Rank |
Compound |
SMILES |
ΔG / kcal M-1 |
pIC50 |
101 |
PET-UNK-14142a25-1
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.3
± 0.1
|
6.77
± 0.08
|
102 |
EDJ-MED-8bb691af-8
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.3
± 0.1
|
6.76
± 0.08
|
103 |
EDJ-MED-ee81482e-5
|
|
c1cc2cncc(c2cc1CN3CC4(C3)COC4)N5CCC6(C5=O)CN(Cc7c6cc(cc7)Cl)S(=O)(=O)CC8(CC8)C#N |
−9.3
± 0.4
|
6.8
± 0.3
|
104 |
VLA-UNK-61877630-6
|
|
CNC(=O)CN1C([C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl)C(F)F |
−9.3
± 0.1
|
6.74
± 0.08
|
105 |
PET-UNK-94036022-5
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−9.2
± 0.2
|
6.7
± 0.2
|
106 |
EDG-MED-b1ef7fe3-1
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)Cl)c5cc(ccc5C1=O)Cl |
−9.2
± 0.1
|
6.72
± 0.08
|
107 |
ALP-POS-ecbed2ba-9
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)N6CC(C6)C#N |
−9.2
± 0.3
|
6.7
± 0.3
|
108 |
LUO-POS-9931618f-1
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.2
± 0.1
|
6.71
± 0.08
|
109 |
EDJ-MED-5cd3920d-4
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)C(F)F)c6cc(ccc6C2=O)Cl |
−9.2
± 0.1
|
6.71
± 0.10
|
110 |
PET-UNK-94036022-12
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−9.2
± 0.2
|
6.7
± 0.2
|
111 |
PET-UNK-aa57768f-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−9.2
± 0.1
|
6.70
± 0.08
|
112 |
EDJ-MED-fed7ac0b-2
|
|
CNC(=O)C1(CC1)N2CC3(CNN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−9.2
± 0.1
|
6.69
± 0.10
|
113 |
EDJ-MED-468565e0-1
|
|
c1cc2cncc(c2cc1OCCN3CCCC3)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−9.2
± 0.5
|
6.7
± 0.4
|
114 |
MAT-POS-853c0ffa-22
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5ccc(c6)S(=O)(=O)C)Cl |
−9.2
± 0.3
|
6.7
± 0.2
|
115 |
EDJ-MED-7e491f08-1
|
|
c1ccc2c(c1)cncc2N3CC([C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)(F)F |
−9.1
± 0.4
|
6.7
± 0.3
|
116 |
EDG-MED-b1ef7fe3-3
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3ccc(c4)F)c5cc(ccc5C1=O)Cl |
−9.14
± 0.09
|
6.66
± 0.07
|
117 |
PET-UNK-77d5678a-5
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−9.14
± 0.08
|
6.66
± 0.06
|
118 |
EDJ-MED-976a33d5-1
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−9.1
± 0.1
|
6.65
± 0.08
|
119 |
ALP-POS-ecbed2ba-18
|
|
CCN(C)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−9.1
± 0.2
|
6.7
± 0.2
|
120 |
MIK-ENA-794411b8-1
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.1
± 0.1
|
6.64
± 0.08
|
121 |
EDJ-MED-159244ea-1
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CCOc5c4cc(cc5)Cl |
−9.11
± 0.06
|
6.64
± 0.04
|
122 |
EDG-MED-b1ef7fe3-2
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)F)c5cc(ccc5C1=O)Cl |
−9.1
± 0.1
|
6.63
± 0.08
|
123 |
EDJ-MED-b6c6ee2b-7
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)F)c6cc(ccc6C2=O)Cl |
−9.1
± 0.1
|
6.61
± 0.08
|
124 |
VLA-UCB-05e51b3f-5
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@]4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
125 |
MAT-POS-94643566-1
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
126 |
VLA-UCB-50c39ae8-2
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
127 |
BEN-BAS-c2bc0d80-6
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
128 |
LUO-POS-868e8996-10
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.1
± 0.3
|
6.6
± 0.2
|
129 |
EDJ-MED-b6c6ee2b-6
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)F)c5cc(ccc5C1=O)Cl |
−9.1
± 0.1
|
6.60
± 0.07
|
130 |
VLA-UNK-f702bf1c-3
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)Cc6nc[nH]n6 |
−9.1
± 0.1
|
6.6
± 0.1
|
131 |
MIK-ENA-37e0b697-1
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.0
± 0.1
|
6.59
± 0.08
|
132 |
MAT-POS-576f7758-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−9.0
± 0.1
|
6.58
± 0.09
|
133 |
ALP-POS-477dc5b7-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CCOc5c4cc(cc5)Cl |
−9.01
± 0.05
|
6.56
± 0.04
|
134 |
MAT-POS-e48723dc-2
|
|
CNC(=O)C1(CC1)N2C[C@@]3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−9.0
± 0.1
|
6.55
± 0.08
|
135 |
PET-UNK-94036022-10
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−9.0
± 0.2
|
6.6
± 0.2
|
136 |
MAT-POS-853c0ffa-1
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3c(ccc4)Cl)c5cc(ccc5C1=O)Cl |
−8.99
± 0.10
|
6.55
± 0.07
|
137 |
ALP-POS-ecbed2ba-3
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−9.0
± 0.2
|
6.5
± 0.2
|
138 |
PET-UNK-aa57768f-3
|
|
C#CCN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.95
± 0.09
|
6.52
± 0.07
|
139 |
LUO-POS-9931618f-2
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.9
± 0.1
|
6.52
± 0.08
|
140 |
LUO-POS-868e8996-7
|
|
CNC(=O)CN1C[C@@]2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.9
± 0.1
|
6.52
± 0.07
|
141 |
EDJ-MED-7d88f880-1
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3ccc(c4)S(=N)(=O)C)c5cc(ccc5C1=O)Cl |
−8.9
± 0.1
|
6.50
± 0.08
|
142 |
EDJ-MED-cc48ee33-4
|
|
Cc1cnn(c1C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl)C |
−8.9
± 0.1
|
6.50
± 0.10
|
143 |
MAT-POS-853c0ffa-11
|
|
CC(C)(c1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)O |
−8.9
± 0.3
|
6.5
± 0.2
|
144 |
EDG-MED-b1ef7fe3-4
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3ccc(c4)Cl)c5cc(ccc5C1=O)Cl |
−8.9
± 0.1
|
6.48
± 0.08
|
145 |
MAT-POS-1d5ab790-3
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3c(ccc4)Cl)c5cc(ccc5C1=O)Cl |
−8.9
± 0.1
|
6.48
± 0.08
|
146 |
MAT-POS-983b399a-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CCOc5c4cc(cc5)Cl |
−8.89
± 0.06
|
6.48
± 0.04
|
147 |
VLA-UNK-61877630-3
|
|
CNC(=O)CN1C([C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl)C(F)(F)F |
−8.9
± 0.1
|
6.47
± 0.09
|
148 |
DAR-DIA-0f7b7cd9-8
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCOc5c4cc(cc5)Cl)C(=O)S3 |
−8.87
± 0.06
|
6.46
± 0.05
|
149 |
EDJ-MED-5cd3920d-1
|
|
c1cc2cncc(c2cc1OC(F)F)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.9
± 0.3
|
6.5
± 0.2
|
150 |
VLA-UNK-56836b69-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(c(c5)Cl)Cl)NC3=O |
−8.83
± 0.09
|
6.43
± 0.07
|
151 |
PET-UNK-94036022-2
|
|
C#CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3[C@]4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−8.8
± 0.2
|
6.4
± 0.2
|
152 |
EDJ-MED-98c0a822-2
|
|
CNC(=O)C1(COC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6S2(=O)=O)Cl |
−8.8
± 0.3
|
6.4
± 0.2
|
153 |
ALP-POS-ecbed2ba-22
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)CC#N |
−8.8
± 0.3
|
6.4
± 0.2
|
154 |
EDJ-MED-b6c6ee2b-4
|
|
c1cc2cncc(c2cc1Cl)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.8
± 0.3
|
6.4
± 0.2
|
155 |
EDJ-MED-7d88f880-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4ccc(c5)S(=N)(=O)C)c6cc(ccc6C2=O)Cl |
−8.8
± 0.1
|
6.40
± 0.08
|
156 |
VLA-UNK-61877630-10
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C(F)(F)F |
−8.8
± 0.3
|
6.4
± 0.2
|
157 |
EDJ-MED-a12e3a20-2
|
|
CNC(=O)CN1CC2(c3cc(ccc3C1=O)Cl)C(=O)CN(C2=O)c4cncc5c4cccc5 |
−8.8
± 0.1
|
6.40
± 0.08
|
158 |
MAT-POS-90505e2b-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCOc5c4cc(cc5)Cl)OC3=O |
−8.76
± 0.04
|
6.38
± 0.03
|
159 |
VLA-UNK-61877630-8
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(c(c5)F)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.7
± 0.3
|
6.4
± 0.2
|
160 |
EDJ-MED-976a33d5-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4ccc(c5)S(=O)(=O)C)c6cc(ccc6C2=O)Cl |
−8.7
± 0.1
|
6.37
± 0.10
|
161 |
MAT-POS-ec6d90b7-1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)OC3=O |
−8.73
± 0.05
|
6.36
± 0.04
|
162 |
ALP-POS-ecbed2ba-13
|
|
CC(C)(CS(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl)C#N |
−8.7
± 0.3
|
6.4
± 0.2
|
163 |
EDJ-MED-468565e0-5
|
|
c1cc2cncc(c2cc1OCCN3CC(C3)(F)F)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−8.7
± 0.5
|
6.4
± 0.4
|
164 |
EDJ-MED-98c0a822-4
|
|
CNC(=O)C1(COC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.7
± 0.1
|
6.35
± 0.08
|
165 |
MAT-POS-50a80394-4
|
|
CC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5 |
−8.7
± 0.2
|
6.3
± 0.2
|
166 |
MAT-POS-ec6d90b7-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@]4(CCOc5c4cc(cc5)Cl)OC3=O |
−8.68
± 0.05
|
6.32
± 0.03
|
167 |
VLA-UNK-61877630-7
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(cc5F)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.7
± 0.3
|
6.3
± 0.2
|
168 |
VLA-UNK-3a43cd95-1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(c(c5)F)Cl)NC3=O |
−8.66
± 0.07
|
6.31
± 0.05
|
169 |
LUO-POS-868e8996-9
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.7
± 0.3
|
6.3
± 0.2
|
170 |
EDJ-MED-fed7ac0b-1
|
|
CNC(=O)CN1CC2(CNN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.6
± 0.1
|
6.29
± 0.08
|
171 |
MAT-POS-853c0ffa-13
|
|
c1cc2cncc(c2cc1F)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.6
± 0.3
|
6.3
± 0.2
|
172 |
MAT-POS-1bed62cf-1
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.6
± 0.3
|
6.3
± 0.2
|
173 |
EDJ-MED-cc48ee33-2
|
|
Cn1c(ccn1)C(=O)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.6
± 0.1
|
6.28
± 0.10
|
174 |
PET-UNK-94036022-3
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−8.6
± 0.2
|
6.3
± 0.2
|
175 |
EDJ-MED-8bb691af-6
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.6
± 0.3
|
6.3
± 0.2
|
176 |
EDJ-MED-468565e0-3
|
|
c1cc2cncc(c2cc1OCCN3CCS(=O)(=O)CC3)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−8.6
± 0.5
|
6.3
± 0.4
|
177 |
EDJ-MED-ee81482e-2
|
|
CN1CC(C1)Oc2ccc3cncc(c3c2)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−8.6
± 0.5
|
6.3
± 0.4
|
178 |
EDJ-MED-5cd3920d-5
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C(F)F |
−8.6
± 0.3
|
6.2
± 0.3
|
179 |
DAR-DIA-6be260fc-5
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CCNc5c4cc(cc5)Cl |
−8.57
± 0.08
|
6.24
± 0.06
|
180 |
DAR-DIA-0f7b7cd9-9
|
|
c1ccc2c(c1)cncc2N3CC(=O)C4(C3=O)CCOc5c4cc(cc5)Cl |
−8.54
± 0.06
|
6.22
± 0.04
|
181 |
MIK-ENA-5d9157e9-2
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.5
± 0.3
|
6.2
± 0.2
|
182 |
EDJ-MED-fd8ed875-3
|
|
CNC(=O)CN1CC2(C=CN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.52
± 0.10
|
6.21
± 0.07
|
183 |
VLA-UCB-34f3ed0c-15
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CN6CCNCC6 |
−8.5
± 0.3
|
6.2
± 0.2
|
184 |
JOH-MSK-1f2dff76-2
|
|
CNC(=O)CN1Cc2ccc(cc2[C@]3(C1)CC(=O)N(C3=O)c4cncc5c4cccc5)Cl |
−8.5
± 0.2
|
6.2
± 0.2
|
185 |
MIK-ENA-5d9157e9-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.5
± 0.4
|
6.2
± 0.3
|
186 |
EDJ-MED-fd8ed875-5
|
|
CNC(=O)CN1CC2(c3cc(ccc3C1=O)Cl)C(=CN(C2=O)c4cncc5c4cccc5)F |
−8.47
± 0.10
|
6.17
± 0.07
|
187 |
EDJ-MED-a12e3a20-1
|
|
c1ccc2c(c1)cncc2N3CC(=O)C4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.5
± 0.4
|
6.2
± 0.3
|
188 |
MAT-POS-50a80394-5
|
|
CCC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5 |
−8.4
± 0.2
|
6.1
± 0.2
|
189 |
EDJ-MED-98c0a822-1
|
|
CNC(=O)C1(CCC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6S2(=O)=O)Cl |
−8.4
± 0.4
|
6.1
± 0.3
|
190 |
MAT-POS-853c0ffa-14
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)F)Cl |
−8.4
± 0.3
|
6.1
± 0.2
|
191 |
MAT-POS-853c0ffa-16
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5ccc(c6)S(=O)(=O)C)Cl |
−8.4
± 0.3
|
6.1
± 0.2
|
192 |
ALP-POS-ecbed2ba-6
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−8.4
± 0.3
|
6.1
± 0.2
|
193 |
EDJ-MED-7587a9ee-3
|
|
CS(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−8.4
± 0.2
|
6.1
± 0.1
|
194 |
ALP-POS-ecbed2ba-10
|
|
COC1CN(C1)S(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−8.3
± 0.3
|
6.1
± 0.3
|
195 |
EDJ-MED-fd8ed875-4
|
|
CNC(=O)C1(CC1)N2CC3(C=CN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.3
± 0.1
|
6.07
± 0.08
|
196 |
PET-UNK-7e9559de-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)Cc6nncs6 |
−8.3
± 0.1
|
6.06
± 0.10
|
197 |
PET-UNK-aa57768f-2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC#N |
−8.31
± 0.08
|
6.05
± 0.06
|
198 |
EDJ-MED-fd8ed875-6
|
|
CNC(=O)C1(CC1)N2CC3(c4cc(ccc4C2=O)Cl)C(=CN(C3=O)c5cncc6c5cccc6)F |
−8.3
± 0.1
|
6.04
± 0.09
|
199 |
JOH-MSK-1f2dff76-4
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CNCc5c4cc(cc5)Cl |
−8.3
± 0.1
|
6.0
± 0.1
|
200 |
EDJ-MED-fed7ac0b-4
|
|
CNC(=O)CN1CC2(C=NN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.3
± 0.1
|
6.03
± 0.07
|