Rank |
Compound |
SMILES |
ΔG / kcal M-1 |
pIC50 |
101 |
ALP-POS-ecbed2ba-21
|
|
CN(CCOC)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−9.9
± 0.2
|
7.2
± 0.2
|
102 |
MIK-ENA-37e0b697-1
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.9
± 0.1
|
7.2
± 0.1
|
103 |
MAT-POS-1d5ab790-3
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3c(ccc4)Cl)c5cc(ccc5C1=O)Cl |
−9.9
± 0.2
|
7.2
± 0.1
|
104 |
EDJ-MED-b6c6ee2b-4
|
|
c1cc2cncc(c2cc1Cl)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.9
± 0.4
|
7.2
± 0.3
|
105 |
BEN-BAS-c2bc0d80-3
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCOc5c4cc(cc5)Cl)CN3 |
−9.85
± 0.06
|
7.18
± 0.04
|
106 |
PET-UNK-77d5678a-6
|
|
COC(=O)CN1CC2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.83
± 0.09
|
7.16
± 0.07
|
107 |
MAT-POS-853c0ffa-20
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)C(C)(C)O)Cl |
−9.8
± 0.3
|
7.1
± 0.3
|
108 |
MAT-POS-50a80394-4
|
|
CC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5 |
−9.8
± 0.2
|
7.1
± 0.2
|
109 |
PET-UNK-77d5678a-5
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−9.8
± 0.1
|
7.13
± 0.08
|
110 |
ALP-POS-ecbed2ba-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.8
± 0.4
|
7.1
± 0.3
|
111 |
MAT-POS-50a80394-2
|
|
CCC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−9.8
± 0.6
|
7.1
± 0.4
|
112 |
MAT-POS-853c0ffa-16
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5ccc(c6)S(=O)(=O)C)Cl |
−9.7
± 0.3
|
7.1
± 0.2
|
113 |
PET-UNK-aa57768f-2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC#N |
−9.74
± 0.08
|
7.09
± 0.06
|
114 |
MAT-POS-e48723dc-2
|
|
CNC(=O)C1(CC1)N2C[C@@]3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−9.7
± 0.2
|
7.1
± 0.1
|
115 |
MAT-POS-40ad851a-3
|
|
CCN(CC)CCOc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.7
± 0.6
|
7.1
± 0.4
|
116 |
VLA-UNK-61877630-10
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C(F)(F)F |
−9.7
± 0.3
|
7.1
± 0.3
|
117 |
VLA-UNK-f702bf1c-1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CCc6cc[nH]n6 |
−9.7
± 0.2
|
7.1
± 0.1
|
118 |
EDJ-MED-98c0a822-4
|
|
CNC(=O)C1(COC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−9.7
± 0.2
|
7.1
± 0.1
|
119 |
ALP-POS-ecbed2ba-16
|
|
CN(CCC#N)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−9.7
± 0.7
|
7.1
± 0.5
|
120 |
MAT-POS-ec6d90b7-1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)OC3=O |
−9.63
± 0.05
|
7.01
± 0.04
|
121 |
EDJ-MED-9f4ac58c-4
|
|
CS(=O)(=O)c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.6
± 0.7
|
7.0
± 0.5
|
122 |
BEN-BAS-c2bc0d80-7
|
|
CN1C(=O)N(C(=O)C12CCOc3c2cc(cc3)Cl)c4cncc5c4cccc5 |
−9.62
± 0.08
|
7.01
± 0.06
|
123 |
MAT-POS-90505e2b-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCOc5c4cc(cc5)Cl)OC3=O |
−9.62
± 0.05
|
7.00
± 0.04
|
124 |
EDG-MED-b1ef7fe3-4
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3ccc(c4)Cl)c5cc(ccc5C1=O)Cl |
−9.6
± 0.2
|
7.0
± 0.1
|
125 |
MAT-POS-96396902-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)Cc6nncs6 |
−9.6
± 0.1
|
7.0
± 0.1
|
126 |
PET-UNK-7e9559de-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)Cc6nncs6 |
−9.6
± 0.2
|
7.0
± 0.1
|
127 |
VLA-UNK-3a43cd95-1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(c(c5)F)Cl)NC3=O |
−9.52
± 0.07
|
6.93
± 0.05
|
128 |
PET-UNK-94036022-13
|
|
C=C1C(=O)C2(CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
−9.5
± 0.4
|
6.9
± 0.3
|
129 |
EDJ-MED-976a33d5-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4ccc(c5)S(=O)(=O)C)c6cc(ccc6C2=O)Cl |
−9.5
± 0.2
|
6.9
± 0.1
|
130 |
MIK-ENA-5d9157e9-2
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.4
± 0.4
|
6.9
± 0.3
|
131 |
LUO-POS-b5068a05-2
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)N=C3NC#N |
−9.4
± 0.3
|
6.9
± 0.2
|
132 |
PET-UNK-94036022-9
|
|
C#CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−9.4
± 0.3
|
6.9
± 0.2
|
133 |
VLA-UCB-34f3ed0c-14
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CC6CCCCC6 |
−9.4
± 0.2
|
6.8
± 0.1
|
134 |
VLA-UNK-61877630-6
|
|
CNC(=O)CN1C([C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl)C(F)F |
−9.4
± 0.2
|
6.8
± 0.1
|
135 |
MAT-POS-ec6d90b7-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@]4(CCOc5c4cc(cc5)Cl)OC3=O |
−9.39
± 0.05
|
6.84
± 0.04
|
136 |
MAT-POS-576f7758-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−9.4
± 0.1
|
6.8
± 0.1
|
137 |
EDJ-MED-5cd3920d-2
|
|
c1cc2cncc(c2cc1C(F)F)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.3
± 0.4
|
6.8
± 0.3
|
138 |
PET-UNK-77d5678a-2
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)Cc6nnco6 |
−9.3
± 0.1
|
6.80
± 0.08
|
139 |
EDJ-MED-5cd3920d-5
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C(F)F |
−9.3
± 0.4
|
6.8
± 0.3
|
140 |
EDJ-MED-7d88f880-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4ccc(c5)S(=N)(=O)C)c6cc(ccc6C2=O)Cl |
−9.3
± 0.2
|
6.8
± 0.2
|
141 |
MAT-POS-c2d406ed-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)NC3=O |
−9.3
± 0.3
|
6.7
± 0.2
|
142 |
MAT-POS-853c0ffa-14
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)F)Cl |
−9.3
± 0.4
|
6.7
± 0.3
|
143 |
ALP-POS-ecbed2ba-19
|
|
CN(CCO)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−9.2
± 0.3
|
6.7
± 0.2
|
144 |
MAT-POS-1d5ab790-1
|
|
c1cc2cncc(c2c(c1)Cl)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.2
± 0.4
|
6.7
± 0.3
|
145 |
MAT-POS-1d5ab790-2
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4c(ccc5)Cl)Cl |
−9.2
± 0.2
|
6.7
± 0.2
|
146 |
VLA-UNK-61877630-8
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(c(c5)F)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.2
± 0.4
|
6.7
± 0.3
|
147 |
VLA-UNK-f702bf1c-6
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CC6CCCCC6 |
−9.2
± 0.1
|
6.7
± 0.1
|
148 |
MAT-POS-38eb6498-3
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cc(cc5)OCCN(C)C)Cl |
−9.1
± 0.4
|
6.6
± 0.3
|
149 |
EDJ-MED-7587a9ee-3
|
|
CS(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−9.1
± 0.2
|
6.6
± 0.1
|
150 |
MAT-POS-94643566-1
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CCOc5c4cc(cc5)Cl |
−9.08
± 0.04
|
6.61
± 0.03
|
151 |
VLA-UCB-05e51b3f-5
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@]4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
152 |
VLA-UCB-50c39ae8-2
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
153 |
BEN-BAS-c2bc0d80-6
|
|
c1ccc2c(c1)cncc2N3C(=O)CC4(C3=O)CCOc5c4cc(cc5)Cl |
−9.07
± 0.04
|
6.61
± 0.03
|
154 |
EDJ-MED-ede5c6cb-2
|
|
c1cc2c(cc1NS(=O)(=O)C3CC3)cncc2N4CCC5(C4=O)CCS(=O)(=O)c6c5cc(cc6)Cl |
−9.1
± 0.2
|
6.6
± 0.1
|
155 |
ALP-POS-4483ae88-2
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5S1(=O)=O)Cl |
−9.1
± 0.2
|
6.6
± 0.2
|
156 |
PET-UNK-94036022-10
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−9.0
± 0.3
|
6.6
± 0.2
|
157 |
12_-111-3e02a1cd-2
|
|
COC(=O)CN1C[C@]2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−9.0
± 0.1
|
6.57
± 0.08
|
158 |
MAT-POS-853c0ffa-22
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5ccc(c6)S(=O)(=O)C)Cl |
−9.0
± 0.3
|
6.5
± 0.2
|
159 |
VLA-UNK-61877630-5
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(c(cc5C1=O)F)Cl |
−9.0
± 0.1
|
6.54
± 0.09
|
160 |
MAT-POS-853c0ffa-15
|
|
CS(=O)(=O)c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−9.0
± 0.5
|
6.5
± 0.3
|
161 |
EDJ-MED-b6c6ee2b-1
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cc(cc5)OCCN(C)C)Cl |
−8.9
± 0.4
|
6.5
± 0.3
|
162 |
ALP-POS-ecbed2ba-3
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−8.9
± 0.3
|
6.5
± 0.2
|
163 |
MAT-POS-c2d406ed-3
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)NC3=S |
−8.9
± 0.3
|
6.5
± 0.2
|
164 |
PET-UNK-7e9559de-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)Cc6nncs6 |
−8.9
± 0.2
|
6.5
± 0.1
|
165 |
EDJ-MED-fed7ac0b-3
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN3)CN(C(=O)c5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−8.9
± 0.7
|
6.5
± 0.5
|
166 |
VLA-UNK-f2612802-3
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(cc(c5S1(=O)=O)F)Cl |
−8.9
± 0.2
|
6.5
± 0.2
|
167 |
LUO-POS-868e8996-7
|
|
CNC(=O)CN1C[C@@]2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.9
± 0.1
|
6.47
± 0.08
|
168 |
VLA-UNK-f702bf1c-4
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CC6CC(=O)NC6 |
−8.9
± 0.2
|
6.5
± 0.1
|
169 |
EDJ-MED-fd8ed875-6
|
|
CNC(=O)C1(CC1)N2CC3(c4cc(ccc4C2=O)Cl)C(=CN(C3=O)c5cncc6c5cccc6)F |
−8.9
± 0.2
|
6.4
± 0.2
|
170 |
EDJ-MED-468565e0-3
|
|
c1cc2cncc(c2cc1OCCN3CCS(=O)(=O)CC3)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−8.8
± 0.6
|
6.4
± 0.4
|
171 |
MAT-POS-853c0ffa-21
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)F)Cl |
−8.8
± 0.3
|
6.4
± 0.2
|
172 |
ALP-POS-ecbed2ba-9
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)N6CC(C6)C#N |
−8.8
± 0.4
|
6.4
± 0.3
|
173 |
PET-UNK-94036022-6
|
|
C=C1C(=O)[C@]2(CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
−8.8
± 0.4
|
6.4
± 0.3
|
174 |
MAT-POS-1bed62cf-2
|
|
CNC(=O)CN1CC2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.8
± 0.1
|
6.42
± 0.08
|
175 |
PET-UNK-77d5678a-3
|
|
COC(=O)CN1C[C@]2(CC(=O)N(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.8
± 0.1
|
6.42
± 0.07
|
176 |
ALP-POS-ecbed2ba-2
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCS(=O)(=O)CC6)C#N |
−8.8
± 0.3
|
6.4
± 0.2
|
177 |
EDJ-MED-98c0a822-2
|
|
CNC(=O)C1(COC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6S2(=O)=O)Cl |
−8.8
± 0.3
|
6.4
± 0.2
|
178 |
MAT-POS-853c0ffa-7
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5c(ccc6)Cl)Cl |
−8.8
± 0.4
|
6.4
± 0.3
|
179 |
EDJ-MED-ede5c6cb-1
|
|
CS(=O)(=O)Nc1ccc2c(c1)cncc2N3CCC4(C3=O)CCS(=O)(=O)c5c4cc(cc5)Cl |
−8.7
± 0.2
|
6.4
± 0.1
|
180 |
MAT-POS-853c0ffa-8
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5c(cc(c6)F)Cl)Cl |
−8.7
± 0.3
|
6.4
± 0.2
|
181 |
JOH-MSK-ccc6e4c0-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN(Cc5c4cc(c(c5)Cl)Cl)S(=O)(=O)CC6(CC6)C#N)NC3=O |
−8.7
± 0.2
|
6.4
± 0.2
|
182 |
VLA-UNK-61877630-4
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(cc(c5C1=O)F)Cl |
−8.7
± 0.1
|
6.36
± 0.09
|
183 |
PET-UNK-94036022-14
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)C(=O)C(=C)N(C3=O)c4cncc5c4cccc5)Cl |
−8.7
± 0.2
|
6.4
± 0.1
|
184 |
BRU-THA-73c97d88-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCOc5c4cc(cc5)Cl)C=N3 |
−8.71
± 0.06
|
6.35
± 0.05
|
185 |
VLA-UNK-3a43cd95-3
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CCOc5c4cc(c(c5)F)Cl |
−8.70
± 0.09
|
6.33
± 0.06
|
186 |
PET-UNK-94036022-3
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−8.7
± 0.2
|
6.3
± 0.2
|
187 |
VLA-UCB-34f3ed0c-15
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CN6CCNCC6 |
−8.7
± 0.4
|
6.3
± 0.3
|
188 |
BRU-THA-55eab31a-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCNc5c4cc(cc5)Cl)C=N3 |
−8.68
± 0.08
|
6.32
± 0.06
|
189 |
MAT-POS-c2d406ed-2
|
|
CN1C(=O)N(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−8.7
± 0.3
|
6.3
± 0.2
|
190 |
MAT-POS-2e8b2191-8
|
|
CN1C(=O)N(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)C)c4cncc5c4cccc5 |
−8.6
± 0.1
|
6.29
± 0.10
|
191 |
VLA-UNK-f702bf1c-5
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CC6CCC(=O)NC6 |
−8.6
± 0.2
|
6.3
± 0.1
|
192 |
ALP-POS-ecbed2ba-11
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCOCC6)C#N |
−8.6
± 0.7
|
6.3
± 0.5
|
193 |
EDJ-MED-fed7ac0b-4
|
|
CNC(=O)CN1CC2(C=NN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−8.6
± 0.1
|
6.25
± 0.08
|
194 |
VLA-UNK-f702bf1c-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)Cc6cc[nH]n6 |
−8.6
± 0.2
|
6.2
± 0.1
|
195 |
EDJ-MED-cc48ee33-2
|
|
Cn1c(ccn1)C(=O)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−8.5
± 0.2
|
6.2
± 0.1
|
196 |
EDJ-MED-f9b78f78-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CNS(=O)(=O)c5c4cc(cc5)Cl |
−8.5
± 0.1
|
6.22
± 0.09
|
197 |
EDJ-MED-7587a9ee-1
|
|
CN1C(=O)N(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)C)c4cncc5c4cccc5 |
−8.5
± 0.1
|
6.21
± 0.08
|
198 |
LUO-POS-d1147590-1
|
|
CN1CCC(CC1)Oc2ccc3cncc(c3c2)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−8.5
± 0.8
|
6.2
± 0.6
|
199 |
MAT-POS-b4d6b7fc-7
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4ccc(c5)NS(=O)(=O)C)Cl |
−8.5
± 0.3
|
6.2
± 0.2
|
200 |
VLA-UNK-56836b69-2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(c(c5)Cl)Cl)NC3=O |
−8.44
± 0.09
|
6.15
± 0.06
|