Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
401 |
MAT-POS-c7726e07-6_2
|
|
CNC(=O)C[N@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−4.2
± 0.3
|
402 |
EDJ-MED-8bb691af-6_2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−4.2
± 0.5
|
403 |
PET-UNK-94036022-13_2
|
|
C=C1C(=O)[C@]2(C[N@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
−4.1
± 0.5
|
404 |
EDJ-MED-e78d5f1a-1_1
|
|
c1cc2cncc(c2c(c1)Cl)N3CC[C@@]4(C3)CCOc5c4cc(cc5)Cl |
−4.1
± 0.1
|
405 |
LUO-POS-b4dec3be-1_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cc(cc5)F)Cl |
−4.1
± 0.3
|
406 |
MAT-POS-69786b79-2_1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@@H+](Cc5c4cc(cc5)Cl)CC(=O)NC6CC6 |
−4.1
± 0.2
|
407 |
EDJ-MED-8bb691af-7_2
|
|
CNC(=O)CN1C[C@]2(CCN(C2)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−4.1
± 0.2
|
408 |
EDJ-MED-a6bab6fb-1_2
|
|
Cc1cccc2c1c(cnc2)N3CC[C@@]4(C3)CCOc5c4cc(cc5)Cl |
−4.06
± 0.10
|
409 |
ALP-POS-ecbed2ba-15_2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCCC6)C#N |
−4.0
± 0.5
|
410 |
EDJ-MED-159244ea-2_1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3)CCOc5c4cc(cc5)Cl |
−4.0
± 0.1
|
411 |
LUO-POS-8484f2d3-2_2
|
|
C[NH+](C)CCOc1ccc2cncc(c2c1)N3CC[C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−4.0
± 0.7
|
412 |
LUO-POS-868e8996-12_2
|
|
CNC(=O)C[N@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−3.9
± 0.2
|
413 |
MAT-POS-40ad851a-1_5
|
|
C[N@@H+]1CCC[C@@H]1COc2ccc3cncc(c3c2)N4CC[C@@]5(C4=O)C[N@](Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−3.9
± 0.7
|
414 |
MAT-POS-853c0ffa-11_1
|
|
CC(C)(c1ccc2cncc(c2c1)N3CC[C@@]4(C3=O)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)O |
−3.9
± 0.5
|
415 |
MAT-POS-853c0ffa-6_1
|
|
c1cc2c(cc1Cl)[C@@]3(CCN(C3=O)c4cncc5c4c(cc(c5)F)Cl)C[N@@](C2)S(=O)(=O)CC6(CC6)C#N |
−3.9
± 0.5
|
416 |
EDJ-MED-8bb691af-2_3
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−3.9
± 0.4
|
417 |
MAT-POS-853c0ffa-9_1
|
|
C[NH+](C)CCOc1ccc2cncc(c2c1)N3CC[C@@]4(C3=O)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−3.9
± 0.4
|
418 |
LUO-POS-eaf50f21-1_2
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)[NH+]=C3N |
−3.8
± 0.4
|
419 |
EDJ-MED-8bb691af-7_1
|
|
CNC(=O)CN1C[C@]2(CCN(C2)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−3.8
± 0.1
|
420 |
MAT-POS-853c0ffa-8_2
|
|
COC1(CC1)CS(=O)(=O)[N@]2Cc3ccc(cc3[C@]4(C2)CCN(C4=O)c5cncc6c5c(cc(c6)F)Cl)Cl |
−3.8
± 0.4
|
421 |
MAT-POS-69786b79-4_2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@H+](Cc5c4cc(cc5)Cl)CC(=O)NC6(CC6)C#N |
−3.7
± 0.3
|
422 |
EDJ-MED-f3cfbbb5-1_2
|
|
Cc1cccc2c1c(cnc2)N3CC[C@@]4(C3)COCc5c4cc(cc5)Cl |
−3.71
± 0.10
|
423 |
MAT-POS-983b399a-2_1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3)CCOc5c4cc(cc5)Cl |
−3.71
± 0.09
|
424 |
MAT-POS-b4d6b7fc-6_2
|
|
CNC(=O)C[N@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4c(ccc5)Cl)Cl |
−3.7
± 0.3
|
425 |
MAT-POS-1d5ab790-2_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4c(ccc5)Cl)Cl |
−3.7
± 0.3
|
426 |
EDJ-MED-e78d5f1a-1_2
|
|
c1cc2cncc(c2c(c1)Cl)N3CC[C@@]4(C3)CCOc5c4cc(cc5)Cl |
−3.67
± 0.09
|
427 |
LUO-POS-868e8996-12_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−3.7
± 0.3
|
428 |
MAT-POS-38eb6498-3_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cc(cc5)OCC[NH+](C)C)Cl |
−3.7
± 0.3
|
429 |
EDJ-MED-a12e3a20-1_1
|
|
c1ccc2c(c1)cncc2N3CC(=O)[C@@]4(C3=O)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−3.6
± 0.3
|
430 |
EDJ-MED-8bb691af-2_4
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−3.6
± 0.3
|
431 |
EDJ-MED-8bb691af-2_2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−3.6
± 0.4
|
432 |
MAT-POS-b4d6b7fc-6_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4c(ccc5)Cl)Cl |
−3.6
± 0.3
|
433 |
MAT-POS-983b399a-2_2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3)CCOc5c4cc(cc5)Cl |
−3.55
± 0.09
|
434 |
EDJ-MED-8bb691af-1_4
|
|
CNC(=O)C[N@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3)c4cncc5c4cccc5)Cl |
−3.5
± 0.2
|
435 |
ALP-POS-ecbed2ba-7_1
|
|
CNC(=O)C1(CC1)[N@@H+]2Cc3ccc(cc3[C@]4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−3.5
± 0.2
|
436 |
EDJ-MED-3656d29d-1_3
|
|
Cc1cccc2c1c(cnc2)N3CC[C@@]4(C3)C[N@H+](Cc5c4cc(cc5)Cl)CC(=O)NC |
−3.5
± 0.2
|
437 |
EDJ-MED-8bb691af-1_2
|
|
CNC(=O)C[N@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3)c4cncc5c4cccc5)Cl |
−3.5
± 0.2
|
438 |
EDJ-MED-f3cfbbb5-1_1
|
|
Cc1cccc2c1c(cnc2)N3CC[C@@]4(C3)COCc5c4cc(cc5)Cl |
−3.44
± 0.09
|
439 |
EDJ-MED-159244ea-2_2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3)CCOc5c4cc(cc5)Cl |
−3.4
± 0.1
|
440 |
ALP-POS-ecbed2ba-13_2
|
|
CC(C)(CS(=O)(=O)[N@]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl)C#N |
−3.4
± 0.4
|
441 |
ALP-POS-ecbed2ba-22_2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)CC#N |
−3.3
± 0.4
|
442 |
PET-UNK-94036022-6_1
|
|
C=C1C(=O)[C@]2(C[N@@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
−3.3
± 0.4
|
443 |
EDG-MED-00af8776-1_2
|
|
c1ccc2c(c1)cncc2N3C=[NH+][C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−3.3
± 0.4
|
444 |
EDJ-MED-3656d29d-1_4
|
|
Cc1cccc2c1c(cnc2)N3CC[C@@]4(C3)C[N@H+](Cc5c4cc(cc5)Cl)CC(=O)NC |
−3.2
± 0.2
|
445 |
EDJ-MED-ee81482e-3_3
|
|
C[NH+](C)C[C@@H](COc1ccc2cncc(c2c1)N3CC[C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)O |
−3.1
± 0.8
|
446 |
LUO-POS-b4dec3be-2_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cc(cc5)F)Cl |
−3.1
± 0.3
|
447 |
ALP-POS-ecbed2ba-8_2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCC6)C#N |
−3.1
± 0.6
|
448 |
MAT-POS-1d5ab790-2_2
|
|
CNC(=O)C[N@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4c(ccc5)Cl)Cl |
−3.0
± 0.3
|
449 |
ALP-POS-ecbed2ba-14_1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@@H+](Cc5c4cc(cc5)Cl)CC(=O)NCC#N |
−3.0
± 0.3
|
450 |
MAT-POS-c7726e07-5_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−2.9
± 0.3
|
451 |
EDJ-MED-8bb691af-2_1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−2.9
± 0.3
|
452 |
ALP-POS-ecbed2ba-11_2
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCOCC6)C#N |
−2.9
± 0.5
|
453 |
EDJ-MED-94fddcec-6_1
|
|
C[N@@](c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CCS(=O)(=O)c5c4cc(cc5)Cl)S(=O)(=O)C |
−2.9
± 0.2
|
454 |
ALP-POS-ecbed2ba-10_2
|
|
COC1CN(C1)S(=O)(=O)[N@]2Cc3ccc(cc3[C@]4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−2.8
± 0.8
|
455 |
PET-UNK-94036022-6_2
|
|
C=C1C(=O)[C@]2(C[N@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
−2.8
± 0.5
|
456 |
EDJ-MED-3656d29d-1_1
|
|
Cc1cccc2c1c(cnc2)N3CC[C@@]4(C3)C[N@@H+](Cc5c4cc(cc5)Cl)CC(=O)NC |
−2.8
± 0.2
|
457 |
EDJ-MED-3656d29d-1_2
|
|
Cc1cccc2c1c(cnc2)N3CC[C@@]4(C3)C[N@@H+](Cc5c4cc(cc5)Cl)CC(=O)NC |
−2.8
± 0.2
|
458 |
EDJ-MED-98c0a822-1_2
|
|
CNC(=O)C1(CCC1)[N@]2C[C@]3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6S2(=O)=O)Cl |
−2.8
± 0.4
|
459 |
ALP-POS-ecbed2ba-8_1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCC6)C#N |
−2.5
± 0.6
|
460 |
EDJ-MED-98c0a822-1_1
|
|
CNC(=O)C1(CCC1)[N@@]2C[C@]3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6S2(=O)=O)Cl |
−2.3
± 0.6
|
461 |
PET-UNK-94036022-7_2
|
|
CNC(=O)C[N@H+]1Cc2ccc(cc2[C@]3(C1)C(=O)C(=C)N(C3=O)c4cncc5c4cccc5)Cl |
−2.3
± 0.2
|
462 |
PET-UNK-94036022-7_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)C(=O)C(=C)N(C3=O)c4cncc5c4cccc5)Cl |
−2.3
± 0.4
|
463 |
EDJ-MED-8bb691af-1_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3)c4cncc5c4cccc5)Cl |
−2.0
± 0.2
|
464 |
LUO-POS-ed2cfb03-1_2
|
|
C[NH+]1CCN(CC1)S(=O)(=O)[N@]2Cc3ccc(cc3[C@]4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−2.0
± 0.6
|
465 |
EDJ-MED-8bb691af-1_3
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)CCN(C3)c4cncc5c4cccc5)Cl |
−2.0
± 0.2
|
466 |
PET-UNK-94036022-14_1
|
|
CNC(=O)C[N@@H+]1Cc2ccc(cc2[C@]3(C1)C(=O)C(=C)N(C3=O)c4cncc5c4cccc5)Cl |
−1.7
± 0.4
|
467 |
ALP-POS-ecbed2ba-5_1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6CS(=O)(=O)C6 |
−1.7
± 0.8
|
468 |
EDG-MED-0c930815-1_2
|
|
c1ccc2c(c1)cncc2N3C=[NH+][C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−1.6
± 0.4
|
469 |
EDJ-MED-976a33d5-3_1
|
|
CNC(=O)C1(CC1)[N@@]2C[C@]3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6S2(=O)=O)Cl |
−1.6
± 0.6
|
470 |
EDG-MED-b6bce001-1_2
|
|
c1ccc2c(c1)cncc2N3C=[NH+][C@@]4(C3=O)C[N@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−1.5
± 0.4
|
471 |
EDG-MED-0c930815-1_1
|
|
c1ccc2c(c1)cncc2N3C=[NH+][C@@]4(C3=O)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−1.4
± 0.4
|
472 |
MAT-POS-853c0ffa-5_1
|
|
c1cc2cncc(c2c(c1)Cl)N3CC[C@@]4(C3=O)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−1.2
± 0.3
|
473 |
LUO-POS-eaf50f21-1_1
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N)[NH+]=C3N |
−1.2
± 0.4
|
474 |
LUO-POS-b5068a05-1_2
|
|
C[NH+](C)NC1=N[C@]2(C[N@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
−1.2
± 0.3
|
475 |
EDJ-MED-fd8ed875-1_1
|
|
CNC(=O)CN1C[C@]2(c3cc(ccc3C1=O)Cl)C(=O)N(C=[NH+]2)c4cncc5c4cccc5 |
−0.8
± 0.2
|
476 |
EDJ-MED-fd8ed875-2_1
|
|
CNC(=O)C1(CC1)N2C[C@]3(c4cc(ccc4C2=O)Cl)C(=O)N(C=[NH+]3)c5cncc6c5cccc6 |
−0.6
± 0.2
|
477 |
EDG-MED-00af8776-1_1
|
|
c1ccc2c(c1)cncc2N3C=[NH+][C@@]4(C3=O)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−0.6
± 0.4
|
478 |
EDJ-MED-976a33d5-3_2
|
|
CNC(=O)C1(CC1)[N@]2C[C@]3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6S2(=O)=O)Cl |
−0.6
± 0.5
|
479 |
EDG-MED-b6bce001-1_1
|
|
c1ccc2c(c1)cncc2N3C=[NH+][C@@]4(C3=O)C[N@@](Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−0.4
± 0.4
|
480 |
PET-UNK-94036022-14_2
|
|
CNC(=O)C[N@H+]1Cc2ccc(cc2[C@]3(C1)C(=O)C(=C)N(C3=O)c4cncc5c4cccc5)Cl |
−0.4
± 0.2
|
481 |
EDG-MED-b6bce001-2_1
|
|
CC1=[NH+][C@]2(C[N@@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
−0.2
± 0.7
|
482 |
LUO-POS-eaf50f21-3_2
|
|
CC(=O)NC1=[NH+][C@]2(C[N@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
−0.2
± 0.5
|
483 |
LUO-POS-eaf50f21-4_1
|
|
CN(C)C1=[NH+][C@]2(C[N@@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
1.1
± 0.4
|
484 |
LUO-POS-b5068a05-1_1
|
|
C[NH+](C)NC1=N[C@]2(C[N@@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
1.2
± 0.5
|
485 |
LUO-POS-eaf50f21-3_1
|
|
CC(=O)NC1=[NH+][C@]2(C[N@@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
1.4
± 0.5
|
486 |
EDG-MED-b6bce001-2_2
|
|
CC1=[NH+][C@]2(C[N@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
1.5
± 0.5
|
487 |
LUO-POS-eaf50f21-4_2
|
|
CN(C)C1=[NH+][C@]2(C[N@](Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)C(=O)N1c5cncc6c5cccc6 |
2.7
± 0.6
|