
C[C@@]1(CCCNC1=O)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.3
± 0.4
|
584 |
EN300-83527_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc6ncccn6n5 |
−11.3
± 0.2
|
585 |
EN300-1644723_1_7_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@@H]5[C@H]6[C@H]5COCC6 |
−11.3
± 0.2
|
586 |
EN300-217343_1_1_1 |
|
Cn1c2c(nn1)CC[C@@H](C2)C(=O)N[C@]3(CCOc4c3cc(cc4)Cl)C(=O)Nc5cncc6c5cccc6 |
−11.3
± 0.3
|
587 |
EN300-246248_2_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)COC[C@H]5CCNC5=O |
−11.3
± 0.2
|
588 |
EN300-637522_2_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCC(=O)N5C6CCC5(CC6)C(=O)N |
−11.3
± 0.3
|
589 |
EN300-20375_1_1_1 |
|
COCCOCC(=O)N[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4 |
−11.3
± 0.2
|
590 |
MIC-UNK-50cce87d-10_2
|
|
c1cc(cc(c1)Cl)[C@H]2CCCN(C2=O)c3cncc4c3c(ccc4)Cl |
−11.3
± 0.2
|
591 |
EN300-270710_3_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCOCCS(=O)(=O)N |
−11.3
± 0.2
|
592 |
EN300-114526_1_1_1 |
|
Cc1c(c([nH]n1)C(=O)N[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5)O |
−11.3
± 0.2
|
593 |
EN300-238234_1_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)c5cc6c([nH]c5=O)CCC[C@H]6O |
−11.2
± 0.4
|
594 |
EN300-139268_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C(=O)NCC(F)(F)F |
−11.2
± 0.2
|
595 |
EN300-343474_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)C[C@@H]5CCNC5=O |
−11.2
± 0.3
|
596 |
EN300-11934_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)CN5CCCC5=O |
−11.2
± 0.3
|
597 |
EN300-90225_3_1_1 |
|
Cn1nc(nn1)COCC[C@]2(CCOc3c2cc(cc3)Cl)C(=O)Nc4cncc5c4cccc5 |
−11.2
± 0.3
|
598 |
EN300-332606_1_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@H]5CCC(=O)O5 |
−11.2
± 0.2
|
599 |
EN300-658559_3_1_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CCNC(=O)C5(CC5)n6ccnn6 |
−11.2
± 0.3
|
600 |
EN300-311920_1_2_1 |
|
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)NC(=O)[C@]5(CCS(=O)(=O)C5)F |
−11.2
± 0.3
|