Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
401 |
MIC-UNK-5a93dd5f-7_2
|
|
CC(=O)N(C)[C@H]1CC[N@@H+](C1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−6.0
± 0.2
|
402 |
NIR-THE-590dedc7-1_2
|
|
CC(=O)N1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−6.0
± 0.2
|
403 |
TRY-UNI-714a760b-6_1
|
|
Cc1ccncc1NC(=O)Cc2cccc(c2)Cl |
−6.02
± 0.08
|
404 |
MIC-UNK-5a93dd5f-4_2
|
|
CC(=O)NC1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−6.0
± 0.3
|
405 |
EDJ-MED-c8e7a002-4_1
|
|
Cc1ccn2cnnc2c1NC(=O)Cc3cccc(c3)Cl |
−6.01
± 0.08
|
406 |
MAT-POS-8293a91a-2_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)[C@H]4CC[C@@H](O4)C(=O)N5CCCC5 |
−6.01
± 0.09
|
407 |
JAN-GHE-83b26c96-7_2
|
|
Cc1c(cncn1)NC(=O)[C@H](c2cccc(c2)Cl)C(C)C |
−6.0
± 0.2
|
408 |
SAM-UNK-2684b532-5_1
|
|
C[C@@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2C(F)F |
−6.0
± 0.1
|
409 |
RUB-POS-1325a9ea-20_1
|
|
c1ccc2c(c1)COC[C@@H]2NC(=O)Cc3cccc(c3)Cl |
−6.00
± 0.08
|
410 |
BEN-DND-02317c5c-8_1
|
|
c1ccn2c(c1)nnc2NC(=O)Cc3cccc(c3)Cl |
−6.0
± 0.1
|
411 |
EDJ-MED-976da9a6-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2OCCC3 |
−5.99
± 0.07
|
412 |
EDJ-MED-cf4b0d25-4_1
|
|
CC(=O)N[C@@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3 |
−5.99
± 0.08
|
413 |
MIC-UNK-5a93dd5f-3_15
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](c3cccc(c3)Cl)[N@H+]4CC[C@H]5CCCC[C@H]5C4 |
−6.0
± 0.2
|
414 |
JOH-UNI-3fc3434e-4_1
|
|
C#CC(=O)N1CCOc2c1c(cnc2)NC(=O)Cc3cccc(c3)Cl |
−6.0
± 0.2
|
415 |
NAU-LAT-a5c7d7cb-2_2
|
|
CC(=O)N1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−6.0
± 0.1
|
416 |
ALP-POS-8b8a49e1-8_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCNC(=O)C2 |
−6.0
± 0.3
|
417 |
ADA-UNI-f8e79267-11_2
|
|
C[NH2+]CC[C@H](c1cccc(c1)Cl)C(=O)Nc2cccnc2 |
−6.0
± 0.2
|
418 |
ADA-UCB-6c2cb422-8_1
|
|
COc1ccccc1OC[C@@H](c2cccc(c2)Cl)C(=O)Nc3cc(=O)[nH]c4c3cccc4 |
−6.0
± 0.3
|
419 |
ALP-POS-90e38439-3_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CC(=O)NC2 |
−6.0
± 0.2
|
420 |
JAN-GHE-5a013bed-8_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccn2 |
−6.0
± 0.3
|
421 |
JOH-UNI-ee5ed7c8-9_1
|
|
CN(c1c2ccccc2cnc1C#N)C(=O)Cc3cccc(c3)Cl |
−5.9
± 0.4
|
422 |
JIN-POS-6dc588a4-20_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c[nH+]cc3c2NCCC3 |
−5.95
± 0.09
|
423 |
MIC-UNK-50cce87d-4_1
|
|
COc1cccc2c1c(cnc2)NC(=O)Cc3cccc(c3)Cl |
−5.9
± 0.2
|
424 |
JIN-POS-6dc588a4-24_1
|
|
c1ccc2c(c1)c(cnc2C#N)NC(=O)Cc3cccc(c3)Cl |
−5.92
± 0.08
|
425 |
EDJ-MED-ee07cf00-9_1
|
|
c1ccc(cc1)c2nnn(n2)CC(=O)N[C@@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−5.92
± 0.09
|
426 |
JIN-POS-6dc588a4-4_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2C(F)(F)F |
−5.91
± 0.10
|
427 |
WIL-UNI-2e73223c-4_1
|
|
Cc1ccncc1OCCNC(=O)C(C)(C)c2cccc(c2)Cl |
−5.9
± 0.3
|
428 |
PET-UNK-f92d7c0c-3_1
|
|
CN([C@H]1CCOC1)C(=O)Cc2cccc(c2)Cl |
−5.9
± 0.2
|
429 |
MIC-UNK-8373f97b-5_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@@H]3CCC[C@@H]3NC2=O |
−5.9
± 0.1
|
430 |
EDG-MED-0da5ad92-12_1
|
|
Cc1cc(cnc1)NC(=O)Cc2cccc(c2)Cl |
−5.9
± 0.1
|
431 |
PET-UNK-f92d7c0c-6_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCCOC2 |
−5.9
± 0.1
|
432 |
DAR-DIA-076fb6ea-10_1
|
|
Cc1ccncc1N(C#C[C@@H]2CCC[NH2+]2)C(=O)Cc3cccc(c3)Cl |
−5.9
± 0.2
|
433 |
JOH-UNI-6fede743-1_1
|
|
c1ccc2c(c1)c(cnc2C(F)F)NC(=O)Cc3cccc(c3)Cl |
−5.9
± 0.1
|
434 |
MAK-UNK-ffc90da7-9_7
|
|
C[C@@H]1[C@H](CCO1)SC[C@H](C)c2ccc3c(c2)cncc3NC(=O)Cc4cccc(c4)Cl |
−5.9
± 0.2
|
435 |
MIC-UNK-5a93dd5f-2_3
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](c3cccc(c3)Cl)[NH+]4C[C@H]5CCCC[C@@H]5C4 |
−5.9
± 0.2
|
436 |
MAR-TRE-f6f5f473-93_1
|
|
Cc1ccc(cc1)Cn2c3cccnc3n(c2=O)CCNC(=O)Cc4cccc(c4)Cl |
−5.9
± 0.2
|
437 |
JAN-GHE-83b26c96-10_1
|
|
Cc1ccncc1NC(=O)[C@@H](c2cccc(c2)Cl)[NH+](C)C |
−5.9
± 0.2
|
438 |
ALP-POS-0c2c77e1-1_1
|
|
c1ccc(cc1)c2ccncc2NC(=O)Cc3cccc(c3)Cl |
−5.88
± 0.08
|
439 |
VLA-UNK-411a133b-2_1
|
|
Cn1c(nnn1)NC(=O)Cc2cccc(c2)Cl |
−5.9
± 0.2
|
440 |
MAT-POS-bb423b95-4_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2C3CC3 |
−5.9
± 0.1
|
441 |
JOH-UNI-a38a7bdd-9_1
|
|
Cc1ccncc1N(C[C@@H]2C[C@@H]2F)C(=O)Cc3cccc(c3)Cl |
−5.9
± 0.1
|
442 |
JAN-GHE-5a013bed-7_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2nncs2 |
−5.9
± 0.1
|
443 |
MIC-UNK-8373f97b-4_3
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@H]3CCCC[C@@H]3NC2=O |
−5.9
± 0.1
|
444 |
MIC-UNK-5a93dd5f-3_8
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[N@H+]4CC[C@H]5CCCC[C@@H]5C4 |
−5.9
± 0.2
|
445 |
MIC-UNK-6ab519a7-1_2
|
|
CC(=O)N1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−5.9
± 0.2
|
446 |
PET-UNK-e44ffd04-1_1
|
|
c1ccn2c(c1)nnc2NC(=O)Cc3cccc(c3)Cl |
−5.8
± 0.1
|
447 |
JIN-POS-6dc588a4-6_1
|
|
CC(C)(C)Oc1ccncc1NC(=O)Cc2cccc(c2)Cl |
−5.85
± 0.08
|
448 |
JAN-GHE-83b26c96-1_1
|
|
CC[C@@H](c1cccc(c1)Cl)C(=O)Nc2cnncc2C |
−5.8
± 0.2
|
449 |
DAR-DIA-076fb6ea-1_1
|
|
C=CC(=O)N(c1cncc2c1cccc2)C(=O)Cc3cccc(c3)Cl |
−5.8
± 0.2
|
450 |
JAN-GHE-83b26c96-3_1
|
|
C[C@@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2n3cccn3 |
−5.8
± 0.2
|
451 |
EDG-MED-0da5ad92-5_1
|
|
Cc1ccncc1NC(=O)[C@@H](CO)c2cccc(c2)Cl |
−5.8
± 0.2
|
452 |
ALP-POS-8b8a49e1-5_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CC(=O)NC2 |
−5.8
± 0.2
|
453 |
SAM-UNK-2684b532-7_1
|
|
C[C@@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2Cl |
−5.8
± 0.1
|
454 |
MAT-POS-500ca5bf-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCNC2=O |
−5.8
± 0.2
|
455 |
MAK-UNK-ffc90da7-9_8
|
|
C[C@H]1[C@H](CCO1)SC[C@H](C)c2ccc3c(c2)cncc3NC(=O)Cc4cccc(c4)Cl |
−5.8
± 0.2
|
456 |
ALP-POS-95b75b4d-8_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2Cl |
−5.79
± 0.10
|
457 |
NAU-LAT-e1818702-4_1
|
|
c1cc(cc(c1)Cl)C(C(=O)Nc2nncn2C3CC3)(F)F |
−5.8
± 0.1
|
458 |
PET-UNK-f92d7c0c-9_1
|
|
CN([C@@H]1COCc2c1cccc2)C(=O)Cc3cccc(c3)Cl |
−5.8
± 0.1
|
459 |
MAK-UNK-c749d764-32_1
|
|
c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3CO)Cl |
−5.8
± 0.1
|
460 |
RUB-POS-1325a9ea-9_1
|
|
COc1cccc2c1c(cnc2)NC(=O)Cc3cccc(c3)Cl |
−5.8
± 0.2
|
461 |
EDG-MED-0da5ad92-10_1
|
|
Cc1ccncc1NC(=O)C(C)(C)c2cccc(c2)Cl |
−5.8
± 0.2
|
462 |
PET-UNK-1320d94d-28_1
|
|
CN([C@@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3)C(=O)[C@@H]4C[C@@H](O4)C(=O)N5CCCC5 |
−5.8
± 0.2
|
463 |
JOH-UNI-ee5ed7c8-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2c(ccc3)C(=O)/C=C/C#N |
−5.8
± 0.2
|
464 |
MIC-UNK-42806bd5-2_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CC(=O)NC2 |
−5.7
± 0.2
|
465 |
SAM-UNK-2684b532-6_1
|
|
C[C@@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2C(F)(F)F |
−5.7
± 0.1
|
466 |
JOH-UNI-abfda500-5_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2C(=O)N |
−5.7
± 0.1
|
467 |
MAT-POS-bb423b95-5_1
|
|
CC(C)c1ccncc1NC(=O)Cc2cccc(c2)Cl |
−5.71
± 0.08
|
468 |
MAK-UNK-f203cb68-4_2
|
|
Cc1ccncc1NC(=O)Cc2ccncc2NC(=O)[C@H](C)c3cccc(c3)Cl |
−5.7
± 0.3
|
469 |
JIN-POS-6dc588a4-23_1
|
|
COc1c2ccccc2c(cn1)NC(=O)Cc3cccc(c3)Cl |
−5.7
± 0.1
|
470 |
MIC-UNK-8373f97b-4_8
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@H]3CCCC[C@H]3NC2=O |
−5.7
± 0.2
|
471 |
MIC-UNK-5a93dd5f-6_2
|
|
CC(=O)N(C)C1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−5.7
± 0.2
|
472 |
DAR-DIA-56cf811e-6_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)C(=O)/C=C/C(F)(F)F |
−5.7
± 0.3
|
473 |
MAK-UNK-f203cb68-14_1
|
|
Cc1ccncc1NC(=O)c2c(cccc2Cl)[C@@H](C)C(=O)Nc3cnccc3C |
−5.7
± 0.3
|
474 |
PET-UNK-8df914d1-2_1
|
|
c1ccn2c(c1)[nH+]cc2NC(=O)Cc3cccc(c3)Cl |
−5.67
± 0.09
|
475 |
EDJ-MED-a364e151-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2CCCC3 |
−5.7
± 0.1
|
476 |
MAK-UNK-ffc90da7-9_5
|
|
C[C@@H]1[C@@H](CCO1)SC[C@H](C)c2ccc3c(c2)cncc3NC(=O)Cc4cccc(c4)Cl |
−5.7
± 0.2
|
477 |
ALP-POS-90e38439-1_1
|
|
c1ccc2c(c1)[C@@H](C(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−5.6
± 0.1
|
478 |
DAR-DIA-076fb6ea-5_1
|
|
c1ccc2c(c1)cncc2N(C#CC#N)C(=O)Cc3cccc(c3)Cl |
−5.6
± 0.3
|
479 |
MAK-UNK-ffc90da7-9_1
|
|
C[C@@H]1[C@@H](CCO1)SC[C@@H](C)c2ccc3c(c2)cncc3NC(=O)Cc4cccc(c4)Cl |
−5.6
± 0.2
|
480 |
JAN-GHE-83b26c96-2_2
|
|
C[C@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2NC(=O)C |
−5.6
± 0.2
|
481 |
JOH-UNI-50ce7ec3-2_1
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)S(=O)(=O)F |
−5.6
± 0.3
|
482 |
BEN-DND-1e24cf73-6_1
|
|
COc1cccc(c1)n2cncc2NC(=O)Cc3cccc(c3)Cl |
−5.6
± 0.2
|
483 |
PET-UNK-e274cad4-6_1
|
|
Cn1ccc2c1c(cnc2)NC(=O)Cc3cccc(c3)Cl |
−5.6
± 0.1
|
484 |
MIC-UNK-8373f97b-5_7
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@H]3CCC[C@H]3NC2=O |
−5.6
± 0.2
|
485 |
TRY-UNI-714a760b-15_1
|
|
Cc1c(cncc1NC(=O)[C@@H](C)c2cccc(c2)Cl)N |
−5.6
± 0.1
|
486 |
JOH-UNI-ee5ed7c8-6_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](CC#N)c3cccc(c3)Cl |
−5.6
± 0.1
|
487 |
PET-UNK-8df914d1-4_1
|
|
Cn1cncc1NC(=O)Cc2cccc(c2)Cl |
−5.60
± 0.08
|
488 |
MIC-UNK-8373f97b-5_6
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@@H]3CCC[C@H]3NC2=O |
−5.6
± 0.2
|
489 |
NAU-LAT-a5c7d7cb-6_2
|
|
CC(=O)N1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cc[nH]c(=O)c3 |
−5.6
± 0.2
|
490 |
EDJ-MED-7bb79bc5-1_1
|
|
COc1c(c2n[nH]c(=O)n2cn1)NC(=O)Cc3cccc(c3)Cl |
−5.6
± 0.1
|
491 |
ROB-UNI-daaf9793-2_2
|
|
c1ccc2c(c1)[C@H](CC(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−5.6
± 0.2
|
492 |
BEN-DND-1e24cf73-5_1
|
|
c1ccc(c(c1)n2cncc2NC(=O)Cc3cccc(c3)Cl)F |
−5.6
± 0.2
|
493 |
EDJ-MED-ee07cf00-6_2
|
|
Cn1cc(cn1)C2=NO[C@H](C2)C(=O)N[C@@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−5.57
± 0.09
|
494 |
JOH-UNI-a38a7bdd-5_2
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@H]4C[C@@H]4F |
−5.6
± 0.3
|
495 |
NAU-LAT-e1818702-10_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2nncs2 |
−5.6
± 0.1
|
496 |
JAN-GHE-5a013bed-11_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2n[n-]nn2 |
−5.55
± 0.09
|
497 |
MAK-UNK-f203cb68-1_2
|
|
Cc1ccncc1NC(=O)[C@H](Cc2ccncc2NC(=O)C)c3cccc(c3)Cl |
−5.6
± 0.2
|
498 |
JAG-UCB-a3ef7265-2_1
|
|
Cn1cnnc1NC(=O)Cc2cccc(c2F)Cl |
−5.6
± 0.2
|
499 |
BAR-COM-ebf5acce-12_1
|
|
Cc1ccncc1N(CNc2ccon2)C(=O)Cc3cccc(c3)Cl |
−5.5
± 0.2
|
500 |
JAN-GHE-d851b096-1_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)NC(=O)C=C |
−5.5
± 0.2
|