Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
601 |
EDJ-MED-6e43a462-9_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c[nH+]c3n2cc(cc3)Cl |
−4.7
± 0.2
|
602 |
EDJ-MED-c8e7a002-14_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c3c(cccn3)[nH]n2 |
−4.7
± 0.1
|
603 |
DAR-DIA-076fb6ea-14_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)C(=O)/C=C/C[NH+]3CCCCC3 |
−4.6
± 0.3
|
604 |
EDJ-MED-6e43a462-1_1
|
|
COc1ccn2c(c1)[nH+]cc2NC(=O)Cc3cccc(c3)Cl |
−4.6
± 0.2
|
605 |
JAN-GHE-83b26c96-2_1
|
|
C[C@@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2NC(=O)C |
−4.6
± 0.1
|
606 |
MAK-UNK-ffc90da7-3_1
|
|
CC(C)OC[C@@H](c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)Cl)[NH2+]C |
−4.6
± 0.2
|
607 |
MIC-UNK-5a93dd5f-3_4
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[N@H+]4CC[C@@H]5CCCC[C@@H]5C4 |
−4.6
± 0.2
|
608 |
ALP-POS-90e38439-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CCNC2=O |
−4.6
± 0.1
|
609 |
ALP-POS-8b8a49e1-7_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CCC(=O)C2 |
−4.6
± 0.2
|
610 |
MAK-UNK-ffc90da7-7_3
|
|
CC(C)OC[C@@H]([C@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3)[NH2+]C |
−4.6
± 0.5
|
611 |
RUB-POS-1325a9ea-19_1
|
|
CC(C)(C)c1ccncc1NC(=O)Cc2cccc(c2)Cl |
−4.5
± 0.1
|
612 |
VLA-UCB-05e51b3f-3_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)C(=O)C[NH+]3CCN(CC3)C(=O)C |
−4.5
± 0.3
|
613 |
MAT-POS-a13804f0-1_2
|
|
Cc1nc2n(n1)C[C@H](CC2)C(=O)N[C@@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−4.50
± 0.09
|
614 |
MIC-UNK-8373f97b-4_5
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@@H]3CCCC[C@H]3NC2=O |
−4.5
± 0.2
|
615 |
ADA-UNI-f8e79267-8_1
|
|
CS(=O)(=O)NCC[C@@H](c1cccc(c1)Cl)C(=O)Nc2cccnc2 |
−4.5
± 0.2
|
616 |
RUB-POS-1325a9ea-16_2
|
|
c1ccc2c(c1)[C@H](CC2=O)NC(=O)Cc3cccc(c3)Cl |
−4.5
± 0.1
|
617 |
EDJ-MED-c8e7a002-12_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cccc3c2[nH]nc3 |
−4.5
± 0.1
|
618 |
JAG-UCB-a3ef7265-15_1
|
|
Cc1nnc(n1C)NC(=O)Cc2cccc(c2)Cl |
−4.5
± 0.1
|
619 |
EDJ-MED-6e43a462-2_1
|
|
COc1ccc2[nH+]cc(n2c1)NC(=O)Cc3cccc(c3)Cl |
−4.5
± 0.2
|
620 |
MIC-UNK-5a93dd5f-3_16
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[N@H+]4CC[C@H]5CCCC[C@H]5C4 |
−4.5
± 0.2
|
621 |
MIC-UNK-8373f97b-4_4
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@H]3CCCC[C@@H]3NC2=O |
−4.4
± 0.2
|
622 |
NAU-LAT-e1818702-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2nncn2C3CC3 |
−4.4
± 0.1
|
623 |
BEN-DND-1e24cf73-1_1
|
|
c1ccc(cc1)n2cncc2NC(=O)Cc3cccc(c3)Cl |
−4.4
± 0.1
|
624 |
MAK-UNK-c749d764-6_2
|
|
C[C@H](C[NH2+]CCCO)[C@@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3 |
−4.4
± 0.3
|
625 |
MAT-POS-a13804f0-1_4
|
|
Cc1nc2n(n1)C[C@H](CC2)C(=O)N[C@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−4.39
± 0.09
|
626 |
JOH-UNI-a38a7bdd-9_2
|
|
Cc1ccncc1N(C[C@H]2C[C@@H]2F)C(=O)Cc3cccc(c3)Cl |
−4.4
± 0.2
|
627 |
JOH-UNI-a38a7bdd-5_1
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@@H]4C[C@@H]4F |
−4.4
± 0.2
|
628 |
JOH-UNI-abfda500-4_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2C(=O)[O-] |
−4.4
± 0.1
|
629 |
EDJ-MED-6e43a462-12_1
|
|
CNc1ccc2[nH+]cc(n2c1)NC(=O)Cc3cccc(c3)Cl |
−4.4
± 0.2
|
630 |
EDJ-MED-6e43a462-8_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c[nH+]c3n2cc(cc3)F |
−4.3
± 0.2
|
631 |
RUB-POS-1325a9ea-7_1
|
|
c1ccc2c(c1)CNC(=O)[C@@H]2NC(=O)Cc3cccc(c3)Cl |
−4.3
± 0.1
|
632 |
JOH-UNI-3fc3434e-6_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](CC#N)c3cccc(c3)Cl |
−4.3
± 0.1
|
633 |
EDJ-MED-ee07cf00-6_1
|
|
Cn1cc(cn1)C2=NO[C@@H](C2)C(=O)N[C@@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−4.31
± 0.09
|
634 |
EDJ-MED-ee07cf00-4_2
|
|
C[C@H](C(=O)N[C@@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3)NC(=O)C4CCC4 |
−4.28
± 0.09
|
635 |
MIC-UNK-8373f97b-5_3
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@H]3CCC[C@@H]3NC2=O |
−4.3
± 0.1
|
636 |
ALP-UNI-44c99a80-1_1
|
|
c1ccc2c(c1)cncc2N(Cc3cnc[nH]3)C(=O)Cc4cccc(c4)Cl |
−4.3
± 0.2
|
637 |
MAT-POS-0bc33984-1_2
|
|
C[C@H]1CCNC(=O)[C@@H]1NC(=O)Cc2cccc(c2)Cl |
−4.26
± 0.08
|
638 |
JOH-UNI-a38a7bdd-6_4
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@H]4C[C@H]4C(F)(F)F |
−4.3
± 0.3
|
639 |
MAK-UNK-f203cb68-22_2
|
|
Cc1ccncc1NC(=O)c2cncc(c2C)NC(=O)[C@H](C)c3cccc(c3)Cl |
−4.2
± 0.2
|
640 |
RUB-POS-1325a9ea-6_1
|
|
c1ccc2c(c1)C[NH2+]C[C@@H]2NC(=O)Cc3cccc(c3)Cl |
−4.2
± 0.3
|
641 |
MAK-UNK-f203cb68-3_1
|
|
Cc1ccncc1NC(=O)C[C@@H](c2cccc(c2)Cl)C(=O)Nc3cnccc3C |
−4.2
± 0.2
|
642 |
RUB-POS-1325a9ea-24_2
|
|
CC1([C@H](c2ccccc2N1)NC(=O)Cc3cccc(c3)Cl)C |
−4.2
± 0.2
|
643 |
ADA-UNI-f8e79267-7_2
|
|
CS(=O)(=O)NCCO[C@H](c1cccc(c1)Cl)C(=O)Nc2cccnc2 |
−4.2
± 0.3
|
644 |
VLA-UCB-05e51b3f-2_2
|
|
Cc1ccncc1NC(=O)[C@H](c2cccc(c2)Cl)[NH+]3CCN(CC3)C(=O)C |
−4.2
± 0.2
|
645 |
MIC-UNK-4c7b8ba7-1_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCCNC2=O |
−4.2
± 0.1
|
646 |
MIC-UNK-8373f97b-4_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@@H]3CCCC[C@@H]3NC2=O |
−4.2
± 0.2
|
647 |
NAU-LAT-a5c7d7cb-3_2
|
|
Cc1ccncc1NC(=O)[C@H](c2cccc(c2)Cl)[NH+]3CCN(CC3)C(=O)C |
−4.1
± 0.2
|
648 |
EDJ-MED-b24713dc-1_1
|
|
Cc1ccn2c(c1)[nH+]cc2NC(=O)Cc3cccc(c3)Cl |
−4.1
± 0.2
|
649 |
EDJ-MED-6e43a462-11_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c[nH+]c3n2CCCC3 |
−4.1
± 0.2
|
650 |
BAR-COM-ebf5acce-1_1
|
|
Cc1ccncc1N(CC2(CC2)O)C(=O)Cc3cccc(c3)Cl |
−4.1
± 0.2
|
651 |
EDJ-MED-c8e7a002-16_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c3cnccc3[nH]n2 |
−4.1
± 0.1
|
652 |
JIN-POS-6dc588a4-8_1
|
|
c1ccc2c(c1)c(no2)NC(=O)Cc3cccc(c3)Cl |
−4.1
± 0.1
|
653 |
RUB-POS-1325a9ea-5_1
|
|
Cc1cccc2c1cncc2NC(=O)Cc3cccc(c3)Cl |
−4.10
± 0.04
|
654 |
ALP-POS-8b8a49e1-6_2
|
|
c1ccc2c(c1)[C@H](CC2=O)NC(=O)Cc3cccc(c3)Cl |
−4.08
± 0.09
|
655 |
JOH-UNI-ee5ed7c8-11_1
|
|
c1ccc2c(c1)cnc(c2NC(=O)Cc3cccc(c3)Cl)CC(F)(F)F |
−4.1
± 0.2
|
656 |
MAK-UNK-f203cb68-22_1
|
|
Cc1ccncc1NC(=O)c2cncc(c2C)NC(=O)[C@@H](C)c3cccc(c3)Cl |
−4.1
± 0.2
|
657 |
MIC-UNK-5a93dd5f-5_3
|
|
CC(=O)N[C@@H]1CC[N@H+](C1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−4.1
± 0.2
|
658 |
BEN-DND-1e24cf73-3_1
|
|
Cc1[nH+]cc(n1c2ccccc2)NC(=O)Cc3cccc(c3)Cl |
−4.1
± 0.2
|
659 |
MAK-UNK-f203cb68-2_1
|
|
C[C@@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2Cc3ccncc3NC(=O)C |
−4.0
± 0.2
|
660 |
MAK-UNK-c749d764-22_1
|
|
C[C@@H](C[NH2+]C[C@@H]1CCCO1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−4.0
± 0.2
|
661 |
JAG-UCB-a3ef7265-4_1
|
|
Cc1nnc(n1C)NC(=O)Cc2cccc(c2F)Cl |
−4.0
± 0.1
|
662 |
MAK-UNK-f203cb68-13_1
|
|
Cc1c(cncc1NC(=O)[C@@H](C)c2cccc(c2)Cl)c3ccncc3NC(=O)C |
−4.0
± 0.2
|
663 |
BAR-COM-0f94fc3d-38_1
|
|
CC[C@@](c1cccc(c1)Cl)(C(=O)Nc2cnccc2C)O |
−4.0
± 0.2
|
664 |
PET-UNK-8df914d1-5_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cncn2C3CC3 |
−3.9
± 0.2
|
665 |
BAR-COM-ebf5acce-13_1
|
|
Cc1ccncc1N(CC2(COC2)C#N)C(=O)Cc3cccc(c3)Cl |
−3.9
± 0.2
|
666 |
JOH-UNI-6fede743-4_1
|
|
c1ccc2c(c1)c[nH]c(=O)c2NC(=O)Cc3cccc(c3)Cl |
−3.9
± 0.1
|
667 |
AGN-NEW-c7b24fe3-5_1
|
|
C#Cc1c(cccn1)NC(=O)Cc2cccc(c2)Cl |
−3.9
± 0.1
|
668 |
MAK-UNK-ffc90da7-7_4
|
|
CC(C)OC[C@H]([C@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3)[NH2+]C |
−3.9
± 0.8
|
669 |
RUB-POS-1325a9ea-7_2
|
|
c1ccc2c(c1)CNC(=O)[C@H]2NC(=O)Cc3cccc(c3)Cl |
−3.9
± 0.1
|
670 |
MAT-POS-0bc33984-1_1
|
|
C[C@@H]1CCNC(=O)[C@@H]1NC(=O)Cc2cccc(c2)Cl |
−3.83
± 0.07
|
671 |
MIC-UNK-5a93dd5f-12_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[N@@]4CC[C@@H](C4)[NH+]5CCCCC5 |
−3.8
± 0.2
|
672 |
BEN-DND-1e24cf73-4_1
|
|
COc1ccccc1n2cncc2NC(=O)Cc3cccc(c3)Cl |
−3.8
± 0.2
|
673 |
MAK-UNK-f203cb68-21_2
|
|
Cc1ccncc1NC(=O)c2cc(c(cn2)NC(=O)[C@H](C)c3cccc(c3)Cl)C |
−3.8
± 0.2
|
674 |
MAT-POS-4211dce8-1_1
|
|
Cn1cc(c2ccccc2c1=O)NC(=O)Cc3cccc(c3)Cl |
−3.8
± 0.1
|
675 |
MIC-UNK-8373f97b-4_7
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@H]3CCCC[C@H]3NC2=O |
−3.7
± 0.2
|
676 |
MIC-UNK-fc94cdb5-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CC(=O)NC2=O |
−3.7
± 0.1
|
677 |
MAK-UNK-f203cb68-20_1
|
|
Cc1ccncc1NC(=O)c2c(c(ccn2)C)NC(=O)[C@@H](C)c3cccc(c3)Cl |
−3.7
± 0.2
|
678 |
ALP-POS-90e38439-1_2
|
|
c1ccc2c(c1)[C@H](C(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−3.7
± 0.1
|
679 |
MAK-UNK-c749d764-22_2
|
|
C[C@H](C[NH2+]C[C@@H]1CCCO1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−3.7
± 0.3
|
680 |
EDJ-MED-c8e7a002-5_1
|
|
Cc1cc(nc2c1c(n[nH]2)NC(=O)Cc3cccc(c3)Cl)C(F)(F)F |
−3.7
± 0.2
|
681 |
EDJ-MED-6e43a462-10_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c[nH+]c3n2cc(cc3)N |
−3.6
± 0.2
|
682 |
RUB-POS-1325a9ea-24_1
|
|
CC1([C@@H](c2ccccc2N1)NC(=O)Cc3cccc(c3)Cl)C |
−3.6
± 0.2
|
683 |
JOH-UNI-50ce7ec3-1_1
|
|
C=CS(=O)(=O)N(c1cncc2c1cccc2)C(=O)Cc3cccc(c3)Cl |
−3.6
± 0.3
|
684 |
NAU-LAT-a5c7d7cb-11_1
|
|
Cn1c2ccccc2c(n1)NC(=O)Cc3cccc(c3)Cl |
−3.6
± 0.1
|
685 |
EDJ-MED-c8e7a002-9_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c3cc(ccc3[nH]n2)F |
−3.6
± 0.1
|
686 |
NAU-LAT-e1818702-9_1
|
|
c1ccc(cc1)Cn2cnnc2NC(=O)Cc3cccc(c3)Cl |
−3.5
± 0.2
|
687 |
VLA-UCB-1dbca3b4-1_2
|
|
c1ccc2c(c1)[C@H](C(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−3.5
± 0.1
|
688 |
JAN-GHE-f4ca5a00-12_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2nncn2C3CC3 |
−3.5
± 0.1
|
689 |
EDJ-MED-ee07cf00-15_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)Cc4ccc(cc4)n5cnnn5 |
−3.43
± 0.09
|
690 |
JOH-UNI-3fc3434e-10_1
|
|
CN(c1c2ccccc2cnc1CC(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−3.4
± 0.2
|
691 |
JOH-UNI-3fc3434e-9_1
|
|
CN(c1c2ccccc2cnc1C#N)C(=O)Cc3cccc(c3)Cl |
−3.4
± 0.2
|
692 |
AGN-NEW-c7b24fe3-1_1
|
|
C=Cc1c(cccn1)NC(=O)Cc2cccc(c2)Cl |
−3.3
± 0.1
|
693 |
AGN-NEW-cce853d0-2_1
|
|
Cc1c(cccn1)NC(=O)Cc2cccc(c2NC(=O)C=C)Cl |
−3.3
± 0.2
|
694 |
MIC-UNK-4c7b8ba7-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CCCNC2=O |
−3.3
± 0.1
|
695 |
BEN-DND-1e24cf73-2_1
|
|
Cc1ccccc1n2cncc2NC(=O)Cc3cccc(c3)Cl |
−3.3
± 0.2
|
696 |
EDJ-MED-b24713dc-4_1
|
|
Cc1cccn2c1[nH+]cc2NC(=O)Cc3cccc(c3)Cl |
−3.3
± 0.2
|
697 |
JOH-UNI-a38a7bdd-8_3
|
|
Cc1ccncc1N(C[C@@H]2C[C@H]2C(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−3.2
± 0.2
|
698 |
MAK-UNK-f203cb68-14_2
|
|
Cc1ccncc1NC(=O)c2c(cccc2Cl)[C@H](C)C(=O)Nc3cnccc3C |
−3.1
± 0.4
|
699 |
JOH-UNI-3fc3434e-11_1
|
|
c1ccc2c(c1)cnc(c2NC(=O)Cc3cccc(c3)Cl)CC(F)(F)F |
−3.0
± 0.2
|
700 |
MAK-UNK-f203cb68-11_2
|
|
Cc1ccnc(c1NC(=O)[C@H](C)c2cccc(c2)Cl)c3ccncc3NC(=O)C |
−2.9
± 0.2
|