Rank |
Compound |
SMILES |
ΔG / kcal M-1 |
pIC50 |
101 |
ALP-POS-ecbed2ba-16
|
|
CN(CCC#N)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−7.8
± 0.5
|
5.7
± 0.3
|
102 |
ALP-POS-ecbed2ba-21
|
|
CN(CCOC)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−7.7
± 0.4
|
5.6
± 0.3
|
103 |
MAT-POS-40ad851a-5
|
|
c1cc2cncc(c2cc1OCCCN3CCCC3)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−7.7
± 0.5
|
5.6
± 0.3
|
104 |
ALP-POS-ecbed2ba-1
|
|
CC1(CS(=O)(=O)C1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.7
± 0.5
|
5.6
± 0.4
|
105 |
EDJ-MED-dfa1d800-4
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN6CCC(CC6)(F)F)c7cc(ccc7C2=O)Cl |
−7.7
± 0.3
|
5.6
± 0.2
|
106 |
LUO-POS-d1147590-1
|
|
CN1CCC(CC1)Oc2ccc3cncc(c3c2)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−7.6
± 0.4
|
5.6
± 0.3
|
107 |
MAT-POS-853c0ffa-14
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)F)Cl |
−7.6
± 0.3
|
5.6
± 0.2
|
108 |
LUO-POS-9931618f-1
|
|
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.6
± 0.1
|
5.55
± 0.10
|
109 |
EDG-MED-b1ef7fe3-3
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3ccc(c4)F)c5cc(ccc5C1=O)Cl |
−7.6
± 0.1
|
5.5
± 0.1
|
110 |
EDJ-MED-ee81482e-1
|
|
c1cc2cncc(c2cc1OC3CNC3)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−7.6
± 0.3
|
5.5
± 0.2
|
111 |
LUO-POS-8c3e556a-2
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cc(cc4)Cl)c5cc(ccc5C1=O)Cl |
−7.5
± 0.1
|
5.5
± 0.1
|
112 |
EDJ-MED-976a33d5-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4ccc(c5)S(=O)(=O)C)c6cc(ccc6C2=O)Cl |
−7.5
± 0.2
|
5.5
± 0.1
|
113 |
EDJ-MED-9f4ac58c-2
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.5
± 0.4
|
5.5
± 0.3
|
114 |
EDJ-MED-fd8ed875-6
|
|
CNC(=O)C1(CC1)N2CC3(c4cc(ccc4C2=O)Cl)C(=CN(C3=O)c5cncc6c5cccc6)F |
−7.5
± 0.2
|
5.5
± 0.1
|
115 |
LUO-POS-9931618f-2
|
|
CNC(=O)CN1C[C@@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.5
± 0.2
|
5.5
± 0.1
|
116 |
JOH-MSK-1f2dff76-4
|
|
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CNCc5c4cc(cc5)Cl |
−7.5
± 0.2
|
5.5
± 0.1
|
117 |
EDJ-MED-9f4ac58c-6
|
|
COC1(CC1)CS(=O)(=O)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−7.5
± 0.4
|
5.4
± 0.3
|
118 |
ALP-POS-ecbed2ba-18
|
|
CCN(C)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−7.5
± 0.4
|
5.4
± 0.3
|
119 |
EDJ-MED-ede5c6cb-2
|
|
c1cc2c(cc1NS(=O)(=O)C3CC3)cncc2N4CCC5(C4=O)CCS(=O)(=O)c6c5cc(cc6)Cl |
−7.5
± 0.2
|
5.4
± 0.2
|
120 |
EDJ-MED-b6c6ee2b-6
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)F)c5cc(ccc5C1=O)Cl |
−7.4
± 0.2
|
5.4
± 0.1
|
121 |
MAT-POS-1d5ab790-3
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3c(ccc4)Cl)c5cc(ccc5C1=O)Cl |
−7.4
± 0.1
|
5.4
± 0.1
|
122 |
MAT-POS-50a80394-4
|
|
CC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5 |
−7.4
± 0.2
|
5.4
± 0.2
|
123 |
PET-UNK-aa57768f-9
|
|
C#CCN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.4
± 0.1
|
5.4
± 0.1
|
124 |
EDJ-MED-fed7ac0b-4
|
|
CNC(=O)CN1CC2(C=NN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.4
± 0.1
|
5.4
± 0.1
|
125 |
EDG-MED-b1ef7fe3-2
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)F)c5cc(ccc5C1=O)Cl |
−7.4
± 0.1
|
5.4
± 0.1
|
126 |
EDJ-MED-98c0a822-4
|
|
CNC(=O)C1(COC1)N2CC3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−7.3
± 0.2
|
5.4
± 0.1
|
127 |
EDJ-MED-5cd3920d-2
|
|
c1cc2cncc(c2cc1C(F)F)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.3
± 0.4
|
5.3
± 0.3
|
128 |
EDJ-MED-dfa1d800-1
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN6CCCC6)c7cc(ccc7C2=O)Cl |
−7.3
± 0.3
|
5.3
± 0.2
|
129 |
PET-UNK-aa57768f-3
|
|
C#CCN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.3
± 0.2
|
5.3
± 0.1
|
130 |
BRU-THA-73c97d88-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCOc5c4cc(cc5)Cl)C=N3 |
−7.3
± 0.1
|
5.31
± 0.07
|
131 |
EDG-MED-b1ef7fe3-1
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cc(cc4)Cl)c5cc(ccc5C1=O)Cl |
−7.3
± 0.2
|
5.3
± 0.1
|
132 |
DAR-DIA-0f7b7cd9-8
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCOc5c4cc(cc5)Cl)C(=O)S3 |
−7.2
± 0.1
|
5.27
± 0.08
|
133 |
DAR-DIA-6be260fc-5
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CCNc5c4cc(cc5)Cl |
−7.2
± 0.1
|
5.25
± 0.08
|
134 |
ALP-POS-ecbed2ba-15
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCCC6)C#N |
−7.2
± 0.4
|
5.2
± 0.3
|
135 |
ALP-POS-ecbed2ba-3
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.2
± 0.2
|
5.2
± 0.2
|
136 |
EDJ-MED-fd8ed875-4
|
|
CNC(=O)C1(CC1)N2CC3(C=CN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl |
−7.1
± 0.2
|
5.2
± 0.1
|
137 |
EDG-MED-b1ef7fe3-4
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3ccc(c4)Cl)c5cc(ccc5C1=O)Cl |
−7.1
± 0.2
|
5.2
± 0.1
|
138 |
MAT-POS-983b399a-1
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CCOc5c4cc(cc5)Cl |
−7.1
± 0.1
|
5.19
± 0.08
|
139 |
MAT-POS-50a80394-6
|
|
CC(C)C1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5 |
−7.1
± 0.2
|
5.2
± 0.1
|
140 |
BRU-THA-55eab31a-1
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CCNc5c4cc(cc5)Cl)C=N3 |
−7.1
± 0.1
|
5.15
± 0.10
|
141 |
PET-UNK-aa57768f-8
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(C(=O)c5c4cc(cc5)Cl)CC#N |
−7.0
± 0.1
|
5.13
± 0.08
|
142 |
MAT-POS-40ad851a-2
|
|
CCN(C)CCOc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−7.0
± 0.6
|
5.1
± 0.4
|
143 |
LUO-POS-ed2cfb03-1
|
|
CN1CCN(CC1)S(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.0
± 0.3
|
5.1
± 0.2
|
144 |
EDJ-MED-fd8ed875-5
|
|
CNC(=O)CN1CC2(c3cc(ccc3C1=O)Cl)C(=CN(C2=O)c4cncc5c4cccc5)F |
−7.0
± 0.1
|
5.08
± 0.09
|
145 |
EDJ-MED-8bb691af-8
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−7.0
± 0.2
|
5.1
± 0.1
|
146 |
EDJ-MED-cc48ee33-5
|
|
Cc1cc(n(n1)C)C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−7.0
± 0.2
|
5.1
± 0.2
|
147 |
MAT-POS-50a80394-1
|
|
CC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)S(=O)(=O)CC4(CC4)C#N)c5cncc6c5cccc6 |
−6.9
± 0.2
|
5.0
± 0.2
|
148 |
PET-UNK-7e9559de-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)Cc6nncs6 |
−6.9
± 0.1
|
5.0
± 0.1
|
149 |
ALP-POS-ecbed2ba-6
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−6.9
± 0.3
|
5.0
± 0.2
|
150 |
PET-UNK-94036022-10
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)Cl |
−6.8
± 0.3
|
5.0
± 0.2
|
151 |
MIK-ENA-5d9157e9-2
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−6.8
± 0.4
|
5.0
± 0.3
|
152 |
ALP-POS-477dc5b7-4
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CCOc5c4cc(cc5)Cl |
−6.8
± 0.1
|
4.95
± 0.08
|
153 |
MAT-POS-853c0ffa-21
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)F)Cl |
−6.8
± 0.3
|
4.9
± 0.2
|
154 |
ALP-POS-ecbed2ba-2
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCS(=O)(=O)CC6)C#N |
−6.8
± 0.4
|
4.9
± 0.3
|
155 |
EDJ-MED-468565e0-1
|
|
c1cc2cncc(c2cc1OCCN3CCCC3)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−6.8
± 0.4
|
4.9
± 0.3
|
156 |
MAT-POS-50a80394-5
|
|
CCC1CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5 |
−6.8
± 0.2
|
4.9
± 0.1
|
157 |
EDJ-MED-fd8ed875-3
|
|
CNC(=O)CN1CC2(C=CN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−6.7
± 0.2
|
4.9
± 0.1
|
158 |
MAT-POS-853c0ffa-19
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)OCCN(C)C)Cl |
−6.7
± 0.3
|
4.9
± 0.2
|
159 |
MAT-POS-853c0ffa-12
|
|
CC(C)(c1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)OC)O |
−6.7
± 0.4
|
4.9
± 0.3
|
160 |
LUO-POS-ed2cfb03-2
|
|
CNS(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−6.7
± 0.4
|
4.9
± 0.3
|
161 |
ALP-POS-4483ae88-2
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5S1(=O)=O)Cl |
−6.7
± 0.1
|
4.9
± 0.1
|
162 |
ALP-POS-ecbed2ba-19
|
|
CN(CCO)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−6.6
± 0.4
|
4.8
± 0.3
|
163 |
MAT-POS-38eb6498-3
|
|
CNC(=O)CN1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cc(cc5)OCCN(C)C)Cl |
−6.6
± 0.3
|
4.8
± 0.3
|
164 |
ALP-POS-ecbed2ba-17
|
|
CN(CC#N)S(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−6.6
± 0.2
|
4.8
± 0.1
|
165 |
PET-UNK-94036022-9
|
|
C#CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−6.6
± 0.2
|
4.8
± 0.2
|
166 |
EDJ-MED-fed7ac0b-3
|
|
c1ccc2c(c1)cncc2N3C(=O)C4(CN3)CN(C(=O)c5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−6.6
± 0.4
|
4.8
± 0.3
|
167 |
MAT-POS-853c0ffa-20
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cc(cc6)C(C)(C)O)Cl |
−6.6
± 0.3
|
4.8
± 0.2
|
168 |
PET-UNK-14142a25-10
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl |
−6.5
± 0.2
|
4.8
± 0.1
|
169 |
ALP-POS-ecbed2ba-20
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)N6CCC6 |
−6.5
± 0.7
|
4.8
± 0.5
|
170 |
EDJ-MED-468565e0-5
|
|
c1cc2cncc(c2cc1OCCN3CC(C3)(F)F)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−6.5
± 0.5
|
4.7
± 0.4
|
171 |
MAT-POS-38eb6498-1
|
|
CN(C)CCOc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−6.5
± 0.6
|
4.7
± 0.4
|
172 |
MAT-POS-40ad851a-4
|
|
CN(C)CCCOc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−6.5
± 0.3
|
4.7
± 0.2
|
173 |
EDJ-MED-ee81482e-5
|
|
c1cc2cncc(c2cc1CN3CC4(C3)COC4)N5CCC6(C5=O)CN(Cc7c6cc(cc7)Cl)S(=O)(=O)CC8(CC8)C#N |
−6.5
± 0.4
|
4.7
± 0.3
|
174 |
EDJ-MED-cc48ee33-4
|
|
Cc1cnn(c1C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl)C |
−6.5
± 0.2
|
4.7
± 0.1
|
175 |
MAT-POS-853c0ffa-9
|
|
CN(C)CCOc1ccc2cncc(c2c1)N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−6.5
± 0.7
|
4.7
± 0.5
|
176 |
EDJ-MED-a12e3a20-2
|
|
CNC(=O)CN1CC2(c3cc(ccc3C1=O)Cl)C(=O)CN(C2=O)c4cncc5c4cccc5 |
−6.5
± 0.2
|
4.7
± 0.1
|
177 |
MAT-POS-853c0ffa-1
|
|
CNC(=O)CN1CC2(CCN(C2=O)c3cncc4c3c(ccc4)Cl)c5cc(ccc5C1=O)Cl |
−6.4
± 0.2
|
4.6
± 0.1
|
178 |
MAT-POS-576f7758-1
|
|
CNC(=O)C1(CC1)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−6.3
± 0.2
|
4.6
± 0.1
|
179 |
EDJ-MED-468565e0-4
|
|
c1cc2cncc(c2cc1OCCN3CCC(CC3)(F)F)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−6.3
± 0.6
|
4.6
± 0.5
|
180 |
PET-UNK-7e9559de-1
|
|
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)Cc6nncs6 |
−6.3
± 0.2
|
4.6
± 0.2
|
181 |
LUO-POS-8484f2d3-1
|
|
CN(C)CCOc1ccc2cncc(c2c1)N3CC[C@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N |
−6.3
± 0.6
|
4.6
± 0.4
|
182 |
EDJ-MED-dfa1d800-2
|
|
CNC(=O)C1(CC1)N2CC3(CCN(C3=O)c4cncc5c4cc(cc5)OCCN6CCOCC6)c7cc(ccc7C2=O)Cl |
−6.3
± 0.3
|
4.6
± 0.2
|
183 |
MAT-POS-853c0ffa-22
|
|
CC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5ccc(c6)S(=O)(=O)C)Cl |
−6.3
± 0.3
|
4.6
± 0.2
|
184 |
MAT-POS-be048f2c-7
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)C(=O)c6ccnn6C7CC7 |
−6.3
± 0.2
|
4.6
± 0.2
|
185 |
VLA-UCB-34f3ed0c-15
|
|
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)N(C3=O)CN6CCNCC6 |
−6.2
± 0.3
|
4.5
± 0.2
|
186 |
EDJ-MED-d4864bdc-4
|
|
CN(C)CCOc1ccc2cncc(c2c1)N3CCC4(C3=O)CCS(=O)(=O)c5c4cc(cc5)Cl |
−6.2
± 0.3
|
4.5
± 0.2
|
187 |
MAT-POS-50a80394-7
|
|
CC1(CN(C(=O)C12CN(Cc3c2cc(cc3)Cl)CC(=O)NC)c4cncc5c4cccc5)C |
−6.1
± 0.2
|
4.5
± 0.1
|
188 |
ALP-POS-ecbed2ba-9
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)N6CC(C6)C#N |
−6.1
± 0.4
|
4.5
± 0.3
|
189 |
EDJ-MED-5cd3920d-5
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C(F)F |
−6.1
± 0.4
|
4.4
± 0.3
|
190 |
DAR-DIA-0f7b7cd9-9
|
|
c1ccc2c(c1)cncc2N3CC(=O)C4(C3=O)CCOc5c4cc(cc5)Cl |
−6.1
± 0.1
|
4.44
± 0.09
|
191 |
MAT-POS-69786b79-2
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)CC(=O)NC6CC6 |
−6.1
± 0.3
|
4.4
± 0.2
|
192 |
MAT-POS-853c0ffa-7
|
|
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5c(ccc6)Cl)Cl |
−6.1
± 0.3
|
4.4
± 0.2
|
193 |
EDJ-MED-468565e0-3
|
|
c1cc2cncc(c2cc1OCCN3CCS(=O)(=O)CC3)N4CCC5(C4=O)CN(Cc6c5cc(cc6)Cl)S(=O)(=O)CC7(CC7)C#N |
−6.0
± 0.4
|
4.4
± 0.3
|
194 |
EDJ-MED-159244ea-1
|
|
c1ccc2c(c1)cncc2N3CC[C@]4(C3=O)CCOc5c4cc(cc5)Cl |
−6.0
± 0.1
|
4.4
± 0.1
|
195 |
EDJ-MED-5cd3920d-6
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C(F)(F)F |
−6.0
± 0.4
|
4.4
± 0.3
|
196 |
ALP-POS-ecbed2ba-13
|
|
CC(C)(CS(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl)C#N |
−5.9
± 0.3
|
4.3
± 0.2
|
197 |
EDJ-MED-cc48ee33-3
|
|
Cn1c(ccn1)C(=O)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−5.9
± 0.2
|
4.3
± 0.2
|
198 |
EDJ-MED-7587a9ee-3
|
|
CS(=O)(=O)N1Cc2ccc(cc2C3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl |
−5.9
± 0.2
|
4.3
± 0.1
|
199 |
ALP-POS-ecbed2ba-7
|
|
CNC(=O)C1(CC1)N2Cc3ccc(cc3C4(C2)CCN(C4=O)c5cncc6c5cccc6)Cl |
−5.9
± 0.2
|
4.3
± 0.1
|
200 |
ALP-POS-ecbed2ba-11
|
|
c1ccc2c(c1)cncc2N3CCC4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CCOCC6)C#N |
−5.9
± 0.5
|
4.3
± 0.4
|