Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
601 |
RIT-UNK-fa3975ff-1_1
|
|
COc1ccnc(c1)NC(=O)[C@@H](C#N)c2cccc(c2)Cl |
−4.6
± 0.2
|
602 |
VLA-UCB-1dbca3b4-1_2
|
|
c1ccc2c(c1)[C@H](C(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−4.6
± 0.2
|
603 |
BEN-DND-1e24cf73-5_1
|
|
c1ccc(c(c1)n2cncc2NC(=O)Cc3cccc(c3)Cl)F |
−4.6
± 0.2
|
604 |
MAT-POS-0bc33984-1_1
|
|
C[C@@H]1CCNC(=O)[C@@H]1NC(=O)Cc2cccc(c2)Cl |
−4.56
± 0.08
|
605 |
ALP-UNI-44c99a80-4_1
|
|
c1ccc2c(c1)cncc2N(Cc3cnco3)C(=O)Cc4cccc(c4)Cl |
−4.6
± 0.4
|
606 |
MIC-UNK-8373f97b-4_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@@H]3CCCC[C@@H]3NC2=O |
−4.5
± 0.1
|
607 |
ALP-POS-8b8a49e1-7_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CCC(=O)C2 |
−4.5
± 0.2
|
608 |
JAN-GHE-83b26c96-10_1
|
|
Cc1ccncc1NC(=O)[C@@H](c2cccc(c2)Cl)[NH+](C)C |
−4.5
± 0.2
|
609 |
JAG-UCB-a3ef7265-5_1
|
|
Cc1c(cnn1C)NC(=O)Cc2cccc(c2F)Cl |
−4.5
± 0.1
|
610 |
PET-UNK-f92d7c0c-3_1
|
|
CN([C@H]1CCOC1)C(=O)Cc2cccc(c2)Cl |
−4.5
± 0.2
|
611 |
DAR-DIA-076fb6ea-1_1
|
|
C=CC(=O)N(c1cncc2c1cccc2)C(=O)Cc3cccc(c3)Cl |
−4.5
± 0.2
|
612 |
MIC-UNK-8373f97b-4_3
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@H]3CCCC[C@@H]3NC2=O |
−4.5
± 0.1
|
613 |
JOH-UNI-a38a7bdd-5_2
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@H]4C[C@@H]4F |
−4.5
± 0.2
|
614 |
EDJ-MED-ee07cf00-15_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)Cc4ccc(cc4)n5cnnn5 |
−4.49
± 0.09
|
615 |
NAU-LAT-e1818702-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2nncn2C3CC3 |
−4.5
± 0.1
|
616 |
RUB-POS-1325a9ea-5_1
|
|
Cc1cccc2c1cncc2NC(=O)Cc3cccc(c3)Cl |
−4.47
± 0.05
|
617 |
MAK-UNK-ffc90da7-9_4
|
|
C[C@H]1[C@H](CCO1)SC[C@@H](C)c2ccc3c(c2)cncc3NC(=O)Cc4cccc(c4)Cl |
−4.5
± 0.2
|
618 |
EDJ-MED-c8e7a002-5_1
|
|
Cc1cc(nc2c1c(n[nH]2)NC(=O)Cc3cccc(c3)Cl)C(F)(F)F |
−4.5
± 0.2
|
619 |
JOH-UNI-6fede743-4_1
|
|
c1ccc2c(c1)c[nH]c(=O)c2NC(=O)Cc3cccc(c3)Cl |
−4.5
± 0.1
|
620 |
DAR-DIA-56cf811e-6_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)C(=O)/C=C/C(F)(F)F |
−4.5
± 0.2
|
621 |
MIC-UNK-fc94cdb5-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CC(=O)NC2=O |
−4.5
± 0.2
|
622 |
JAG-UCB-a3ef7265-2_1
|
|
Cn1cnnc1NC(=O)Cc2cccc(c2F)Cl |
−4.4
± 0.2
|
623 |
MAK-UNK-f203cb68-5_2
|
|
Cc1ccncc1NC(=O)[C@H](C)c2cccc(c2c3ccncc3NC(=O)C)Cl |
−4.4
± 0.4
|
624 |
JOH-UNI-a38a7bdd-5_1
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@@H]4C[C@@H]4F |
−4.4
± 0.2
|
625 |
JOH-UNI-6fede743-2_1
|
|
c1ccc2c(c1)cnc(c2NC(=O)Cc3cccc(c3)Cl)C(F)F |
−4.4
± 0.2
|
626 |
MIC-UNK-5a93dd5f-4_2
|
|
CC(=O)NC1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−4.4
± 0.3
|
627 |
MIC-UNK-8373f97b-4_6
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@@H]3CCCC[C@H]3NC2=O |
−4.3
± 0.2
|
628 |
BAR-COM-ebf5acce-10_1
|
|
Cc1ccncc1N(CC[C@H](CO)[NH3+])C(=O)Cc2cccc(c2)Cl |
−4.3
± 0.3
|
629 |
MIC-UNK-8373f97b-5_7
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@H]3CCC[C@H]3NC2=O |
−4.3
± 0.1
|
630 |
MAK-UNK-c749d764-6_2
|
|
C[C@H](C[NH2+]CCCO)[C@@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3 |
−4.3
± 0.2
|
631 |
JAN-GHE-d851b096-1_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)NC(=O)C=C |
−4.3
± 0.2
|
632 |
JAN-GHE-83b26c96-1_2
|
|
CC[C@H](c1cccc(c1)Cl)C(=O)Nc2cnncc2C |
−4.3
± 0.2
|
633 |
BRU-CON-67e07230-1_1
|
|
C[C@@H](c1cccc(c1)Cl)C(=O)Nc2nncn2C3CC3 |
−4.3
± 0.1
|
634 |
BAR-COM-0f94fc3d-38_1
|
|
CC[C@@](c1cccc(c1)Cl)(C(=O)Nc2cnccc2C)O |
−4.2
± 0.2
|
635 |
RUB-POS-1325a9ea-22_1
|
|
c1ccc2c(c1)C(=[NH+]C2=O)NC(=O)Cc3cccc(c3)Cl |
−4.2
± 0.2
|
636 |
VLA-UCB-05e51b3f-2_2
|
|
Cc1ccncc1NC(=O)[C@H](c2cccc(c2)Cl)[NH+]3CCN(CC3)C(=O)C |
−4.2
± 0.2
|
637 |
ALP-POS-90e38439-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CCNC2=O |
−4.2
± 0.1
|
638 |
RUB-POS-1325a9ea-7_2
|
|
c1ccc2c(c1)CNC(=O)[C@H]2NC(=O)Cc3cccc(c3)Cl |
−4.2
± 0.1
|
639 |
ALP-UNI-44c99a80-1_1
|
|
c1ccc2c(c1)cncc2N(Cc3cnc[nH]3)C(=O)Cc4cccc(c4)Cl |
−4.2
± 0.2
|
640 |
MAT-POS-4211dce8-1_1
|
|
Cn1cc(c2ccccc2c1=O)NC(=O)Cc3cccc(c3)Cl |
−4.1
± 0.2
|
641 |
MAK-UNK-ffc90da7-7_3
|
|
CC(C)OC[C@@H]([C@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3)[NH2+]C |
−4.1
± 0.6
|
642 |
AGN-NEW-c7b24fe3-1_1
|
|
C=Cc1c(cccn1)NC(=O)Cc2cccc(c2)Cl |
−4.1
± 0.1
|
643 |
JOH-UNI-3fc3434e-10_1
|
|
CN(c1c2ccccc2cnc1CC(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−4.1
± 0.2
|
644 |
ADA-UNI-f8e79267-8_1
|
|
CS(=O)(=O)NCC[C@@H](c1cccc(c1)Cl)C(=O)Nc2cccnc2 |
−4.1
± 0.2
|
645 |
MIC-UNK-67d4a29a-3_1
|
|
Cc1cccc2c1c(cnc2)N(C)C(=O)Cc3cccc(c3)Cl |
−4.0
± 0.2
|
646 |
AGN-NEW-c7b24fe3-4_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cccnc2C#N |
−4.0
± 0.1
|
647 |
EDJ-MED-c8e7a002-14_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c3c(cccn3)[nH]n2 |
−4.0
± 0.1
|
648 |
MIC-UNK-8373f97b-4_4
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@H]3CCCC[C@@H]3NC2=O |
−4.0
± 0.2
|
649 |
JOH-UNI-a38a7bdd-9_2
|
|
Cc1ccncc1N(C[C@H]2C[C@@H]2F)C(=O)Cc3cccc(c3)Cl |
−4.0
± 0.1
|
650 |
MAT-POS-0bc33984-1_4
|
|
C[C@H]1CCNC(=O)[C@H]1NC(=O)Cc2cccc(c2)Cl |
−3.99
± 0.08
|
651 |
RUB-POS-1325a9ea-6_1
|
|
c1ccc2c(c1)C[NH2+]C[C@@H]2NC(=O)Cc3cccc(c3)Cl |
−4.0
± 0.3
|
652 |
PET-UNK-8df914d1-5_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cncn2C3CC3 |
−3.9
± 0.1
|
653 |
DAR-DIA-076fb6ea-14_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)C(=O)/C=C/C[NH+]3CCCCC3 |
−3.9
± 0.3
|
654 |
MAK-UNK-f203cb68-21_2
|
|
Cc1ccncc1NC(=O)c2cc(c(cn2)NC(=O)[C@H](C)c3cccc(c3)Cl)C |
−3.9
± 0.2
|
655 |
EDJ-MED-c8e7a002-9_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c3cc(ccc3[nH]n2)F |
−3.9
± 0.1
|
656 |
MAK-UNK-ffc90da7-4_3
|
|
C[C@@H](C[NH2+]C[C@H]1CCCO1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−3.9
± 0.3
|
657 |
EDJ-MED-ee07cf00-5_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)CNC(=O)c4ccc(cc4)C#N |
−3.86
± 0.09
|
658 |
MIC-UNK-42806bd5-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CCNC2=O |
−3.9
± 0.1
|
659 |
DAR-DIA-076fb6ea-12_1
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)/C=C/C[NH+]4CCCCC4 |
−3.9
± 0.4
|
660 |
NAU-LAT-a5c7d7cb-3_2
|
|
Cc1ccncc1NC(=O)[C@H](c2cccc(c2)Cl)[NH+]3CCN(CC3)C(=O)C |
−3.9
± 0.2
|
661 |
EDJ-MED-6e43a462-12_1
|
|
CNc1ccc2[nH+]cc(n2c1)NC(=O)Cc3cccc(c3)Cl |
−3.8
± 0.2
|
662 |
JAN-GHE-83b26c96-16_1
|
|
CCCN(c1cccnc1)C(=O)Cc2cccc(c2)Cl |
−3.8
± 0.1
|
663 |
JIN-POS-6dc588a4-8_1
|
|
c1ccc2c(c1)c(no2)NC(=O)Cc3cccc(c3)Cl |
−3.8
± 0.1
|
664 |
MAK-UNK-ffc90da7-1_2
|
|
C[C@H](C[NH2+]CCCO)[C@@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3 |
−3.8
± 0.2
|
665 |
RUB-POS-1325a9ea-6_2
|
|
c1ccc2c(c1)C[NH2+]C[C@H]2NC(=O)Cc3cccc(c3)Cl |
−3.8
± 0.3
|
666 |
MIC-UNK-c66144cb-2_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](CCc3ccc(cc3)F)c4cccc(c4)Cl |
−3.8
± 0.2
|
667 |
NAU-LAT-e1818702-9_1
|
|
c1ccc(cc1)Cn2cnnc2NC(=O)Cc3cccc(c3)Cl |
−3.8
± 0.2
|
668 |
BEN-DND-1e24cf73-3_1
|
|
Cc1[nH+]cc(n1c2ccccc2)NC(=O)Cc3cccc(c3)Cl |
−3.7
± 0.2
|
669 |
MIC-UNK-8373f97b-5_5
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@@H]3CCC[C@H]3NC2=O |
−3.7
± 0.2
|
670 |
BAR-COM-ebf5acce-1_1
|
|
Cc1ccncc1N(CC2(CC2)O)C(=O)Cc3cccc(c3)Cl |
−3.7
± 0.2
|
671 |
JAG-UCB-a3ef7265-4_1
|
|
Cc1nnc(n1C)NC(=O)Cc2cccc(c2F)Cl |
−3.7
± 0.1
|
672 |
EDJ-MED-6e43a462-9_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c[nH+]c3n2cc(cc3)Cl |
−3.7
± 0.2
|
673 |
VLA-UCB-05e51b3f-3_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)C(=O)C[NH+]3CCN(CC3)C(=O)C |
−3.6
± 0.4
|
674 |
MIC-UNK-8373f97b-4_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@@H]3CCCC[C@@H]3NC2=O |
−3.5
± 0.2
|
675 |
MIC-UNK-8373f97b-2_2
|
|
c1ccc2c(c1)[C@](C(=O)N2)(CC(=O)N)NC(=O)Cc3cccc(c3)Cl |
−3.5
± 0.3
|
676 |
ALP-POS-8b8a49e1-6_2
|
|
c1ccc2c(c1)[C@H](CC2=O)NC(=O)Cc3cccc(c3)Cl |
−3.49
± 0.08
|
677 |
AGN-NEW-cce853d0-2_1
|
|
Cc1c(cccn1)NC(=O)Cc2cccc(c2NC(=O)C=C)Cl |
−3.4
± 0.2
|
678 |
JAN-GHE-f4ca5a00-12_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2nncn2C3CC3 |
−3.4
± 0.1
|
679 |
JOH-UNI-ee5ed7c8-10_1
|
|
CN(c1c2ccccc2cnc1CC(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−3.4
± 0.2
|
680 |
EDG-MED-0da5ad92-12_1
|
|
Cc1cc(cnc1)NC(=O)Cc2cccc(c2)Cl |
−3.4
± 0.1
|
681 |
MAT-POS-1e5f28a7-1_2
|
|
Cc1ccncc1NC(=O)[C@H](c2cccc(c2)Cl)C(=O)OC |
−3.32
± 0.08
|
682 |
JOH-UNI-50ce7ec3-1_1
|
|
C=CS(=O)(=O)N(c1cncc2c1cccc2)C(=O)Cc3cccc(c3)Cl |
−3.2
± 0.3
|
683 |
JOH-UNI-a38a7bdd-9_4
|
|
Cc1ccncc1N(C[C@H]2C[C@H]2F)C(=O)Cc3cccc(c3)Cl |
−3.2
± 0.1
|
684 |
MIC-UNK-5a93dd5f-12_8
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[N@]4CC[C@H](C4)[NH+]5CCCCC5 |
−3.2
± 0.2
|
685 |
MIC-UNK-4c7b8ba7-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CCCNC2=O |
−3.2
± 0.1
|
686 |
RUB-POS-1325a9ea-23_2
|
|
c1ccc2c(c1)[C@H](C(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−3.1
± 0.1
|
687 |
JAN-GHE-83b26c96-8_1
|
|
CCC[C@@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2C |
−3.13
± 0.08
|
688 |
JOH-UNI-a38a7bdd-8_1
|
|
Cc1ccncc1N(C[C@@H]2C[C@@H]2C(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−3.1
± 0.2
|
689 |
EDJ-MED-b24713dc-1_1
|
|
Cc1ccn2c(c1)[nH+]cc2NC(=O)Cc3cccc(c3)Cl |
−3.1
± 0.2
|
690 |
EDJ-MED-6e43a462-4_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c[nH+]c3n2cccn3 |
−3.1
± 0.2
|
691 |
EDJ-MED-50fe53e8-4_1
|
|
c1ccn2c(c1)c[nH+]c2NC(=O)Cc3cccc(c3)Cl |
−3.1
± 0.1
|
692 |
PET-UNK-bbe8d7ff-2_1
|
|
Cc1ccncc1N(CC#N)C(=O)Cc2cccc(c2)Cl |
−3.0
± 0.2
|
693 |
RUB-POS-1325a9ea-21_1
|
|
c1ccc2c(c1)CS(=O)(=O)C[C@@H]2NC(=O)Cc3cccc(c3)Cl |
−3.0
± 0.3
|
694 |
MIC-UNK-8373f97b-5_8
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@H]3CCC[C@H]3NC2=O |
−3.0
± 0.1
|
695 |
NAU-LAT-a5c7d7cb-11_1
|
|
Cn1c2ccccc2c(n1)NC(=O)Cc3cccc(c3)Cl |
−3.0
± 0.1
|
696 |
BEN-DND-1e24cf73-7_1
|
|
Cc1[nH+]cc(n1c2cccc(c2)OC)NC(=O)Cc3cccc(c3)Cl |
−2.9
± 0.2
|
697 |
BAR-COM-ebf5acce-3_1
|
|
CC[C@H](CN(c1cnccc1C)C(=O)Cc2cccc(c2)Cl)O |
−2.9
± 0.2
|
698 |
EDJ-MED-c8e7a002-16_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c3cnccc3[nH]n2 |
−2.9
± 0.1
|
699 |
BAR-COM-ebf5acce-13_1
|
|
Cc1ccncc1N(CC2(COC2)C#N)C(=O)Cc3cccc(c3)Cl |
−2.8
± 0.2
|
700 |
MIC-UNK-4c7b8ba7-1_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCCNC2=O |
−2.8
± 0.1
|