Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
501 |
JOH-UNI-6fede743-5_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c3cc(ccc3cnc2C(F)F)F |
−5.5
± 0.2
|
502 |
NAU-LAT-a5c7d7cb-14_2
|
|
c1ccc2c(c1)[C@H](CC(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−5.5
± 0.3
|
503 |
JAN-GHE-83b26c96-6_1
|
|
C[C@@H](c1cccc(c1)Cl)C(=O)Nc2cncnc2C(C)C |
−5.5
± 0.2
|
504 |
MAT-POS-8293a91a-6_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)[C@@H]4CC[C@H](O4)C(=O)N5CCCC5 |
−5.52
± 0.09
|
505 |
NAU-LAT-a5c7d7cb-12_1
|
|
c1ccn2c(c1)nnc2NC(=O)Cc3cccc(c3)Cl |
−5.5
± 0.1
|
506 |
EDJ-MED-ee07cf00-7_1
|
|
Cc1c(c(=O)ccn1CC(=O)N[C@@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4)[O-] |
−5.5
± 0.2
|
507 |
NAU-LAT-a5c7d7cb-6_1
|
|
CC(=O)N1CC[NH+](CC1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cc[nH]c(=O)c3 |
−5.5
± 0.2
|
508 |
MIC-UNK-5a93dd5f-12_6
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[N@@]4CC[C@H](C4)[NH+]5CCCCC5 |
−5.5
± 0.2
|
509 |
EDG-MED-0da5ad92-21_1
|
|
Cc1c(cn[nH]1)NC(=O)Cc2cccc(c2)Cl |
−5.5
± 0.1
|
510 |
JIN-POS-6dc588a4-10_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2nccn3 |
−5.50
± 0.08
|
511 |
EDJ-MED-49816e9b-3_1
|
|
Cc1cnn(c1NC(=O)Cc2cccc(c2)Cl)C |
−5.5
± 0.2
|
512 |
MIC-UNK-d36ab305-4_1
|
|
CN(C)c1ccc(cc1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−5.5
± 0.2
|
513 |
JOH-UNI-a38a7bdd-5_4
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@H]4C[C@H]4F |
−5.5
± 0.2
|
514 |
JOH-UNI-a38a7bdd-6_1
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@@H]4C[C@@H]4C(F)(F)F |
−5.4
± 0.3
|
515 |
EDG-MED-0da5ad92-5_2
|
|
Cc1ccncc1NC(=O)[C@H](CO)c2cccc(c2)Cl |
−5.4
± 0.2
|
516 |
JOH-UNI-3fc3434e-13_1
|
|
CN(c1cncc2c1c(ccc2)CC(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−5.4
± 0.2
|
517 |
VLA-UCB-05e51b3f-17_1
|
|
CC(=O)N(c1cncc2c1cccc2)C(=O)Cc3cccc(c3)Cl |
−5.4
± 0.1
|
518 |
JIN-POS-6dc588a4-12_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2cc[nH]3 |
−5.4
± 0.1
|
519 |
JAN-GHE-83b26c96-1_2
|
|
CC[C@H](c1cccc(c1)Cl)C(=O)Nc2cnncc2C |
−5.4
± 0.2
|
520 |
MIC-UNK-8373f97b-4_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@@H]3CCCC[C@@H]3NC2=O |
−5.4
± 0.2
|
521 |
ALP-POS-3b848b35-4_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](CCC3CCCCC3)c4cccc(c4)Cl |
−5.4
± 0.2
|
522 |
EDJ-MED-ee07cf00-10_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)Cn4cnc(n4)C(F)(F)F |
−5.40
± 0.09
|
523 |
BAR-COM-ebf5acce-5_1
|
|
Cc1ccncc1N(c2c(cn[nH]2)OC)C(=O)Cc3cccc(c3)Cl |
−5.4
± 0.2
|
524 |
MAT-POS-8293a91a-7_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)[C@H]4CC[C@H](O4)C(=O)N5CCCC5 |
−5.38
± 0.09
|
525 |
TRY-UNI-714a760b-18_1
|
|
Cc1ccncc1NC(=O)[C@@H](C)c2cccc(c2)Cl |
−5.38
± 0.08
|
526 |
JAN-GHE-83b26c96-5_1
|
|
Cc1ccncc1NC(=O)[C@@H](C)c2cccc(c2)Cl |
−5.4
± 0.1
|
527 |
EDJ-MED-976da9a6-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2CCCO3 |
−5.4
± 0.1
|
528 |
EDG-MED-0da5ad92-17_1
|
|
Cc1cc(ncc1NC(=O)Cc2cccc(c2)Cl)N |
−5.4
± 0.2
|
529 |
PET-UNK-f92d7c0c-7_1
|
|
CN([C@H]1CCCOC1)C(=O)Cc2cccc(c2)Cl |
−5.4
± 0.2
|
530 |
EDG-MED-0da5ad92-16_1
|
|
Cc1cnncc1NC(=O)Cc2cccc(c2)Cl |
−5.3
± 0.1
|
531 |
BAR-COM-ebf5acce-7_1
|
|
Cc1ccncc1N(CNc2ncco2)C(=O)Cc3cccc(c3)Cl |
−5.3
± 0.2
|
532 |
MAK-UNK-f203cb68-20_2
|
|
Cc1ccncc1NC(=O)c2c(c(ccn2)C)NC(=O)[C@H](C)c3cccc(c3)Cl |
−5.3
± 0.2
|
533 |
JAN-GHE-83b26c96-10_2
|
|
Cc1ccncc1NC(=O)[C@H](c2cccc(c2)Cl)[NH+](C)C |
−5.3
± 0.2
|
534 |
JOH-UNI-ee5ed7c8-8_1
|
|
c1ccc2c(c1)cnc(c2NC(=O)Cc3cccc(c3)Cl)C#N |
−5.3
± 0.1
|
535 |
JOH-UNI-a38a7bdd-7_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)C(=O)[C@@H]3C[C@@H]3C(F)(F)F |
−5.3
± 0.2
|
536 |
PET-UNK-158bee2a-3_1
|
|
Cc1cnsc1NC(=O)Cc2cccc(c2)Cl |
−5.3
± 0.1
|
537 |
MAT-POS-a13804f0-1_1
|
|
Cc1nc2n(n1)C[C@@H](CC2)C(=O)N[C@@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−5.30
± 0.09
|
538 |
EDG-MED-0da5ad92-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cccnc2 |
−5.24
± 0.08
|
539 |
MAK-UNK-f203cb68-9_1
|
|
Cc1ccncc1NC(=O)[C@@](C)(c2cccc(c2)Cl)c3ccncc3NC(=O)C |
−5.2
± 0.2
|
540 |
MIC-UNK-c66144cb-1_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](CCc3cccc(c3)F)c4cccc(c4)Cl |
−5.2
± 0.2
|
541 |
EDJ-MED-ee07cf00-3_1
|
|
Cn1c2c(cn1)c(=O)n(cn2)CC(=O)N[C@@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−5.22
± 0.09
|
542 |
MIC-UNK-42806bd5-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CCNC2=O |
−5.2
± 0.1
|
543 |
MIC-UNK-5a93dd5f-8_2
|
|
C[NH+](C)C1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−5.2
± 0.3
|
544 |
MAT-POS-bb423b95-3_1
|
|
c1ccc(cc1)c2ccncc2NC(=O)Cc3cccc(c3)Cl |
−5.2
± 0.1
|
545 |
JAN-GHE-83b26c96-3_2
|
|
C[C@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2n3cccn3 |
−5.2
± 0.1
|
546 |
JOH-UNI-a38a7bdd-8_4
|
|
Cc1ccncc1N(C[C@H]2C[C@H]2C(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−5.2
± 0.1
|
547 |
MIC-UNK-5a93dd5f-10_2
|
|
CC(=O)N1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−5.2
± 0.2
|
548 |
MIC-UNK-c66144cb-3_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](CCC3CCCCC3)c4cccc(c4)Cl |
−5.2
± 0.2
|
549 |
PET-UNK-f92d7c0c-8_1
|
|
c1ccc2c(c1)COC[C@H]2NC(=O)Cc3cccc(c3)Cl |
−5.2
± 0.2
|
550 |
JOH-UNI-a38a7bdd-8_2
|
|
Cc1ccncc1N(C[C@H]2C[C@@H]2C(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−5.2
± 0.2
|
551 |
ADA-UNI-f8e79267-7_1
|
|
CS(=O)(=O)NCCO[C@@H](c1cccc(c1)Cl)C(=O)Nc2cccnc2 |
−5.2
± 0.3
|
552 |
MIC-UNK-5a93dd5f-1_6
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[NH+]4C[C@@H]5CCC[C@H]5C4 |
−5.2
± 0.2
|
553 |
MAK-UNK-f203cb68-4_1
|
|
Cc1ccncc1NC(=O)Cc2ccncc2NC(=O)[C@@H](C)c3cccc(c3)Cl |
−5.1
± 0.2
|
554 |
VLA-UCB-1dbca3b4-1_1
|
|
c1ccc2c(c1)[C@@H](C(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−5.1
± 0.2
|
555 |
NAU-LAT-e1818702-7_1
|
|
Cn1cnnc1NC(=O)Cc2cccc(c2)Cl |
−5.1
± 0.1
|
556 |
JAG-UCB-a3ef7265-17_1
|
|
Cn1cnnc1NC(=O)Cc2cccc(c2)Cl |
−5.1
± 0.1
|
557 |
NAU-LAT-a5c7d7cb-3_1
|
|
Cc1ccncc1NC(=O)[C@@H](c2cccc(c2)Cl)[NH+]3CCN(CC3)C(=O)C |
−5.1
± 0.2
|
558 |
JOH-UNI-a38a7bdd-9_3
|
|
Cc1ccncc1N(C[C@@H]2C[C@H]2F)C(=O)Cc3cccc(c3)Cl |
−5.1
± 0.1
|
559 |
RUB-POS-1325a9ea-20_2
|
|
c1ccc2c(c1)COC[C@H]2NC(=O)Cc3cccc(c3)Cl |
−5.05
± 0.09
|
560 |
ALP-POS-90e38439-3_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CC(=O)NC2 |
−5.0
± 0.2
|
561 |
EDJ-MED-ee07cf00-4_1
|
|
C[C@@H](C(=O)N[C@@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3)NC(=O)C4CCC4 |
−5.01
± 0.09
|
562 |
ALP-POS-90e38439-2_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCNC2=O |
−5.0
± 0.2
|
563 |
JOH-UNI-6fede743-3_1
|
|
c1ccc2c(c1)c(c[nH]c2=O)NC(=O)Cc3cccc(c3)Cl |
−5.0
± 0.1
|
564 |
EDJ-MED-c8e7a002-6_1
|
|
Cc1c2c([nH]nc2n(n1)C)NC(=O)Cc3cccc(c3)Cl |
−5.0
± 0.2
|
565 |
JOH-UNI-a38a7bdd-6_2
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@H]4C[C@@H]4C(F)(F)F |
−5.0
± 0.3
|
566 |
ALP-POS-8b8a49e1-8_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CCNC(=O)C2 |
−5.0
± 0.3
|
567 |
MIC-UNK-42806bd5-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CC(=O)NC2 |
−5.0
± 0.2
|
568 |
EDJ-MED-cf4b0d25-2_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[NH2+]C[C@@H]4CC[C@@H](O4)C(=O)N5CCCC5 |
−4.99
± 0.10
|
569 |
PET-UNK-ac320b15-4_1
|
|
c1cc(cc(c1)Cl)[C@@H](C(=O)Nc2cccnc2)NC(=O)[C@@H]3CC[C@@H](O3)C(=O)N4CCCC4 |
−5.0
± 0.2
|
570 |
EDJ-MED-49816e9b-5_1
|
|
Cc1c(n(nn1)C)NC(=O)Cc2cccc(c2)Cl |
−5.0
± 0.2
|
571 |
MIC-UNK-c66144cb-2_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](CCc3ccc(cc3)F)c4cccc(c4)Cl |
−5.0
± 0.2
|
572 |
ALP-POS-8b8a49e1-7_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCC(=O)C2 |
−5.0
± 0.2
|
573 |
MIC-UNK-d935700b-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cn[nH]c(=O)c2C3CC3 |
−5.0
± 0.1
|
574 |
RUB-POS-1325a9ea-22_1
|
|
c1ccc2c(c1)C(=[NH+]C2=O)NC(=O)Cc3cccc(c3)Cl |
−5.0
± 0.1
|
575 |
MAK-UNK-ffc90da7-3_2
|
|
CC(C)OC[C@H](c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)Cl)[NH2+]C |
−4.9
± 0.2
|
576 |
MAK-UNK-f203cb68-1_1
|
|
Cc1ccncc1NC(=O)[C@@H](Cc2ccncc2NC(=O)C)c3cccc(c3)Cl |
−4.9
± 0.2
|
577 |
EDJ-MED-ee07cf00-5_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)CNC(=O)c4ccc(cc4)C#N |
−4.91
± 0.09
|
578 |
BRU-CON-67e07230-1_2
|
|
C[C@H](c1cccc(c1)Cl)C(=O)Nc2nncn2C3CC3 |
−4.9
± 0.1
|
579 |
MIC-UNK-8373f97b-5_5
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@@H]3CCC[C@H]3NC2=O |
−4.9
± 0.2
|
580 |
MAK-UNK-c749d764-22_3
|
|
C[C@@H](C[NH2+]C[C@H]1CCCO1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−4.9
± 0.4
|
581 |
DAR-DIA-56cf811e-2_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)C(=O)C#C |
−4.9
± 0.2
|
582 |
RUB-POS-1325a9ea-23_1
|
|
c1ccc2c(c1)[C@@H](C(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−4.8
± 0.2
|
583 |
MIC-UNK-42806bd5-1_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCNC2=O |
−4.8
± 0.2
|
584 |
MIC-UNK-8373f97b-4_6
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@@H]3CCCC[C@H]3NC2=O |
−4.8
± 0.2
|
585 |
BAR-COM-ebf5acce-10_1
|
|
Cc1ccncc1N(CC[C@H](CO)[NH3+])C(=O)Cc2cccc(c2)Cl |
−4.8
± 0.3
|
586 |
EDJ-MED-c8e7a002-15_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c3c(ccnc3Br)[nH]n2 |
−4.8
± 0.2
|
587 |
MAT-POS-0bc33984-1_4
|
|
C[C@H]1CCNC(=O)[C@H]1NC(=O)Cc2cccc(c2)Cl |
−4.80
± 0.08
|
588 |
MAK-UNK-f203cb68-12_2
|
|
Cc1cc(ncc1NC(=O)[C@H](C)c2cccc(c2)Cl)c3ccncc3NC(=O)C |
−4.8
± 0.4
|
589 |
MAT-POS-0bc33984-1_3
|
|
C[C@@H]1CCNC(=O)[C@H]1NC(=O)Cc2cccc(c2)Cl |
−4.76
± 0.08
|
590 |
JAG-UCB-a3ef7265-5_1
|
|
Cc1c(cnn1C)NC(=O)Cc2cccc(c2F)Cl |
−4.8
± 0.1
|
591 |
MIC-UNK-8373f97b-2_2
|
|
c1ccc2c(c1)[C@](C(=O)N2)(CC(=O)N)NC(=O)Cc3cccc(c3)Cl |
−4.7
± 0.3
|
592 |
NAU-LAT-4ce8bf23-2_1
|
|
c1ccc2c(c1)cncc2N(CCC(=O)N)C(=O)Cc3cccc(c3)Cl |
−4.7
± 0.2
|
593 |
VLA-UCB-05e51b3f-2_1
|
|
Cc1ccncc1NC(=O)[C@@H](c2cccc(c2)Cl)[NH+]3CCN(CC3)C(=O)C |
−4.7
± 0.2
|
594 |
MIC-UNK-8373f97b-5_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@@H]3CCC[C@@H]3NC2=O |
−4.7
± 0.1
|
595 |
JIN-POS-6dc588a4-15_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c3c(cccn3)on2 |
−4.7
± 0.1
|
596 |
MAT-POS-0bc33984-2_1
|
|
C[C@@]1(CCNC1=O)NC(=O)Cc2cccc(c2)Cl |
−4.7
± 0.2
|
597 |
BAR-COM-ebf5acce-3_1
|
|
CC[C@H](CN(c1cnccc1C)C(=O)Cc2cccc(c2)Cl)O |
−4.7
± 0.2
|
598 |
BRU-CON-67e07230-1_1
|
|
C[C@@H](c1cccc(c1)Cl)C(=O)Nc2nncn2C3CC3 |
−4.7
± 0.1
|
599 |
MAT-POS-1e5f28a7-1_2
|
|
Cc1ccncc1NC(=O)[C@H](c2cccc(c2)Cl)C(=O)OC |
−4.68
± 0.08
|
600 |
JAN-GHE-83b26c96-9_2
|
|
Cc1ccncc1NC(=O)[C@H](c2cccc(c2)Cl)C(C)C |
−4.7
± 0.2
|