Rank |
Microstate |
SMILES |
ΔG / kcal M-1 |
501 |
MIC-UNK-8373f97b-4_7
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@H]3CCCC[C@H]3NC2=O |
−5.4
± 0.2
|
502 |
MAK-UNK-ffc90da7-9_8
|
|
C[C@H]1[C@H](CCO1)SC[C@H](C)c2ccc3c(c2)cncc3NC(=O)Cc4cccc(c4)Cl |
−5.4
± 0.2
|
503 |
MAK-UNK-ffc90da7-3_2
|
|
CC(C)OC[C@H](c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)Cl)[NH2+]C |
−5.3
± 0.2
|
504 |
ALP-POS-a9ad2217-2_2
|
|
CN([C@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3)C(=O)[C@@H]4CC[C@@H](O4)C(=O)N5CCCC5 |
−5.3
± 0.2
|
505 |
EDJ-MED-ee07cf00-10_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)Cn4cnc(n4)C(F)(F)F |
−5.34
± 0.09
|
506 |
MIC-UNK-c66144cb-1_1
|
|
c1ccc2c(c1)cncc2NC(=O)[C@@H](CCc3cccc(c3)F)c4cccc(c4)Cl |
−5.3
± 0.2
|
507 |
EDJ-MED-ee07cf00-17_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)Cn4c(=O)c5ccnn5cn4 |
−5.33
± 0.09
|
508 |
BAR-COM-ebf5acce-11_1
|
|
Cc1ccncc1N(C[C@@]2(CCOC2)O)C(=O)Cc3cccc(c3)Cl |
−5.3
± 0.3
|
509 |
JOH-UNI-abfda500-4_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2C(=O)[O-] |
−5.3
± 0.2
|
510 |
RUB-POS-1325a9ea-7_1
|
|
c1ccc2c(c1)CNC(=O)[C@@H]2NC(=O)Cc3cccc(c3)Cl |
−5.3
± 0.1
|
511 |
MAT-POS-a13804f0-1_2
|
|
Cc1nc2n(n1)C[C@H](CC2)C(=O)N[C@@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−5.31
± 0.09
|
512 |
EDJ-MED-6e43a462-1_1
|
|
COc1ccn2c(c1)[nH+]cc2NC(=O)Cc3cccc(c3)Cl |
−5.3
± 0.2
|
513 |
VLA-UCB-1dbca3b4-1_1
|
|
c1ccc2c(c1)[C@@H](C(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−5.3
± 0.2
|
514 |
TRY-UNI-714a760b-18_1
|
|
Cc1ccncc1NC(=O)[C@@H](C)c2cccc(c2)Cl |
−5.28
± 0.08
|
515 |
EDJ-MED-ee07cf00-4_2
|
|
C[C@H](C(=O)N[C@@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3)NC(=O)C4CCC4 |
−5.28
± 0.09
|
516 |
JIN-POS-6dc588a4-19_1
|
|
c1ccc2c(c1)c(c[nH]c2=O)NC(=O)Cc3cccc(c3)Cl |
−5.3
± 0.1
|
517 |
EDJ-MED-ee07cf00-3_1
|
|
Cn1c2c(cn1)c(=O)n(cn2)CC(=O)N[C@@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−5.26
± 0.09
|
518 |
JAG-UCB-a3ef7265-17_1
|
|
Cn1cnnc1NC(=O)Cc2cccc(c2)Cl |
−5.3
± 0.1
|
519 |
EDJ-MED-c8e7a002-6_1
|
|
Cc1c2c([nH]nc2n(n1)C)NC(=O)Cc3cccc(c3)Cl |
−5.3
± 0.2
|
520 |
BEN-DND-1e24cf73-4_1
|
|
COc1ccccc1n2cncc2NC(=O)Cc3cccc(c3)Cl |
−5.2
± 0.2
|
521 |
EDJ-MED-ee07cf00-4_1
|
|
C[C@@H](C(=O)N[C@@H](c1cccc(c1)Cl)C(=O)Nc2cncc3c2cccc3)NC(=O)C4CCC4 |
−5.24
± 0.09
|
522 |
ALP-POS-8b8a49e1-7_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCC(=O)C2 |
−5.2
± 0.2
|
523 |
ALP-POS-95b75b4d-7_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2S(=O)(=O)N |
−5.2
± 0.2
|
524 |
BAR-COM-ebf5acce-15_1
|
|
Cc1ccncc1N(C[C@H](C[NH3+])O)C(=O)Cc2cccc(c2)Cl |
−5.2
± 0.3
|
525 |
MAT-POS-bb423b95-5_1
|
|
CC(C)c1ccncc1NC(=O)Cc2cccc(c2)Cl |
−5.21
± 0.07
|
526 |
MIC-UNK-5a93dd5f-3_4
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[N@H+]4CC[C@@H]5CCCC[C@@H]5C4 |
−5.2
± 0.2
|
527 |
BRU-CON-67e07230-1_2
|
|
C[C@H](c1cccc(c1)Cl)C(=O)Nc2nncn2C3CC3 |
−5.2
± 0.1
|
528 |
JOH-UNI-ee5ed7c8-13_1
|
|
CN(c1cncc2c1c(ccc2)CC(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−5.2
± 0.2
|
529 |
RUB-POS-1325a9ea-20_2
|
|
c1ccc2c(c1)COC[C@H]2NC(=O)Cc3cccc(c3)Cl |
−5.18
± 0.08
|
530 |
PET-UNK-8df914d1-4_1
|
|
Cn1cncc1NC(=O)Cc2cccc(c2)Cl |
−5.17
± 0.08
|
531 |
MAT-POS-3cc264b0-1_1
|
|
c1ccc2c(c1)cnnc2NC(=O)Cc3cccc(c3)Cl |
−5.2
± 0.1
|
532 |
JAN-GHE-5a013bed-8_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccn2 |
−5.2
± 0.3
|
533 |
MIC-UNK-8373f97b-5_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2[C@@H]3CCC[C@@H]3NC2=O |
−5.2
± 0.1
|
534 |
MAR-TRE-f6f5f473-93_1
|
|
Cc1ccc(cc1)Cn2c3cccnc3n(c2=O)CCNC(=O)Cc4cccc(c4)Cl |
−5.2
± 0.3
|
535 |
EDG-MED-0da5ad92-14_1
|
|
Cc1c(cccn1)NC(=O)Cc2cccc(c2)Cl |
−5.1
± 0.1
|
536 |
EDJ-MED-ee07cf00-6_2
|
|
Cn1cc(cn1)C2=NO[C@H](C2)C(=O)N[C@@H](c3cccc(c3)Cl)C(=O)Nc4cncc5c4cccc5 |
−5.14
± 0.09
|
537 |
JOH-UNI-a38a7bdd-6_2
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@H]4C[C@@H]4C(F)(F)F |
−5.1
± 0.2
|
538 |
EDJ-MED-ee07cf00-8_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)Cn4cc(c(=O)[nH]c4=O)C#N |
−5.13
± 0.09
|
539 |
MIC-UNK-8373f97b-2_1
|
|
c1ccc2c(c1)[C@@](C(=O)N2)(CC(=O)N)NC(=O)Cc3cccc(c3)Cl |
−5.1
± 0.3
|
540 |
MAK-UNK-f203cb68-20_2
|
|
Cc1ccncc1NC(=O)c2c(c(ccn2)C)NC(=O)[C@H](C)c3cccc(c3)Cl |
−5.1
± 0.2
|
541 |
JOH-UNI-3fc3434e-13_1
|
|
CN(c1cncc2c1c(ccc2)CC(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−5.1
± 0.2
|
542 |
JOH-UNI-50ce7ec3-3_1
|
|
C=CS(=O)(=O)N(c1cnc(c2c1cccc2)C(F)F)C(=O)Cc3cccc(c3)Cl |
−5.1
± 0.3
|
543 |
MIC-UNK-8373f97b-5_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2[C@@H]3CCC[C@@H]3NC2=O |
−5.1
± 0.2
|
544 |
MIC-UNK-5a93dd5f-3_16
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)[N@H+]4CC[C@H]5CCCC[C@H]5C4 |
−5.1
± 0.2
|
545 |
VLA-UCB-00f2c2b3-7_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cccc3c2cn[nH]3 |
−5.1
± 0.1
|
546 |
NAU-LAT-a5c7d7cb-6_1
|
|
CC(=O)N1CC[NH+](CC1)[C@@H](c2cccc(c2)Cl)C(=O)Nc3cc[nH]c(=O)c3 |
−5.1
± 0.2
|
547 |
EDG-MED-0da5ad92-21_1
|
|
Cc1c(cn[nH]1)NC(=O)Cc2cccc(c2)Cl |
−5.0
± 0.2
|
548 |
ADA-UNI-f8e79267-10_2
|
|
C[NH2+]CCO[C@H](c1cccc(c1)Cl)C(=O)Nc2cccnc2 |
−5.0
± 0.2
|
549 |
JOH-UNI-a38a7bdd-5_4
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@H]4C[C@H]4F |
−5.0
± 0.2
|
550 |
JOH-UNI-a38a7bdd-9_1
|
|
Cc1ccncc1N(C[C@@H]2C[C@@H]2F)C(=O)Cc3cccc(c3)Cl |
−5.0
± 0.1
|
551 |
ALP-POS-90e38439-2_2
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCNC2=O |
−5.0
± 0.2
|
552 |
EDG-MED-0da5ad92-5_1
|
|
Cc1ccncc1NC(=O)[C@@H](CO)c2cccc(c2)Cl |
−5.0
± 0.2
|
553 |
JOH-UNI-3fc3434e-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2c(ccc3)C(=O)/C=C/C#N |
−5.0
± 0.2
|
554 |
RIT-UNK-fa3975ff-1_2
|
|
COc1ccnc(c1)NC(=O)[C@H](C#N)c2cccc(c2)Cl |
−5.0
± 0.2
|
555 |
PET-UNK-158bee2a-3_1
|
|
Cc1cnsc1NC(=O)Cc2cccc(c2)Cl |
−5.0
± 0.1
|
556 |
JAN-GHE-83b26c96-5_1
|
|
Cc1ccncc1NC(=O)[C@@H](C)c2cccc(c2)Cl |
−5.0
± 0.2
|
557 |
ALP-POS-3fc1724e-8_1
|
|
c1ccc2c(c1)[nH]c(n2)NC(=O)[C@@H](CCC3CCCCC3)c4cccc(c4)Cl |
−5.0
± 0.3
|
558 |
PET-UNK-f92d7c0c-7_1
|
|
CN([C@H]1CCCOC1)C(=O)Cc2cccc(c2)Cl |
−5.0
± 0.1
|
559 |
JOH-UNI-50ce7ec3-2_1
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)S(=O)(=O)F |
−5.0
± 0.3
|
560 |
ADA-UNI-f8e79267-7_2
|
|
CS(=O)(=O)NCCO[C@H](c1cccc(c1)Cl)C(=O)Nc2cccnc2 |
−5.0
± 0.3
|
561 |
MIC-UNK-5a93dd5f-8_2
|
|
C[NH+](C)C1CC[NH+](CC1)[C@H](c2cccc(c2)Cl)C(=O)Nc3cncc4c3cccc4 |
−5.0
± 0.3
|
562 |
VLA-UCB-05e51b3f-16_1
|
|
C=CC(=O)N(c1cncc2c1cccc2)C(=O)Cc3cccc(c3)Cl |
−5.0
± 0.2
|
563 |
EDJ-MED-ee07cf00-16_2
|
|
c1ccc2c(c1)cncc2NC(=O)[C@H](c3cccc(c3)Cl)NC(=O)Cn4cc(c(=O)[nH]c4=O)Cl |
−4.97
± 0.09
|
564 |
MAT-POS-0bc33984-2_2
|
|
C[C@]1(CCNC1=O)NC(=O)Cc2cccc(c2)Cl |
−5.0
± 0.2
|
565 |
DAR-DIA-076fb6ea-6_1
|
|
Cc1ccncc1N(C#CC#N)C(=O)Cc2cccc(c2)Cl |
−5.0
± 0.2
|
566 |
MIC-UNK-d935700b-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cn[nH]c(=O)c2C3CC3 |
−4.9
± 0.1
|
567 |
AGN-NEW-c7b24fe3-5_1
|
|
C#Cc1c(cccn1)NC(=O)Cc2cccc(c2)Cl |
−4.9
± 0.1
|
568 |
ADA-UNI-f8e79267-10_1
|
|
C[NH2+]CCO[C@@H](c1cccc(c1)Cl)C(=O)Nc2cccnc2 |
−4.9
± 0.2
|
569 |
EDG-MED-0da5ad92-13_1
|
|
Cc1ccc(cn1)NC(=O)Cc2cccc(c2)Cl |
−4.9
± 0.1
|
570 |
JAG-UCB-a3ef7265-8_1
|
|
Cc1c(c(n(n1)C)OC)NC(=O)Cc2cccc(c2Cl)Cl |
−4.9
± 0.1
|
571 |
RUB-POS-1325a9ea-21_2
|
|
c1ccc2c(c1)CS(=O)(=O)C[C@H]2NC(=O)Cc3cccc(c3)Cl |
−4.9
± 0.3
|
572 |
RUB-POS-1325a9ea-16_1
|
|
c1ccc2c(c1)[C@@H](CC2=O)NC(=O)Cc3cccc(c3)Cl |
−4.9
± 0.1
|
573 |
SAM-UNK-2684b532-11_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2C(F)F |
−4.9
± 0.1
|
574 |
JAN-GHE-83b26c96-3_2
|
|
C[C@H](c1cccc(c1)Cl)C(=O)Nc2cnccc2n3cccn3 |
−4.9
± 0.1
|
575 |
NAU-LAT-e1818702-4_1
|
|
c1cc(cc(c1)Cl)C(C(=O)Nc2nncn2C3CC3)(F)F |
−4.9
± 0.1
|
576 |
JOH-UNI-a38a7bdd-8_3
|
|
Cc1ccncc1N(C[C@@H]2C[C@H]2C(F)(F)F)C(=O)Cc3cccc(c3)Cl |
−4.9
± 0.3
|
577 |
VLA-UCB-05e51b3f-2_1
|
|
Cc1ccncc1NC(=O)[C@@H](c2cccc(c2)Cl)[NH+]3CCN(CC3)C(=O)C |
−4.9
± 0.2
|
578 |
EDJ-MED-7bb79bc5-1_1
|
|
COc1c(c2n[nH]c(=O)n2cn1)NC(=O)Cc3cccc(c3)Cl |
−4.8
± 0.1
|
579 |
MAK-UNK-f203cb68-14_1
|
|
Cc1ccncc1NC(=O)c2c(cccc2Cl)[C@@H](C)C(=O)Nc3cnccc3C |
−4.8
± 0.3
|
580 |
JOH-UNI-a38a7bdd-7_1
|
|
Cc1ccncc1N(C(=O)Cc2cccc(c2)Cl)C(=O)[C@@H]3C[C@@H]3C(F)(F)F |
−4.8
± 0.2
|
581 |
RUB-POS-1325a9ea-16_2
|
|
c1ccc2c(c1)[C@H](CC2=O)NC(=O)Cc3cccc(c3)Cl |
−4.8
± 0.2
|
582 |
MAK-UNK-ffc90da7-9_5
|
|
C[C@@H]1[C@@H](CCO1)SC[C@H](C)c2ccc3c(c2)cncc3NC(=O)Cc4cccc(c4)Cl |
−4.8
± 0.2
|
583 |
NAU-LAT-a5c7d7cb-13_1
|
|
c1ccc2c(c1)[C@@H](C(=O)N2)NC(=O)Cc3cccc(c3)Cl |
−4.8
± 0.2
|
584 |
MAT-POS-500ca5bf-2_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@H]2CCNC2=O |
−4.8
± 0.2
|
585 |
RUB-POS-1325a9ea-19_1
|
|
CC(C)(C)c1ccncc1NC(=O)Cc2cccc(c2)Cl |
−4.8
± 0.1
|
586 |
MAT-POS-0bc33984-1_3
|
|
C[C@@H]1CCNC(=O)[C@H]1NC(=O)Cc2cccc(c2)Cl |
−4.77
± 0.08
|
587 |
EDJ-MED-c8e7a002-2_1
|
|
COc1ccc2c(c1)c(n[nH]2)NC(=O)Cc3cccc(c3)Cl |
−4.7
± 0.2
|
588 |
ALP-POS-8b8a49e1-5_1
|
|
c1cc(cc(c1)Cl)CC(=O)N[C@@H]2CC(=O)NC2 |
−4.7
± 0.2
|
589 |
JOH-UNI-ee5ed7c8-9_1
|
|
CN(c1c2ccccc2cnc1C#N)C(=O)Cc3cccc(c3)Cl |
−4.7
± 0.2
|
590 |
BAR-COM-ebf5acce-5_1
|
|
Cc1ccncc1N(c2c(cn[nH]2)OC)C(=O)Cc3cccc(c3)Cl |
−4.7
± 0.2
|
591 |
MAT-POS-0bc33984-1_2
|
|
C[C@H]1CCNC(=O)[C@@H]1NC(=O)Cc2cccc(c2)Cl |
−4.69
± 0.08
|
592 |
MAK-UNK-f203cb68-12_2
|
|
Cc1cc(ncc1NC(=O)[C@H](C)c2cccc(c2)Cl)c3ccncc3NC(=O)C |
−4.7
± 0.3
|
593 |
JAN-GHE-83b26c96-10_2
|
|
Cc1ccncc1NC(=O)[C@H](c2cccc(c2)Cl)[NH+](C)C |
−4.7
± 0.2
|
594 |
MAT-POS-0bc33984-2_1
|
|
C[C@@]1(CCNC1=O)NC(=O)Cc2cccc(c2)Cl |
−4.6
± 0.2
|
595 |
NAU-LAT-a5c7d7cb-3_1
|
|
Cc1ccncc1NC(=O)[C@@H](c2cccc(c2)Cl)[NH+]3CCN(CC3)C(=O)C |
−4.6
± 0.3
|
596 |
MAT-POS-bb423b95-3_1
|
|
c1ccc(cc1)c2ccncc2NC(=O)Cc3cccc(c3)Cl |
−4.6
± 0.1
|
597 |
JAG-UCB-a3ef7265-15_1
|
|
Cc1nnc(n1C)NC(=O)Cc2cccc(c2)Cl |
−4.6
± 0.1
|
598 |
MIC-UNK-66895286-1_1
|
|
c1cc(cc(c1)Cl)CC(=O)Nc2c[nH]nc2 |
−4.6
± 0.1
|
599 |
MAK-UNK-f203cb68-22_2
|
|
Cc1ccncc1NC(=O)c2cncc(c2C)NC(=O)[C@H](C)c3cccc(c3)Cl |
−4.6
± 0.2
|
600 |
JOH-UNI-a38a7bdd-6_4
|
|
c1ccc2c(c1)cncc2N(C(=O)Cc3cccc(c3)Cl)C(=O)[C@H]4C[C@H]4C(F)(F)F |
−4.6
± 0.3
|